MX2017011655A - Compuestos de aza-piridona y usos de estos. - Google Patents

Compuestos de aza-piridona y usos de estos.

Info

Publication number
MX2017011655A
MX2017011655A MX2017011655A MX2017011655A MX2017011655A MX 2017011655 A MX2017011655 A MX 2017011655A MX 2017011655 A MX2017011655 A MX 2017011655A MX 2017011655 A MX2017011655 A MX 2017011655A MX 2017011655 A MX2017011655 A MX 2017011655A
Authority
MX
Mexico
Prior art keywords
aza
pyridone compounds
pyridone
infection
disclosed
Prior art date
Application number
MX2017011655A
Other languages
English (en)
Inventor
Leonid Beigelman
David Bernard Smith
Than Hendricks Robert
Dimitrova Stoycheva Antitsa
Original Assignee
Alios Biopharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alios Biopharma Inc filed Critical Alios Biopharma Inc
Publication of MX2017011655A publication Critical patent/MX2017011655A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms

Abstract

En la presente descripción se describen compuestos de aza-piridona, composiciones farmacéuticas que incluyen uno o más compuestos de aza-piridona y métodos para sintetizarlos; además, en la presente descripción se describen métodos para mejorar y/o tratar una enfermedad y/o una afección, incluida una infección por ortomixovirus, con un compuesto de aza-piridona; los ejemplos de una infección viral por ortomixovirus incluyen una infección por influenza.
MX2017011655A 2015-03-11 2016-03-09 Compuestos de aza-piridona y usos de estos. MX2017011655A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562131708P 2015-03-11 2015-03-11
PCT/US2016/021598 WO2016145103A1 (en) 2015-03-11 2016-03-09 Aza-pyridone compounds and uses thereof

Publications (1)

Publication Number Publication Date
MX2017011655A true MX2017011655A (es) 2018-04-30

Family

ID=56879649

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2017011655A MX2017011655A (es) 2015-03-11 2016-03-09 Compuestos de aza-piridona y usos de estos.

Country Status (10)

Country Link
US (1) US10208045B2 (es)
EP (1) EP3268368A4 (es)
CN (1) CN107531717B (es)
AU (1) AU2016229147C1 (es)
CA (1) CA2979216A1 (es)
EA (1) EA036776B1 (es)
HK (1) HK1246780A1 (es)
MX (1) MX2017011655A (es)
TW (1) TWI772256B (es)
WO (1) WO2016145103A1 (es)

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JOP20170169A1 (ar) 2016-08-29 2019-01-30 Novartis Ag مركبات بيريدازين ثلاثية الحلقة مندمجة تفيد في علاج العدوى بفيروس أورثوميكسو
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ES2937837T3 (es) * 2018-09-10 2023-03-31 Cocrystal Pharma Inc Inhibidores de piridopirazina y piridotriazina de la replicación del virus de la gripe

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Also Published As

Publication number Publication date
EA201792008A1 (ru) 2018-05-31
WO2016145103A1 (en) 2016-09-15
AU2016229147C1 (en) 2021-03-25
CA2979216A1 (en) 2016-09-15
EP3268368A1 (en) 2018-01-17
TWI772256B (zh) 2022-08-01
TW201639850A (zh) 2016-11-16
EP3268368A4 (en) 2018-11-14
AU2016229147B2 (en) 2020-10-22
HK1246780A1 (zh) 2018-09-14
AU2016229147A1 (en) 2017-09-28
CN107531717B (zh) 2021-07-27
CN107531717A (zh) 2018-01-02
EA036776B1 (ru) 2020-12-21
US20160264581A1 (en) 2016-09-15
US10208045B2 (en) 2019-02-19

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