MX2009006339A - Compuestos y composiciones como inhibidores de actividad de receptor 1 de cannabinoide. - Google Patents

Compuestos y composiciones como inhibidores de actividad de receptor 1 de cannabinoide.

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Publication number
MX2009006339A
MX2009006339A MX2009006339A MX2009006339A MX2009006339A MX 2009006339 A MX2009006339 A MX 2009006339A MX 2009006339 A MX2009006339 A MX 2009006339A MX 2009006339 A MX2009006339 A MX 2009006339A MX 2009006339 A MX2009006339 A MX 2009006339A
Authority
MX
Mexico
Prior art keywords
compounds
activity
cannabinoid receptor
compositions
inhibitors
Prior art date
Application number
MX2009006339A
Other languages
English (en)
Inventor
Xiaohui He
Kunyong Yang
Hong Liu
Yongping Xie
Xing Wang
Baogen Wu
Dean Phillips
Xuefeng Zhu
Thomas Lau
Truc Ngoc Nguyen
Original Assignee
Irmc Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Irmc Llc filed Critical Irmc Llc
Publication of MX2009006339A publication Critical patent/MX2009006339A/es

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    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/72—Two oxygen atoms, e.g. hydantoin
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    • C07D263/18—Oxygen atoms
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    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
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    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages

Abstract

La invención proporciona compuestos, composiciones farmacéuticas que comprenden tales compuestos y métodos para usar tales compuestos para tratar o prevenir enfermedades o trastornos asociados con la actividad del receptor 1 de cannabinoide (CB1).
MX2009006339A 2006-12-15 2007-12-12 Compuestos y composiciones como inhibidores de actividad de receptor 1 de cannabinoide. MX2009006339A (es)

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PCT/US2007/087230 WO2008076754A2 (en) 2006-12-15 2007-12-12 Compounds and compositions as inhibitors of cannabinoid receptor 1 activity

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AR064353A1 (es) 2009-04-01
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PE20081512A1 (es) 2009-01-04
KR20090092322A (ko) 2009-08-31
EP2121598A2 (en) 2009-11-25
EA017696B1 (ru) 2013-02-28
AU2007333992A1 (en) 2008-06-26
WO2008076754A3 (en) 2008-12-24
JP2010513299A (ja) 2010-04-30
CL2007003629A1 (es) 2008-08-08
TW200831080A (en) 2008-08-01
US20100234365A1 (en) 2010-09-16
AU2007333992B2 (en) 2012-05-17
EA200900828A1 (ru) 2009-12-30
KR101245918B1 (ko) 2013-03-20
JP2013014596A (ja) 2013-01-24
KR20120054106A (ko) 2012-05-29
US8431607B2 (en) 2013-04-30
CA2672271C (en) 2013-01-22
CA2672271A1 (en) 2008-06-26
WO2008076754A2 (en) 2008-06-26

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