MX2007008474A - Sulfonamidas de heteroarilo y ccr2. - Google Patents
Sulfonamidas de heteroarilo y ccr2.Info
- Publication number
- MX2007008474A MX2007008474A MX2007008474A MX2007008474A MX2007008474A MX 2007008474 A MX2007008474 A MX 2007008474A MX 2007008474 A MX2007008474 A MX 2007008474A MX 2007008474 A MX2007008474 A MX 2007008474A MX 2007008474 A MX2007008474 A MX 2007008474A
- Authority
- MX
- Mexico
- Prior art keywords
- ccr2
- compounds
- useful
- antagonists
- heteroaryl sulfonamides
- Prior art date
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- C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
- C07C311/21—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
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- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Se proporcionan compuestos que actuan como antagonistas potentes del receptor CCR2. Las pruebas en animales demuestran que estos compuestos son utiles en el tratamiento de la inflamacion, un trastorno con sello distintivo para el CCR2. Los compuestos generalmente son derivados de la aril-sulfonamida y son utiles en composiciones farmaceuticas, metodos para el tratamiento de trastornos mediados con CCR2, y como controles en ensayos para la identificacion de antagonistas CCR2.
Applications Claiming Priority (4)
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US64410305P | 2005-01-14 | 2005-01-14 | |
US74282105P | 2005-12-06 | 2005-12-06 | |
US75098505P | 2005-12-16 | 2005-12-16 | |
PCT/US2006/001341 WO2006076644A2 (en) | 2005-01-14 | 2006-01-13 | Heteroaryl sulfonamides and ccr2 |
Publications (1)
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MX2007008474A true MX2007008474A (es) | 2008-02-19 |
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MX2007008474A MX2007008474A (es) | 2005-01-14 | 2006-01-13 | Sulfonamidas de heteroarilo y ccr2. |
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US (1) | US20060173019A1 (es) |
EP (3) | EP2474532A1 (es) |
JP (1) | JP5253815B2 (es) |
AT (1) | ATE503741T1 (es) |
AU (1) | AU2006204750C1 (es) |
CA (1) | CA2594726C (es) |
DE (1) | DE602006020979D1 (es) |
DK (2) | DK1838674T3 (es) |
ES (1) | ES2440965T3 (es) |
HK (2) | HK1109404A1 (es) |
IL (1) | IL184539A (es) |
MX (1) | MX2007008474A (es) |
PL (2) | PL2354126T3 (es) |
WO (1) | WO2006076644A2 (es) |
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2006
- 2006-01-13 ES ES11002389.2T patent/ES2440965T3/es active Active
- 2006-01-13 CA CA2594726A patent/CA2594726C/en active Active
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- 2006-01-13 EP EP12162572A patent/EP2474532A1/en not_active Withdrawn
- 2006-01-13 US US11/332,786 patent/US20060173019A1/en not_active Abandoned
- 2006-01-13 EP EP11002389.2A patent/EP2354126B1/en active Active
- 2006-01-13 WO PCT/US2006/001341 patent/WO2006076644A2/en active Application Filing
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- 2006-01-13 MX MX2007008474A patent/MX2007008474A/es active IP Right Grant
- 2006-01-13 JP JP2007551428A patent/JP5253815B2/ja active Active
- 2006-01-13 DK DK06718419.2T patent/DK1838674T3/da active
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Also Published As
Publication number | Publication date |
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DK2354126T3 (da) | 2014-01-13 |
PL2354126T3 (pl) | 2014-03-31 |
EP2474532A1 (en) | 2012-07-11 |
EP1838674B1 (en) | 2011-03-30 |
CA2594726C (en) | 2013-03-19 |
EP1838674A2 (en) | 2007-10-03 |
WO2006076644A3 (en) | 2007-02-15 |
AU2006204750B2 (en) | 2011-09-22 |
EP1838674B9 (en) | 2011-11-02 |
ATE503741T1 (de) | 2011-04-15 |
ES2440965T3 (es) | 2014-01-31 |
AU2006204750A1 (en) | 2006-07-20 |
WO2006076644A2 (en) | 2006-07-20 |
US20060173019A1 (en) | 2006-08-03 |
PL1838674T3 (pl) | 2011-08-31 |
AU2006204750C1 (en) | 2012-11-01 |
JP2008526996A (ja) | 2008-07-24 |
HK1109404A1 (en) | 2008-06-06 |
CA2594726A1 (en) | 2006-07-20 |
HK1160856A1 (en) | 2012-08-17 |
IL184539A (en) | 2016-03-31 |
EP2354126A1 (en) | 2011-08-10 |
DK1838674T3 (da) | 2011-06-14 |
DE602006020979D1 (en) | 2011-05-12 |
EP1838674A4 (en) | 2010-01-06 |
IL184539A0 (en) | 2007-10-31 |
JP5253815B2 (ja) | 2013-07-31 |
EP2354126B1 (en) | 2013-09-25 |
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