ME01184B - Postupak smanjenja alfa, beta nezasićenih ketona u opioidnim kompozicijama - Google Patents

Postupak smanjenja alfa, beta nezasićenih ketona u opioidnim kompozicijama

Info

Publication number
ME01184B
ME01184B MEP-2009-248A MEP24809A ME01184B ME 01184 B ME01184 B ME 01184B ME P24809 A MEP24809 A ME P24809A ME 01184 B ME01184 B ME 01184B
Authority
ME
Montenegro
Prior art keywords
unsaturated ketones
beta unsaturated
reducing alpha
opioid compositions
opioid
Prior art date
Application number
MEP-2009-248A
Other languages
English (en)
French (fr)
Inventor
Robert J Kupper
Original Assignee
Euro Celtique Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Euro Celtique Sa filed Critical Euro Celtique Sa
Publication of ME01184B publication Critical patent/ME01184B/me

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/02—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with oxygen atoms attached in positions 3 and 6, e.g. morphine, morphinone

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
MEP-2009-248A 2005-03-04 2006-02-27 Postupak smanjenja alfa, beta nezasićenih ketona u opioidnim kompozicijama ME01184B (me)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US65879105P 2005-03-04 2005-03-04
EP06707309A EP1861405B1 (en) 2005-03-04 2006-02-27 Method of reducing alpha, beta- unsaturated ketones in opioid compositions
PCT/EP2006/001798 WO2006094672A1 (en) 2005-03-04 2006-02-27 Method of reducing alpha, beta unsaturated ketones in opioid compositions

Publications (1)

Publication Number Publication Date
ME01184B true ME01184B (me) 2013-03-20

Family

ID=36301669

Family Applications (2)

Application Number Title Priority Date Filing Date
MEP-2009-248A ME01184B (me) 2005-03-04 2006-02-27 Postupak smanjenja alfa, beta nezasićenih ketona u opioidnim kompozicijama
MEP-2011-17A ME01594B (me) 2005-03-04 2006-02-27 Postupak smanjenja alfa, beta nezasićenih ketona u opioidnim kompozicijama

Family Applications After (1)

Application Number Title Priority Date Filing Date
MEP-2011-17A ME01594B (me) 2005-03-04 2006-02-27 Postupak smanjenja alfa, beta nezasićenih ketona u opioidnim kompozicijama

Country Status (19)

Country Link
US (1) US7939543B2 (me)
EP (2) EP2112153B1 (me)
JP (1) JP5314894B2 (me)
KR (1) KR100941761B1 (me)
CN (1) CN101133062B (me)
AT (2) ATE487722T1 (me)
CA (1) CA2598774C (me)
CY (2) CY1109262T1 (me)
DE (2) DE602006006558D1 (me)
DK (2) DK2112153T3 (me)
ES (2) ES2355870T3 (me)
HK (2) HK1111695A1 (me)
HR (2) HRP20090387T1 (me)
ME (2) ME01184B (me)
PL (2) PL1861405T3 (me)
PT (2) PT2112153E (me)
RS (2) RS51131B (me)
SI (2) SI1861405T1 (me)
WO (1) WO2006094672A1 (me)

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EP2580218B1 (en) 2010-06-11 2015-02-25 Rhodes Technologies Process for n-dealkylation of tertiary amines
ES2666404T3 (es) 2010-06-11 2018-05-04 Rhodes Technologies Procesos catalizados por metales de transición para la preparación de compuestos de N-alilo y uso de los mismos
CN103179954A (zh) 2010-09-02 2013-06-26 格吕伦塔尔有限公司 包含阴离子聚合物的抗破碎剂型
MX2013002377A (es) 2010-09-02 2013-04-29 Gruenenthal Gmbh Forma de dosificacion resistente a manipulacion que comprende una sal inorganica.
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Also Published As

Publication number Publication date
DK1861405T3 (da) 2009-07-20
CN101133062A (zh) 2008-02-27
RS51131B (sr) 2010-10-31
ES2355870T3 (es) 2011-03-31
DE602006006558D1 (de) 2009-06-10
ATE430153T1 (de) 2009-05-15
HRP20090387T1 (en) 2009-08-31
DK2112153T3 (da) 2011-02-14
HRP20110078T1 (hr) 2011-03-31
JP2008531626A (ja) 2008-08-14
US7939543B2 (en) 2011-05-10
KR20070108931A (ko) 2007-11-13
WO2006094672A1 (en) 2006-09-14
EP2112153A1 (en) 2009-10-28
EP2112153B1 (en) 2010-11-10
PL1861405T3 (pl) 2009-10-30
CN101133062B (zh) 2014-08-06
CA2598774C (en) 2010-12-21
SI1861405T1 (sl) 2009-10-31
EP1861405B1 (en) 2009-04-29
PT2112153E (pt) 2010-12-17
JP5314894B2 (ja) 2013-10-16
RS51568B (en) 2011-08-31
PT1861405E (pt) 2009-07-27
PL2112153T3 (pl) 2011-04-29
HK1111695A1 (en) 2008-08-15
HK1135107A1 (en) 2010-05-28
SI2112153T1 (sl) 2011-02-28
ATE487722T1 (de) 2010-11-15
DE602006018208D1 (de) 2010-12-23
CY1109262T1 (el) 2014-07-02
CY1111241T1 (el) 2015-06-11
CA2598774A1 (en) 2006-09-14
US20080132702A1 (en) 2008-06-05
KR100941761B1 (ko) 2010-02-11
ES2326491T3 (es) 2009-10-13
ME01594B (me) 2014-09-20
EP1861405A1 (en) 2007-12-05

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