ITMI20000050A0 - Procedimento per la preparazione della 5-carbossiftalide - Google Patents
Procedimento per la preparazione della 5-carbossiftalideInfo
- Publication number
- ITMI20000050A0 ITMI20000050A0 IT2000MI000050A ITMI20000050A ITMI20000050A0 IT MI20000050 A0 ITMI20000050 A0 IT MI20000050A0 IT 2000MI000050 A IT2000MI000050 A IT 2000MI000050A IT MI20000050 A ITMI20000050 A IT MI20000050A IT MI20000050 A0 ITMI20000050 A0 IT MI20000050A0
- Authority
- IT
- Italy
- Prior art keywords
- carboxyphtalide
- procedure
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D307/83—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Life Sciences & Earth Sciences (AREA)
- Psychiatry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Furan Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Seasonings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Priority Applications (26)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT2000MI000050A IT1317729B1 (it) | 2000-01-18 | 2000-01-18 | Procedimento per la preparazione della 5-carbossiftalide. |
US09/690,301 US6458973B1 (en) | 2000-01-18 | 2000-10-17 | Process for the preparation of 5-carboxyphthalide |
DK00203602.8T DK1118614T4 (da) | 2000-01-18 | 2000-10-17 | Fremgangsmåde til fremstilling af 5-carboxyphthalid |
ES00203602T ES2178626T5 (es) | 2000-01-18 | 2000-10-17 | Procedimiento para la preparación de 5-carboxiftalida. |
DE60000226T DE60000226T3 (de) | 2000-01-18 | 2000-10-17 | Verfahren zur Herstellung von 5-Carboxyphthalid |
AT00203602T ATE219489T1 (de) | 2000-01-18 | 2000-10-17 | Verfahren zur herstellung von 5-carboxyphthalid |
EP00203602A EP1118614B2 (en) | 2000-01-18 | 2000-10-17 | Process for the preparation of 5-carboxyphthalide |
PT00203602T PT1118614E (pt) | 2000-01-18 | 2000-10-17 | Processo para a preparacao de 5-carboxiftalida |
JP2000372224A JP4558182B2 (ja) | 2000-01-18 | 2000-12-07 | 5−カルボキシフタライドの製造法 |
HU0204187A HUP0204187A3 (en) | 2000-01-18 | 2001-01-17 | Process for the preparation of 1-oxo-1,3-dihydro-5-isobenzofurancarboxylic acid and its use for the production of citalopram |
PCT/EP2001/000617 WO2001053284A1 (en) | 2000-01-18 | 2001-01-17 | Process for the preparation of 5-carboxyphthalide and its use for the production of citalopram |
KR1020027009223A KR100730623B1 (ko) | 2000-01-18 | 2001-01-17 | 5-카복시프탈리드의 제조방법 및 시탈로프람의 생성을위한 그것의 사용 |
CA2397497A CA2397497C (en) | 2000-01-18 | 2001-01-17 | Process for the preparation of 5-carboxyphthalide and its use for the production of citalopram |
CNB018038484A CN1184220C (zh) | 2000-01-18 | 2001-01-17 | 制备5-羧基-2-苯并[c]呋喃酮的方法及其用于生产西酞普兰的用途 |
BR0107853-4A BR0107853A (pt) | 2000-01-18 | 2001-01-17 | Processo para a preparação de 5-carboxiftalida e seu uso para a produção de citalopram |
MXPA02007031A MXPA02007031A (es) | 2000-01-18 | 2001-01-17 | Proceso para la preparacion de 5-carboxiftaluro y su uso para la produccion de citalopram. |
ROA200200989A RO121737B1 (ro) | 2000-01-18 | 2001-01-17 | Procedeu de preparare a 5-carboxiftalidei şi utilizarea sa pentru producerea de citalopram |
PL01356563A PL356563A1 (en) | 2000-01-18 | 2001-01-17 | Process for the preparation of 5-carboxyphthalide and its use for the production of citalopram |
EP01901181A EP1187822A1 (en) | 2000-01-18 | 2001-01-17 | Process for the preparation of 5-carboxphthalide and its use for the production of citalopram |
AU26798/01A AU779581B2 (en) | 2000-01-18 | 2001-01-17 | Process for the preparation of 5-carboxyphthalide and its use for the production of citalopram |
HK02100631.3A HK1042290B (zh) | 2000-01-18 | 2002-01-25 | 製備5-羧基2-苯並呋喃酮的方法 |
ZA200205475A ZA200205475B (en) | 2000-01-18 | 2002-07-09 | Process for the preparation of 5-carboxyphthalide and its use for the production of citalopram. |
BG106925A BG65763B1 (bg) | 2000-01-18 | 2002-07-16 | Метод за получаване на 5-карбоксифталид и неговото използване за получаване на циталопрам |
US10/227,038 US6703516B2 (en) | 2000-01-18 | 2002-08-23 | Process for the preparation of 5-carboxyphthalide |
US10/796,336 US20040171851A1 (en) | 2000-01-18 | 2004-03-08 | Process for the preparation of 5-carboxyphthalide |
US11/975,842 US20080249319A1 (en) | 2000-01-18 | 2007-10-22 | Process for the preparation of 5-Carboxyphthalide |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT2000MI000050A IT1317729B1 (it) | 2000-01-18 | 2000-01-18 | Procedimento per la preparazione della 5-carbossiftalide. |
US09/690,301 US6458973B1 (en) | 2000-01-18 | 2000-10-17 | Process for the preparation of 5-carboxyphthalide |
Publications (3)
Publication Number | Publication Date |
---|---|
ITMI20000050A0 true ITMI20000050A0 (it) | 2000-01-18 |
ITMI20000050A1 ITMI20000050A1 (it) | 2001-07-18 |
IT1317729B1 IT1317729B1 (it) | 2003-07-15 |
Family
ID=26332721
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT2000MI000050A IT1317729B1 (it) | 2000-01-18 | 2000-01-18 | Procedimento per la preparazione della 5-carbossiftalide. |
Country Status (21)
Country | Link |
---|---|
US (4) | US6458973B1 (it) |
EP (2) | EP1118614B2 (it) |
JP (1) | JP4558182B2 (it) |
CN (1) | CN1184220C (it) |
AT (1) | ATE219489T1 (it) |
AU (1) | AU779581B2 (it) |
BG (1) | BG65763B1 (it) |
BR (1) | BR0107853A (it) |
CA (1) | CA2397497C (it) |
DE (1) | DE60000226T3 (it) |
DK (1) | DK1118614T4 (it) |
ES (1) | ES2178626T5 (it) |
HK (1) | HK1042290B (it) |
HU (1) | HUP0204187A3 (it) |
IT (1) | IT1317729B1 (it) |
MX (1) | MXPA02007031A (it) |
PL (1) | PL356563A1 (it) |
PT (1) | PT1118614E (it) |
RO (1) | RO121737B1 (it) |
WO (1) | WO2001053284A1 (it) |
ZA (1) | ZA200205475B (it) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR026063A1 (es) * | 1999-11-01 | 2002-12-26 | Lundbeck & Co As H | Metodo para la preparacion de 5-carboxiftalida. |
NL1017417C1 (nl) | 2000-03-03 | 2001-03-16 | Lundbeck & Co As H | Werkwijze voor de bereiding van Citalopram. |
GB0005477D0 (en) | 2000-03-07 | 2000-04-26 | Resolution Chemicals Limited | Process for the preparation of citalopram |
NZ521204A (en) * | 2000-03-13 | 2004-03-26 | H | Stepwise alkylation of 5-substituted 1-(4-fluorophenyl)- 1,3-dihydroisobenzofurans for preparing citalopram, an anti depressant |
AR032455A1 (es) | 2000-05-12 | 2003-11-12 | Lundbeck & Co As H | Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva |
CN101362743A (zh) | 2003-03-21 | 2009-02-11 | H.隆德贝克有限公司 | 用于制备西酞普兰和依他普仑的中间体 |
TR200504022T1 (tr) * | 2003-03-24 | 2006-08-21 | Hetero Drugs Limited | (S)-sitalopram oksalatın yeni sıvı kristal formları. |
CN100569765C (zh) | 2003-12-19 | 2009-12-16 | 杭州民生药业集团有限公司 | 西酞普兰中间体晶体碱 |
WO2006090409A1 (en) * | 2005-02-28 | 2006-08-31 | Kekule Pharma Ltd., | An improved process for the preparation of 5 - carboxyphthalide |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3607884A (en) * | 1969-03-11 | 1971-09-21 | Mobil Oil Corp | Preparation of 5-carboxyphthalide in liquid sodium trioxide |
US3976751A (en) † | 1974-10-21 | 1976-08-24 | Allied Chemical Corporation | Stabilization of liquid sulfur trioxide |
DE2630927A1 (de) | 1976-07-09 | 1978-01-19 | Basf Ag | Verfahren zur herstellung von phthalidcarbonsaeure-(5) |
DE3605716A1 (de) | 1986-02-22 | 1987-09-03 | Henkel Kgaa | Verwendung von unloeslichen schmutzsammlern zur regenerierung von wasch- und reinigungsloesungen |
ES2148120T3 (es) * | 1997-07-08 | 2002-01-16 | Lundbeck & Co As H | Metodo para la preparacion de citalopram. |
CN1129592C (zh) * | 1998-10-20 | 2003-12-03 | H·隆德贝克有限公司 | 制备西酞普兰的方法 |
AR026063A1 (es) | 1999-11-01 | 2002-12-26 | Lundbeck & Co As H | Metodo para la preparacion de 5-carboxiftalida. |
WO2001032643A1 (en) | 1999-11-01 | 2001-05-10 | H. Lundbeck A/S | Method for the preparation of 5-carboxyphthalide |
GB0005477D0 (en) | 2000-03-07 | 2000-04-26 | Resolution Chemicals Limited | Process for the preparation of citalopram |
-
2000
- 2000-01-18 IT IT2000MI000050A patent/IT1317729B1/it active
- 2000-10-17 DE DE60000226T patent/DE60000226T3/de not_active Expired - Lifetime
- 2000-10-17 AT AT00203602T patent/ATE219489T1/de not_active IP Right Cessation
- 2000-10-17 ES ES00203602T patent/ES2178626T5/es not_active Expired - Lifetime
- 2000-10-17 DK DK00203602.8T patent/DK1118614T4/da active
- 2000-10-17 US US09/690,301 patent/US6458973B1/en not_active Expired - Fee Related
- 2000-10-17 EP EP00203602A patent/EP1118614B2/en not_active Expired - Lifetime
- 2000-10-17 PT PT00203602T patent/PT1118614E/pt unknown
- 2000-12-07 JP JP2000372224A patent/JP4558182B2/ja not_active Expired - Lifetime
-
2001
- 2001-01-17 BR BR0107853-4A patent/BR0107853A/pt not_active Application Discontinuation
- 2001-01-17 RO ROA200200989A patent/RO121737B1/ro unknown
- 2001-01-17 HU HU0204187A patent/HUP0204187A3/hu unknown
- 2001-01-17 WO PCT/EP2001/000617 patent/WO2001053284A1/en active IP Right Grant
- 2001-01-17 CA CA2397497A patent/CA2397497C/en not_active Expired - Fee Related
- 2001-01-17 EP EP01901181A patent/EP1187822A1/en not_active Withdrawn
- 2001-01-17 AU AU26798/01A patent/AU779581B2/en not_active Revoked
- 2001-01-17 MX MXPA02007031A patent/MXPA02007031A/es active IP Right Grant
- 2001-01-17 PL PL01356563A patent/PL356563A1/xx not_active IP Right Cessation
- 2001-01-17 CN CNB018038484A patent/CN1184220C/zh not_active Expired - Lifetime
-
2002
- 2002-01-25 HK HK02100631.3A patent/HK1042290B/zh not_active IP Right Cessation
- 2002-07-09 ZA ZA200205475A patent/ZA200205475B/xx unknown
- 2002-07-16 BG BG106925A patent/BG65763B1/bg unknown
- 2002-08-23 US US10/227,038 patent/US6703516B2/en not_active Expired - Fee Related
-
2004
- 2004-03-08 US US10/796,336 patent/US20040171851A1/en not_active Abandoned
-
2007
- 2007-10-22 US US11/975,842 patent/US20080249319A1/en not_active Abandoned
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CY2007029I1 (el) | Μεθοδος για την παρασκευη υποκατεστημενων οκτανοϋλ-αμιδιων | |
ITMI20010602A0 (it) | Procedimento per la preparazione di talopram puro | |
AR028253A1 (es) | Inhibidores de la glucogeno fosforilasa | |
AR028567A1 (es) | Nuevos derivados de fenil-propargileter | |
FI20011578A0 (fi) | Menetelmä puhtaan sitalopraamin valmistamiseksi | |
AR028596A1 (es) | Nuevos derivados de fenilglicina | |
FI20011621A0 (fi) | Menetelmä sitalopraamin valmistamiseksi | |
ITMI991658A0 (it) | Procedimento per la preparazione di epossidi | |
NO20042667L (no) | Fremgangsmate for fremstilling av escitalopram | |
ITMI20001883A0 (it) | Procedimento integrato per la preparazione di epossidi | |
EE200300294A (et) | Sulfoonamiid-asendatud imidasotriasinoonide valmistamismeetod | |
FI20011889A (fi) | Menetelmä ksylitolin valmistamiseksi | |
ITMI20000050A0 (it) | Procedimento per la preparazione della 5-carbossiftalide | |
NO20025423D0 (no) | FremgangsmÕte for fremstilling av Citalopram | |
ITMI20001869A0 (it) | Procedimento per la preparazione di derivati della baccatina iii | |
ITMI20000681A0 (it) | Procedimento per la preparazione di miscele di metilendianilina e suoi omologhi superiori | |
ITMI981796A0 (it) | Procedimento per la preparazione di r-(-)-carnitina | |
ITMI20021031A1 (it) | Procedimento per preparare policarbonato-polioli | |
ITMI20000334A0 (it) | Procedimento di preparazione di miscele cementizie | |
ITMI20012131A0 (it) | Procedimento per la preparazione di alo-benzonitrili | |
AR028111A1 (es) | Procedimiento para la produccion de isocianatos | |
ITMI20000810A0 (it) | Procedimento per la preparazione di 5'-acetilstavudina | |
ITMI991329A0 (it) | Procedimento per la preparazione di tetrafluoroalogenobenzeni | |
ITMI20001600A1 (it) | Procedimento per la preparazione di 5-amino-4-alo-3-alchil isossazoli. | |
DE60107973D1 (de) | Gewebehandlungszubereitung |