IT1282950B1 - Derivati eterociclo-condensati di morfinoidi - Google Patents
Derivati eterociclo-condensati di morfinoidiInfo
- Publication number
- IT1282950B1 IT1282950B1 ITMI960029A IT1282950B1 IT 1282950 B1 IT1282950 B1 IT 1282950B1 IT MI960029 A ITMI960029 A IT MI960029A IT 1282950 B1 IT1282950 B1 IT 1282950B1
- Authority
- IT
- Italy
- Prior art keywords
- alkyl
- alkoxy
- mcor
- cycloalkylalkyl
- alkenyl
- Prior art date
Links
- 229940127450 Opioid Agonists Drugs 0.000 title 1
- 230000000202 analgesic effect Effects 0.000 title 1
- 239000005557 antagonist Substances 0.000 title 1
- 230000003266 anti-allergic effect Effects 0.000 title 1
- 230000003110 anti-inflammatory effect Effects 0.000 title 1
- 230000001861 immunosuppressant effect Effects 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 11
- 125000003545 alkoxy group Chemical group 0.000 abstract 6
- 125000003342 alkenyl group Chemical group 0.000 abstract 5
- 125000001316 cycloalkyl alkyl group Chemical group 0.000 abstract 5
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 3
- 125000003118 aryl group Chemical group 0.000 abstract 3
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 3
- 125000005843 halogen group Chemical group 0.000 abstract 3
- 125000006570 (C5-C6) heteroaryl group Chemical group 0.000 abstract 2
- 125000003302 alkenyloxy group Chemical group 0.000 abstract 2
- 125000002877 alkyl aryl group Chemical group 0.000 abstract 2
- 125000002947 alkylene group Chemical group 0.000 abstract 2
- 125000005842 heteroatom Chemical group 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 125000002941 2-furyl group Chemical group O1C([*])=C([H])C([H])=C1[H] 0.000 abstract 1
- 125000003682 3-furyl group Chemical group O1C([H])=C([*])C([H])=C1[H] 0.000 abstract 1
- 101100496169 Arabidopsis thaliana CLH1 gene Proteins 0.000 abstract 1
- 101100044057 Mesocricetus auratus SYCP3 gene Proteins 0.000 abstract 1
- JCXJVPUVTGWSNB-UHFFFAOYSA-N Nitrogen dioxide Chemical compound O=[N]=O JCXJVPUVTGWSNB-UHFFFAOYSA-N 0.000 abstract 1
- 101100080600 Schizosaccharomyces pombe (strain 972 / ATCC 24843) nse6 gene Proteins 0.000 abstract 1
- 101150111293 cor-1 gene Proteins 0.000 abstract 1
- 125000001188 haloalkyl group Chemical group 0.000 abstract 1
- 125000001072 heteroaryl group Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 125000006237 oxymethylenoxy group Chemical group [H]C([H])([*:1])[*:2] 0.000 abstract 1
- 125000000951 phenoxy group Chemical group [H]C1=C([H])C([H])=C(O*)C([H])=C1[H] 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
- 125000003107 substituted aryl group Chemical group 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (23)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITMI960029 IT1282950B1 (it) | 1996-01-10 | 1996-01-10 | Derivati eterociclo-condensati di morfinoidi |
| DE69717967T DE69717967T2 (de) | 1996-01-10 | 1997-01-08 | Heterocyclische kondensierte morphin-derivate |
| HU9900974A HUP9900974A3 (en) | 1996-01-10 | 1997-01-08 | Heterocycle-condensed morphinoid derivatives, process for the preparation thereof, their use and pharmaceutical compositions containing them |
| JP9524871A JP2000503019A (ja) | 1996-01-10 | 1997-01-08 | 複素環縮合モルフィノイド誘導体（ｉｉ） |
| NZ326331A NZ326331A (en) | 1996-01-10 | 1997-01-08 | Heterocycle-condensed morphinoid derivatives and medicaments |
| AT97901009T ATE229958T1 (de) | 1996-01-10 | 1997-01-08 | Heterocyclische kondensierte morphin-derivate |
| EP97901009A EP0880526B1 (en) | 1996-01-10 | 1997-01-08 | Heterocycle-condensed morphinoid derivatives (ii) |
| CA002242609A CA2242609A1 (en) | 1996-01-10 | 1997-01-08 | Heterocycle-condensed morphinoid derivatives (ii) |
| AU14410/97A AU706370B2 (en) | 1996-01-10 | 1997-01-08 | Heterocycle-condensed morphinoid derivatives (II) |
| IL12522697A IL125226A0 (en) | 1996-01-10 | 1997-01-08 | Heterocycle-condensed morphinoid derivatives (II) |
| US09/101,213 US6365594B1 (en) | 1996-01-10 | 1997-01-08 | Heterocycle-condensed morphinoid derivatives (II) |
| ARP970100077A AR005423A1 (es) | 1996-01-10 | 1997-01-08 | Derivados morfinoides condensados con heterociclos (ii), su uso como sustancia terapeutica y para preparar medicamentos, composiciones farmaceuticasque los contienen y procedimiento para preparar dichos derivados. |
| BR9707136-6A BR9707136A (pt) | 1996-01-10 | 1997-01-08 | Derivados morfinóides condesados em heterociclo (ii) |
| KR1019980705261A KR19990077125A (ko) | 1996-01-10 | 1997-01-08 | 헤테로고리-축합 모르핀 유도체 (ⅱ) |
| CN97192879A CN1090190C (zh) | 1996-01-10 | 1997-01-08 | 杂环稠合的***类衍生物,制备方法和用途 |
| TR1998/01348T TR199801348T2 (xx) | 1996-01-10 | 1997-01-08 | Heterosikl-kondanse morfinoid t�revleri(II). |
| PCT/EP1997/000120 WO1997025331A1 (en) | 1996-01-10 | 1997-01-08 | Heterocycle-condensed morphinoid derivatives (ii) |
| PL97327943A PL327943A1 (en) | 1996-01-10 | 1997-01-08 | Condensed heterocyclic derivatives of morphonoide (ii) |
| ES97901009T ES2188888T3 (es) | 1996-01-10 | 1997-01-08 | Derivados morfinoides 8ii) con condensados con heterociclos. |
| CZ982182A CZ218298A3 (cs) | 1996-01-10 | 1997-01-08 | Heterocyklický kondenzovaný morfiátový derivát (II), způsob jeho přípravy a použití |
| ZA97172A ZA97172B (en) | 1996-01-10 | 1997-01-09 | Heterocycle-condensed morphinoid derivatives |
| TW086100197A TW357148B (en) | 1996-01-10 | 1997-01-10 | Heterocycle-condensed morphinoid derivatives (II) the invention relates to a substituted mono heterocycle-condensed morphinoid derivatives as analgesics and for treating pathological conditions |
| NO983169A NO983169L (no) | 1996-01-10 | 1998-07-09 | Hetrosykel-kondenserte morfinoidderivater (31) |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITMI960029 IT1282950B1 (it) | 1996-01-10 | 1996-01-10 | Derivati eterociclo-condensati di morfinoidi |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| ITMI960029A0 ITMI960029A0 (it) | 1996-01-10 |
| ITMI960029A1 ITMI960029A1 (it) | 1997-07-10 |
| IT1282950B1 true IT1282950B1 (it) | 1998-04-02 |
Family
ID=11372871
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ITMI960029 IT1282950B1 (it) | 1996-01-10 | 1996-01-10 | Derivati eterociclo-condensati di morfinoidi |
Country Status (2)
| Country | Link |
|---|---|
| IT (1) | IT1282950B1 (it) |
| ZA (1) | ZA97172B (it) |
-
1996
- 1996-01-10 IT ITMI960029 patent/IT1282950B1/it active IP Right Grant
-
1997
- 1997-01-09 ZA ZA97172A patent/ZA97172B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ITMI960029A1 (it) | 1997-07-10 |
| ZA97172B (en) | 1998-07-09 |
| ITMI960029A0 (it) | 1996-01-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 0001 | Granted | ||
| TA | Fee payment date (situation as of event date), data collected since 19931001 |
Effective date: 19990129 |