IN2013DN02555A - - Google Patents

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Publication number
IN2013DN02555A
IN2013DN02555A IN2555DEN2013A IN2013DN02555A IN 2013DN02555 A IN2013DN02555 A IN 2013DN02555A IN 2555DEN2013 A IN2555DEN2013 A IN 2555DEN2013A IN 2013DN02555 A IN2013DN02555 A IN 2013DN02555A
Authority
IN
India
Prior art keywords
compounds
processes
relates
disorders
preparing
Prior art date
Application number
Other languages
English (en)
Inventor
Alessandra Bartolozzi
Todd Bosanac
Zhidong Chen
Lombaert Stéphane De
Jonathon Alan Dines
John D Huber
Weimin Liu
Pui Leng Loke
Tina Marie Morwick
Alan Olague
Doris Riether
Heather Tye
Lifen Wu
Renee M Zindell
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44720163&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2013DN02555(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of IN2013DN02555A publication Critical patent/IN2013DN02555A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965Non-condensed pyrazines
    • A61K31/497Non-condensed pyrazines containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
IN2555DEN2013 2010-09-23 2011-09-20 IN2013DN02555A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US38573310P 2010-09-23 2010-09-23
US201161533349P 2011-09-12 2011-09-12
PCT/US2011/052254 WO2012040139A1 (en) 2010-09-23 2011-09-20 Oxadiazole inhibitors of leukotriene production

Publications (1)

Publication Number Publication Date
IN2013DN02555A true IN2013DN02555A (pt) 2015-08-07

Family

ID=44720163

Family Applications (1)

Application Number Title Priority Date Filing Date
IN2555DEN2013 IN2013DN02555A (pt) 2010-09-23 2011-09-20

Country Status (18)

Country Link
US (1) US8575201B2 (pt)
EP (1) EP2619197B1 (pt)
JP (1) JP5713511B2 (pt)
KR (1) KR20130109122A (pt)
CN (1) CN103261193A (pt)
AU (1) AU2011305667A1 (pt)
BR (1) BR112013008638A2 (pt)
CA (1) CA2812449A1 (pt)
CL (1) CL2013000788A1 (pt)
CO (1) CO6710902A2 (pt)
EA (1) EA201300389A1 (pt)
EC (1) ECSP13012548A (pt)
IN (1) IN2013DN02555A (pt)
MX (1) MX2013003202A (pt)
PE (1) PE20131398A1 (pt)
SG (1) SG188604A1 (pt)
WO (1) WO2012040139A1 (pt)
ZA (1) ZA201301747B (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5862669B2 (ja) * 2010-08-26 2016-02-16 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ロイコトリエン産生のオキサジアゾール阻害剤
US8580825B2 (en) * 2010-09-23 2013-11-12 Boehringer Ingelheim International Gmbh Oxadiazole inhibitors of leukotriene production
CN103261193A (zh) 2010-09-23 2013-08-21 贝林格尔.英格海姆国际有限公司 抑制白三烯生成的*二唑抑制剂
AR089853A1 (es) 2012-02-01 2014-09-24 Boehringer Ingelheim Int Inhibidores de oxadiazol de la produccion de leucotrienos para terapia de combinacion, composicion farmaceutica, uso
US9079866B2 (en) * 2013-02-04 2015-07-14 Janssen Pharmaceutica Nv Flap modulators
EP2875736B1 (en) 2013-11-26 2016-07-27 Citrage N-Carbamoylputrescine to enhance muscle protein synthesis

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ516506A (en) 1999-08-06 2004-02-27 Janssen Pharmaceutica Nv Interleukin-5 inhibiting 6-azauracil derivatives
EP1653970A4 (en) * 2003-08-13 2008-10-15 Novartis Vaccines & Diagnostic GSK-3 INHIBITORS AND USES
US7319108B2 (en) 2004-01-25 2008-01-15 Sanofi-Aventis Deutschland Gmbh Aryl-substituted heterocycles, process for their preparation and their use as medicaments
US20070287736A1 (en) 2004-10-18 2007-12-13 Lin Chu Diphenyl Substituted Alkanes as Flap Inhibitors
US8399666B2 (en) * 2005-11-04 2013-03-19 Panmira Pharmaceuticals, Llc 5-lipoxygenase-activating protein (FLAP) inhibitors
US7977359B2 (en) * 2005-11-04 2011-07-12 Amira Pharmaceuticals, Inc. 5-lipdxygenase-activating protein (FLAP) inhibitors
GB2431927B (en) 2005-11-04 2010-03-17 Amira Pharmaceuticals Inc 5-Lipoxygenase-activating protein (FLAP) inhibitors
CA2648555A1 (en) * 2006-04-11 2007-10-25 Merck & Co., Inc. Diaryl substituted alkanes
CA2787343C (en) 2006-06-26 2016-08-02 Amgen Inc. Compositions comprising modified lcat and uses thereof
JP2010502615A (ja) * 2006-09-01 2010-01-28 メルク エンド カムパニー インコーポレーテッド 5−リポキシゲナーゼ活性化タンパク質(flap)の阻害剤
WO2008128335A1 (en) 2007-04-20 2008-10-30 Merck Frosst Canada Ltd. Novel heteroaromatic compounds as inhibitors of stearoyl-coenzyme a delta-9 desaturase
EP2170065A4 (en) 2007-06-20 2011-11-23 Merck Sharp & Dohme DIPHENYL SUBSTITUTED ALKANES
US20110003815A1 (en) 2007-10-10 2011-01-06 Merck & Co., Inc. Diphenyl substituted cycloalkanes
DE102008037790A1 (de) * 2008-08-14 2010-02-18 Merck Patent Gmbh Bicyclische Triazolderivate
MX2011004570A (es) * 2008-10-31 2011-06-17 Merck Sharp & Dohme Antagonistas del receptor p2x3 para el tratamiento del dolor.
JP2012516885A (ja) 2009-02-04 2012-07-26 ファイザー・インク 4−アミノ−7,8−ジヒドロピリド[4,3−d]ピリミジン−5(6H)−オン誘導体
SG185414A1 (en) 2010-05-12 2012-12-28 Univ Vanderbilt Heterocyclic sulfone mglur4 allosteric potentiators, compositions, and methods of treating neurological dysfunction
JP5619284B2 (ja) * 2010-08-16 2014-11-05 ベーリンガーインゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ロイコトリエン産生のオキサジアゾール阻害薬
JP5862669B2 (ja) * 2010-08-26 2016-02-16 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ロイコトリエン産生のオキサジアゾール阻害剤
US8580825B2 (en) * 2010-09-23 2013-11-12 Boehringer Ingelheim International Gmbh Oxadiazole inhibitors of leukotriene production
CN103261193A (zh) 2010-09-23 2013-08-21 贝林格尔.英格海姆国际有限公司 抑制白三烯生成的*二唑抑制剂

Also Published As

Publication number Publication date
AU2011305667A1 (en) 2013-03-21
ECSP13012548A (es) 2013-06-28
MX2013003202A (es) 2013-04-24
WO2012040139A1 (en) 2012-03-29
KR20130109122A (ko) 2013-10-07
JP2013537909A (ja) 2013-10-07
US20120295896A1 (en) 2012-11-22
CL2013000788A1 (es) 2013-06-28
ZA201301747B (en) 2014-08-27
US8575201B2 (en) 2013-11-05
EA201300389A1 (ru) 2013-09-30
EP2619197B1 (en) 2015-08-05
EP2619197A1 (en) 2013-07-31
CO6710902A2 (es) 2013-07-15
CN103261193A (zh) 2013-08-21
CA2812449A1 (en) 2012-03-29
BR112013008638A2 (pt) 2016-06-21
SG188604A1 (en) 2013-04-30
PE20131398A1 (es) 2013-12-19
JP5713511B2 (ja) 2015-05-07

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