IN2012DN01961A - - Google Patents

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IN2012DN01961A
IN2012DN01961A IN1961DEN2012A IN2012DN01961A IN 2012DN01961 A IN2012DN01961 A IN 2012DN01961A IN 1961DEN2012 A IN1961DEN2012 A IN 1961DEN2012A IN 2012DN01961 A IN2012DN01961 A IN 2012DN01961A
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IN
India
Prior art keywords
entities
kinase activity
heterocyclic
modulate
methods
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Inventor
Pingda Ren
Yi Liu
Liansheng Li
Katrina Chan
Troy Edward Wilson
Simon Fraser Campbell
Original Assignee
Intellikine Llc
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43607312&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2012DN01961(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Intellikine Llc filed Critical Intellikine Llc
Publication of IN2012DN01961A publication Critical patent/IN2012DN01961A/en

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/423—Oxazoles condensed with carbocyclic rings
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
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Abstract

Heterocyclic entities that modulate PI3 kinase activity, pharmaceutical compositions containing the heterocyclic entities, and methods of using these chemical entities for treating diseases and conditions associated with PI3 kinase activity are described herein.
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