IL80193A0 - Esters of dihydrolysergic acid - Google Patents
Esters of dihydrolysergic acidInfo
- Publication number
- IL80193A0 IL80193A0 IL80193A IL8019386A IL80193A0 IL 80193 A0 IL80193 A0 IL 80193A0 IL 80193 A IL80193 A IL 80193A IL 8019386 A IL8019386 A IL 8019386A IL 80193 A0 IL80193 A0 IL 80193A0
- Authority
- IL
- Israel
- Prior art keywords
- esters
- dihydrolysergic acid
- dihydrolysergic
- acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
- C07D457/04—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 8
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/48—Ergoline derivatives, e.g. lysergic acid, ergotamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/782,340 US4714704A (en) | 1985-10-01 | 1985-10-01 | Alkoxy cycloalkanol esters of dihydrolysergic acid useful as 5HT receptor antagonists |
US06/782,341 US4713385A (en) | 1985-10-01 | 1985-10-01 | Alkoxy and dialkoxyalkyl esters of dihydrolysergic acid and related compounds useful as 5HT receptor antagonists |
US06/782,342 US4772709A (en) | 1985-10-01 | 1985-10-01 | Process of making ketoalkanol esters of dihydrolysergic acid |
US06/782,337 US4683236A (en) | 1985-10-01 | 1985-10-01 | Cycloalkanol esters of dihydrolysergic acid useful as 5Ht2 receptor antagonists |
US06/782,338 US4713384A (en) | 1985-10-01 | 1985-10-01 | Selective method for blocking 5HT2 receptors |
Publications (1)
Publication Number | Publication Date |
---|---|
IL80193A0 true IL80193A0 (en) | 1986-12-31 |
Family
ID=27542204
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL80193A IL80193A0 (en) | 1985-10-01 | 1986-09-29 | Esters of dihydrolysergic acid |
Country Status (17)
Country | Link |
---|---|
EP (1) | EP0219257B1 (pt) |
JP (1) | JPH0723376B2 (pt) |
KR (1) | KR880001009B1 (pt) |
AR (1) | AR244687A1 (pt) |
AU (1) | AU594373B2 (pt) |
CY (1) | CY1784A (pt) |
DE (1) | DE3689702T2 (pt) |
DK (1) | DK466886A (pt) |
ES (1) | ES2002392A6 (pt) |
GR (1) | GR862466B (pt) |
HK (1) | HK51894A (pt) |
HU (1) | HU206711B (pt) |
IE (1) | IE61976B1 (pt) |
IL (1) | IL80193A0 (pt) |
MY (1) | MY102598A (pt) |
NZ (1) | NZ217724A (pt) |
PT (1) | PT83450B (pt) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4734501A (en) * | 1985-10-01 | 1988-03-29 | Eli Lilly And Company | N-alkylation of dihydrolysergic acid |
US4782063A (en) * | 1987-05-11 | 1988-11-01 | Eli Lilly And Company | Ergoline esters useful as serotonin antagonists |
GB8824744D0 (en) * | 1988-10-21 | 1988-11-30 | Erba Carlo Spa | Antiemesis ergoline derivatives |
JPH11503757A (ja) * | 1995-04-18 | 1999-03-30 | イーライ・リリー・アンド・カンパニー | 5−ht▲下7▼レセプターにおいて生理学的および病理学的機能を生じるエルゴリン化合物の使用方法 |
US5880134A (en) * | 1996-03-20 | 1999-03-09 | Eli Lilly And Company | Method for using ergoline compounds to effect physiological and pathological functions at the 5-HT7 receptor |
WO2013167220A1 (de) * | 2012-05-08 | 2013-11-14 | Merck Patent Gmbh | Verwendung von cyclohexanolethers mit antimikrobiellen eigenschaften |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3580916A (en) * | 1969-02-20 | 1971-05-25 | Lilly Co Eli | Hydroxyesters of hexa- and octahydroindoloquinolines |
CH549571A (de) * | 1970-09-16 | 1974-05-31 | Lilly Co Eli | Verfahren zur herstellung von estern der lysergsaeure bzw. dihydrolysergsaeure und deren verwendung. |
US4563461A (en) * | 1983-03-10 | 1986-01-07 | Eli Lilly And Company | Selective method for blocking 5HT2 receptors |
US4734501A (en) * | 1985-10-01 | 1988-03-29 | Eli Lilly And Company | N-alkylation of dihydrolysergic acid |
US4713384A (en) * | 1985-10-01 | 1987-12-15 | Eli Lilly And Company | Selective method for blocking 5HT2 receptors |
-
1986
- 1986-09-29 PT PT83450A patent/PT83450B/pt not_active IP Right Cessation
- 1986-09-29 EP EP86307443A patent/EP0219257B1/en not_active Expired - Lifetime
- 1986-09-29 NZ NZ217724A patent/NZ217724A/xx unknown
- 1986-09-29 AU AU63210/86A patent/AU594373B2/en not_active Ceased
- 1986-09-29 IL IL80193A patent/IL80193A0/xx not_active IP Right Cessation
- 1986-09-29 DE DE3689702T patent/DE3689702T2/de not_active Expired - Fee Related
- 1986-09-29 GR GR862466A patent/GR862466B/el unknown
- 1986-09-30 AR AR86305427A patent/AR244687A1/es active
- 1986-09-30 ES ES8602320A patent/ES2002392A6/es not_active Expired
- 1986-09-30 HU HU864146A patent/HU206711B/hu not_active IP Right Cessation
- 1986-09-30 KR KR1019860008205A patent/KR880001009B1/ko not_active IP Right Cessation
- 1986-09-30 IE IE258886A patent/IE61976B1/en not_active IP Right Cessation
- 1986-09-30 DK DK466886A patent/DK466886A/da not_active Application Discontinuation
- 1986-09-30 JP JP61234256A patent/JPH0723376B2/ja not_active Expired - Lifetime
-
1987
- 1987-09-24 MY MYPI87001918A patent/MY102598A/en unknown
-
1994
- 1994-05-19 HK HK51894A patent/HK51894A/xx unknown
-
1995
- 1995-10-20 CY CY178495A patent/CY1784A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
PT83450B (pt) | 1989-05-12 |
NZ217724A (en) | 1989-02-24 |
IE862588L (en) | 1987-04-01 |
JPS6284084A (ja) | 1987-04-17 |
IE61976B1 (en) | 1994-12-14 |
HUT41780A (en) | 1987-05-28 |
CY1784A (en) | 1995-10-20 |
HU206711B (en) | 1992-12-28 |
JPH0723376B2 (ja) | 1995-03-15 |
KR870004028A (ko) | 1987-05-07 |
PT83450A (en) | 1986-10-01 |
EP0219257A2 (en) | 1987-04-22 |
ES2002392A6 (es) | 1988-08-01 |
DK466886A (da) | 1987-04-02 |
DK466886D0 (da) | 1986-09-30 |
EP0219257B1 (en) | 1994-03-09 |
DE3689702D1 (de) | 1994-04-14 |
HK51894A (en) | 1994-05-27 |
KR880001009B1 (ko) | 1988-06-13 |
AR244687A1 (es) | 1993-11-30 |
MY102598A (en) | 1992-08-17 |
GR862466B (en) | 1987-02-02 |
AU594373B2 (en) | 1990-03-08 |
EP0219257A3 (en) | 1988-12-28 |
AU6321086A (en) | 1987-04-02 |
DE3689702T2 (de) | 1994-07-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RH | Patent void |