IL57450A - Aminothiazole derivatives and pharmaceutical compositions containing them - Google Patents

Aminothiazole derivatives and pharmaceutical compositions containing them

Info

Publication number: IL57450A
Authority: IL; Israel
Prior art keywords: pharmaceutical compositions; compositions containing; aminothiazole derivatives; aminothiazole; derivatives
Prior art date: 1978-06-02

Application number

IL57450A

Other languages

English (en)

Other versions

IL57450A0 (en

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1978-06-02

Filing date

1979-05-31

Publication date

1982-11-30

1979-05-31 Application filed by Pfizer filed Critical Pfizer

1979-09-30 Publication of IL57450A0 publication Critical patent/IL57450A0/xx

1982-11-30 Publication of IL57450A publication Critical patent/IL57450A/xx

Links

RAIPHJJURHTUIC-UHFFFAOYSA-N 1,3-thiazol-2-amine Chemical class NC1=NC=CS1 RAIPHJJURHTUIC-UHFFFAOYSA-N 0.000 title 1
239000008194 pharmaceutical composition Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D307/52—Radicals substituted by nitrogen atoms not forming part of a nitro radical
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
- C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
- F—MECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
- F16—ENGINEERING ELEMENTS AND UNITS; GENERAL MEASURES FOR PRODUCING AND MAINTAINING EFFECTIVE FUNCTIONING OF MACHINES OR INSTALLATIONS; THERMAL INSULATION IN GENERAL
- F16B—DEVICES FOR FASTENING OR SECURING CONSTRUCTIONAL ELEMENTS OR MACHINE PARTS TOGETHER, e.g. NAILS, BOLTS, CIRCLIPS, CLAMPS, CLIPS OR WEDGES; JOINTS OR JOINTING
- F16B15/00—Nails; Staples
- F16B15/0023—Nail plates
- F16B2015/0076—Nail plates with provisions for additional fastening means, e.g. hooks, holes for separate screws or nails, adhesive

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Immunology (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

IL57450A 1978-06-02 1979-05-31 Aminothiazole derivatives and pharmaceutical compositions containing them IL57450A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US91183078A	1978-06-02	1978-06-02

Publications (2)

Publication Number	Publication Date
IL57450A0 IL57450A0 (en)	1979-09-30
IL57450A true IL57450A (en)	1982-11-30

Family

ID=25430923

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL57450A IL57450A (en)	1978-06-02	1979-05-31	Aminothiazole derivatives and pharmaceutical compositions containing them

Country Status (36)

Country	Link
JP (1)	JPS5936988B2 (de)
AR (1)	AR226285A1 (de)
AT (1)	AT373248B (de)
AU (1)	AU511242B2 (de)
BE (1)	BE876732A (de)
CA (1)	CA1117949A (de)
CH (1)	CH639653A5 (de)
CS (1)	CS216927B2 (de)
DD (1)	DD144055A5 (de)
DE (1)	DE2922523C2 (de)
DK (1)	DK150068C (de)
EG (1)	EG14354A (de)
ES (1)	ES481220A1 (de)
FI (1)	FI68820C (de)
FR (1)	FR2427333A1 (de)
GB (1)	GB2022085B (de)
GR (1)	GR73142B (de)
HK (1)	HK66487A (de)
HU (1)	HU180045B (de)
IE (1)	IE48426B1 (de)
IL (1)	IL57450A (de)
IT (1)	IT1121238B (de)
KE (1)	KE3459A (de)
LU (1)	LU81349A1 (de)
MY (1)	MY8500318A (de)
NL (1)	NL178421C (de)
NO (1)	NO150760C (de)
NZ (1)	NZ190623A (de)
PH (1)	PH17020A (de)
PL (1)	PL117515B1 (de)
PT (1)	PT69718A (de)
SE (1)	SE438333B (de)
SG (1)	SG56184G (de)
SU (1)	SU843746A3 (de)
YU (1)	YU40997B (de)
ZA (1)	ZA792729B (de)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0063575A4 (de) *	1980-10-24	1983-02-14	Ronald Peter Hansen	Staub-ermässigungssystem.
JPS57136579A (en) *	1981-01-21	1982-08-23	Mitsui Toatsu Chem Inc	Thiazolylurea derivative, its preparation, and pharmaceutical composition containing the same
EP0068033B1 (de) *	1981-01-08	1985-07-10	Mitsui Toatsu Kagaku Kabushiki Kaisha	N-(4-phenyl-2-thiazolyl)karbamatabkömmlinge, verfahren zu deren herstellung und diese enthaltendes arzneimittel
JPS57116067A (en) *	1981-01-12	1982-07-19	Sankyo Kagaku Kk	Novel 8-quinolinesulfonyl derivative, its synthesis and use
WO1982002386A1 (en) *	1981-01-13	1982-07-22	Sakano Isao	Aminothiazole derivatives,process for their preparation,and medicinal composition containing same
US4501750A (en) *	1981-01-13	1985-02-26	Mitsui Toatsu Kaguku Kabushiki Kaisha	Thiazole compounds, a process for preparing same and a pharmaceutical composition containing the thiazole compounds
JPS57154175A (en) *	1981-03-16	1982-09-22	Mitsui Toatsu Chem Inc	2-thiazoleamine derivative, its preparation, and drug composition comprising it
DE3227329A1 (de) *	1982-07-22	1984-01-26	Basf Ag, 6700 Ludwigshafen	Verfahren zur herstellung von 2-n,n-disubstituierten aminothiazolen
WO1986003203A1 (en) *	1984-11-22	1986-06-05	Yoshitomi Pharmaceutical Industries, Ltd.	Thienylthiazole derivatives
FR2581063B1 (fr) *	1985-04-30	1987-07-17	Chauvin Blache Lab	Amino-2 thiazoles n-substitues, leur procede de preparation et leur application en therapeutique
JPS63152368A (ja) *	1986-06-03	1988-06-24	Sumitomo Pharmaceut Co Ltd	新規なアミノアゾ−ル誘導体およびその酸付加塩
JPH075579B2 (ja) *	1986-09-01	1995-01-25	吉富製薬株式会社	アミノチアゾ−ル化合物
JPH0753666B2 (ja) *	1987-09-14	1995-06-07	久光製薬株式会社	置換ジフェニルチアゾール誘導体からなる抗炎症剤
WO1991002394A1 (en) *	1989-08-10	1991-02-21	Commonwealth Scientific And Industrial Research Organisation	Producing electrosuspensions
AU654125B2 (en) *	1991-03-07	1994-10-27	Hisamitsu Pharmaceutical Co., Inc.	Novel diphenylthyazole derivative
FR2692893B1 (fr) *	1992-06-24	1994-09-02	Sanofi Elf	Dérivés alkylamino ramifiés du thiazole, leurs procédés de préparation et les compositions pharmaceutiques qui les contiennent.
EP1125932A3 (de) *	1994-07-27	2001-08-29	G.D. Searle & Co.	Substituierte Thiazole zur Behandlung von Entzündungen
FR2754258B1 (fr)	1996-10-08	1998-12-31	Sanofi Sa	Derives d'aminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenant
WO2001064674A1 (en) *	2000-03-01	2001-09-07	Janssen Pharmaceutica N.V.	2,4-disubstituted thiazolyl derivatives
EP1423113A4 (de) *	2001-08-13	2007-04-18	Phenex Pharmaceuticals Ag	Nr1h4-nuklearrezeptorbindende verbindungen
AU2002340010A1 (en) *	2001-09-26	2003-04-07	Bayer Corporation	Substituted 3-pyridyl indoles and indazoles as c17,20 lyase inhibitors
AU2003202495B2 (en)	2002-01-11	2006-07-20	Sankyo Company, Limited	Amino alcohol derivative or phosphonic acid derivative and medicinal composition containing these
EP1555264A1 (de) *	2004-01-15	2005-07-20	Sireen AG	Fünfringheterocyclische Verbindungen als Inhibitoren der Familie der SRC Proteinkinasen.
KR101182619B1 (ko)	2004-02-24	2012-09-18	상꾜 가부시키가이샤	아미노 알코올 화합물
KR20080019213A (ko) *	2005-05-09	2008-03-03	아칠리온 파르마세우티칼스 인코포레이티드	티아졸 화합물 및 그 사용방법
KR20080091369A (ko)	2006-01-18	2008-10-10	암젠 인크	단백질 키나제 ｂ（ｐｋｂ） 억제제로서 티아졸 화합물
JP2010533715A (ja)	2007-07-17	2010-10-28	アムジエン・インコーポレーテツド	複素環系ｐｋｂ調節剤
US7919504B2 (en)	2007-07-17	2011-04-05	Amgen Inc.	Thiadiazole modulators of PKB
US20120316182A1 (en)	2011-06-10	2012-12-13	Calcimedica, Inc.	Compounds that modulate intracellular calcium
WO2012170951A2 (en) *	2011-06-10	2012-12-13	Calcimedica, Inc.	Compounds that modulate intracellular calcium
WO2013059677A1 (en)	2011-10-19	2013-04-25	Calcimedica, Inc.	Compounds that modulate intracellular calcium
CN110590785B (zh) *	2019-09-23	2021-02-02	武汉大学	一种氨基噻唑类化合物及其制备方法与抗肠道病毒71型的应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3458526A (en) *	1966-09-26	1969-07-29	Upjohn Co	Certain 2-amino-4,5-bis(p-methoxyphenyl)thiazoles

1979
- 1979-04-30 DK DK177679A patent/DK150068C/da not_active IP Right Cessation
- 1979-05-23 GB GB7917872A patent/GB2022085B/en not_active Expired
- 1979-05-29 CH CH501679A patent/CH639653A5/fr not_active IP Right Cessation
- 1979-05-30 EG EG333/79A patent/EG14354A/xx active
- 1979-05-30 CS CS793728A patent/CS216927B2/cs unknown
- 1979-05-31 HU HU79PI679A patent/HU180045B/hu not_active IP Right Cessation
- 1979-05-31 SE SE7904798A patent/SE438333B/sv not_active IP Right Cessation
- 1979-05-31 YU YU1288/79A patent/YU40997B/xx unknown
- 1979-05-31 LU LU81349A patent/LU81349A1/xx unknown
- 1979-05-31 AU AU47634/79A patent/AU511242B2/en not_active Ceased
- 1979-05-31 PH PH22588A patent/PH17020A/en unknown
- 1979-05-31 SU SU792773929A patent/SU843746A3/ru active
- 1979-05-31 CA CA000328805A patent/CA1117949A/en not_active Expired
- 1979-05-31 IL IL57450A patent/IL57450A/xx unknown
- 1979-06-01 PL PL1979216030A patent/PL117515B1/pl unknown
- 1979-06-01 NL NLAANVRAGE7904337,A patent/NL178421C/xx not_active IP Right Cessation
- 1979-06-01 FR FR7914164A patent/FR2427333A1/fr active Granted
- 1979-06-01 ZA ZA792729A patent/ZA792729B/xx unknown
- 1979-06-01 NZ NZ190623A patent/NZ190623A/en unknown
- 1979-06-01 DD DD79213371A patent/DD144055A5/de not_active IP Right Cessation
- 1979-06-01 AT AT0401679A patent/AT373248B/de not_active IP Right Cessation
- 1979-06-01 JP JP54068781A patent/JPS5936988B2/ja not_active Expired
- 1979-06-01 DE DE2922523A patent/DE2922523C2/de not_active Expired
- 1979-06-01 NO NO791831A patent/NO150760C/no unknown
- 1979-06-01 BE BE0/195534A patent/BE876732A/xx not_active IP Right Cessation
- 1979-06-01 FI FI791754A patent/FI68820C/fi not_active IP Right Cessation
- 1979-06-01 ES ES481220A patent/ES481220A1/es not_active Expired
- 1979-06-01 IT IT23228/79A patent/IT1121238B/it active
- 1979-06-01 AR AR276782A patent/AR226285A1/es active
- 1979-06-01 GR GR59240A patent/GR73142B/el unknown
- 1979-06-01 PT PT69718A patent/PT69718A/pt unknown
- 1979-08-08 IE IE1069/79A patent/IE48426B1/en unknown
1984
- 1984-08-13 SG SG561/84A patent/SG56184G/en unknown
- 1984-09-24 KE KE3459A patent/KE3459A/xx unknown
1985
- 1985-12-30 MY MY318/85A patent/MY8500318A/xx unknown
1987
- 1987-09-17 HK HK664/87A patent/HK66487A/xx unknown

Also Published As

Publication number	Publication date
GR73142B (de)	1984-02-09
JPS5936988B2 (ja)	1984-09-06
DE2922523A1 (de)	1979-12-06
FI791754A (fi)	1979-11-26
NO791831L (no)	1979-12-04
JPS54160369A (en)	1979-12-19
PH17020A (en)	1984-05-11
LU81349A1 (fr)	1979-12-07
AU511242B2 (en)	1980-08-07
GB2022085B (en)	1983-01-12
NL7904337A (nl)	1979-12-04
SU843746A3 (ru)	1981-06-30
PL117515B1 (en)	1981-08-31
PT69718A (en)	1979-07-01
SE438333B (sv)	1985-04-15
FR2427333B1 (de)	1983-05-20
YU40997B (en)	1986-10-31
MY8500318A (en)	1985-12-31
AT373248B (de)	1983-12-27
ZA792729B (en)	1981-03-25
CA1117949A (en)	1982-02-09
DK150068C (da)	1987-06-29
KE3459A (en)	1984-10-12
CH639653A5 (fr)	1983-11-30
ATA401679A (de)	1983-05-15
EG14354A (en)	1984-06-30
DE2922523C2 (de)	1982-10-21
AR226285A1 (es)	1982-06-30
DK150068B (da)	1986-12-01
SG56184G (en)	1985-03-08
HK66487A (en)	1987-09-25
DD144055A5 (de)	1980-09-24
BE876732A (fr)	1979-12-03
FR2427333A1 (fr)	1979-12-28
NO150760C (no)	1984-12-12
NL178421B (nl)	1985-10-16
FI68820B (fi)	1985-07-31
YU128879A (en)	1982-10-31
PL216030A1 (de)	1980-03-10
CS216927B2 (en)	1982-12-31
NZ190623A (en)	1984-07-06
NL178421C (nl)	1986-03-17
DK177679A (da)	1979-12-03
GB2022085A (en)	1979-12-12
FI68820C (fi)	1985-11-11
IT1121238B (it)	1986-03-26
IE48426B1 (en)	1985-01-23
ES481220A1 (es)	1980-09-01
IL57450A0 (en)	1979-09-30
AU4763479A (en)	1979-12-06
SE7904798L (sv)	1979-12-03
IE791069L (en)	1979-12-02
HU180045B (en)	1983-01-28
IT7923228A0 (it)	1979-06-01
NO150760B (no)	1984-09-03

Publication	Publication Date	Title
IL57450A (en)	1982-11-30	Aminothiazole derivatives and pharmaceutical compositions containing them
NZ189378A (en)	1983-03-15	4-amino-5-alkylsulphonyl-ortho-anisamdes and pharmaceutical compositions
NZ190784A (en)	1982-03-16	Benzofuranyl-piperidines and pharmaceutical compositions
NZ190758A (en)	1980-10-24	Phenylpiperazine derivatives and pharmaceutical compositions
IL56407A (en)	1983-05-15	4-amino-3-sulfamoylpyridyl derivatives and pharmaceutical compositions containing them
IL58730A (en)	1984-01-31	Spiro-polycyclic imidazolidinedione derivatives and pharmaceutical compositions containing them
PH15937A (en)	1983-04-29	Thiazolidine derivatives and their pharmaceutical compositions
IL56821A0 (en)	1979-05-31	Heterocycylcarbonyl derivatives of ure and pharmaceutical composition containing them
IL57268A0 (en)	1979-09-30	Di-o-n-alkyl clycerol derivatives and pharmaceutical compositions containing them
IL60376A0 (en)	1980-09-16	3-methyleneazetidine derivatives and pharmaceutical compositions containing them
PH13392A (en)	1980-03-28	Thiourea derivatives and pharmaceutical compositions containing them
IL51955A0 (en)	1977-06-30	Novel thiazole derivatives their preparation and pharmaceutical compositions containing them
NZ192142A (en)	1982-12-21	Cephalosporin derivatives and pharmaceutical compositions
IL58620A0 (en)	1980-02-29	Aryltrifluoroethanol derivatives their preparation and pharmaceutical compositions containing them
NZ189899A (en)	1982-05-25	Dilignols and dilignol-type compounds pharmaceutical compositions
NZ189896A (en)	1980-05-27	Phenylaniline derivatives and pharmaceutical compositions
NZ189769A (en)	1981-07-13	Benzylidene derivatives and pharmaceutical compositions
PH16220A (en)	1983-08-09	Pyrro-lidine derivatives and pharmaceutical compositions thereof
NZ189279A (en)	1980-08-26	Arylaminoimidazolines and pharmaceutical compositions
IL57882A0 (en)	1979-11-30	2-thiophenecarboxamido-alkylmercaptans and pharmaceutical compositions containing them
IL60695A (en)	1983-11-30	Hexahydro-trans-pyridoindole-alkanamine derivatives and pharmaceutical compositions containing them
IL61038A (en)	1983-12-30	15-sulfonamidoprostaglandin derivatives and pharmaceutical compositions containing them
NZ191556A (en)	1981-03-16	Aurone derivatives and pharmaceutical compositions
IL57436A0 (en)	1979-09-30	Hydantoin derivatives and pharmaceutical compositions containing them
NZ190293A (en)	1980-11-28	Benzimidoyl-piperazines and pharmaceutical compositions