IL140586A - Phenyl ester derivatives of a-amino acid and pharmaceuticals containing them - Google Patents
Phenyl ester derivatives of a-amino acid and pharmaceuticals containing themInfo
- Publication number
- IL140586A IL140586A IL14058699A IL14058699A IL140586A IL 140586 A IL140586 A IL 140586A IL 14058699 A IL14058699 A IL 14058699A IL 14058699 A IL14058699 A IL 14058699A IL 140586 A IL140586 A IL 140586A
- Authority
- IL
- Israel
- Prior art keywords
- acid
- amino acid
- alkoxy
- alkyl
- acid phenyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/38—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to acyclic carbon atoms and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C229/06—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton
- C07C229/10—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings
- C07C229/12—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings to carbon atoms of acyclic carbon skeletons
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C229/06—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton
- C07C229/10—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings
- C07C229/16—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings to carbon atoms of hydrocarbon radicals substituted by amino or carboxyl groups, e.g. ethylenediamine-tetra-acetic acid, iminodiacetic acids
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Psychiatry (AREA)
- Rheumatology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP98305837 | 1998-07-22 | ||
PCT/EP1999/005051 WO2000005196A1 (en) | 1998-07-22 | 1999-07-16 | α-AMINO ACID PHENYL ESTER DERIVATIVES |
Publications (2)
Publication Number | Publication Date |
---|---|
IL140586A0 IL140586A0 (en) | 2002-02-10 |
IL140586A true IL140586A (en) | 2004-06-01 |
Family
ID=8234960
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL14058699A IL140586A (en) | 1998-07-22 | 1999-07-16 | Phenyl ester derivatives of a-amino acid and pharmaceuticals containing them |
Country Status (27)
Country | Link |
---|---|
US (1) | US6451854B1 (no) |
EP (1) | EP1098871B1 (no) |
JP (1) | JP2002521358A (no) |
KR (1) | KR100599142B1 (no) |
CN (1) | CN1183101C (no) |
AR (1) | AR021165A1 (no) |
AT (1) | ATE244697T1 (no) |
AU (1) | AU758808B2 (no) |
BR (1) | BR9912291A (no) |
CA (1) | CA2337945A1 (no) |
CO (1) | CO5080742A1 (no) |
DE (1) | DE69909486T2 (no) |
DK (1) | DK1098871T3 (no) |
ES (1) | ES2203163T3 (no) |
HU (1) | HUP0102705A3 (no) |
ID (1) | ID27261A (no) |
IL (1) | IL140586A (no) |
NO (1) | NO20010280L (no) |
NZ (1) | NZ509327A (no) |
PE (1) | PE20000880A1 (no) |
PL (1) | PL345621A1 (no) |
PT (1) | PT1098871E (no) |
RU (1) | RU2223947C2 (no) |
SK (1) | SK1032001A3 (no) |
TR (1) | TR200100166T2 (no) |
TW (1) | TW565546B (no) |
WO (1) | WO2000005196A1 (no) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR031473A1 (es) * | 2000-11-20 | 2003-09-24 | Lundbeck & Co As H | Intensificadores de gaba en el tratamiento de enfermedades relacionadas con una reducida actividad neuroesteroide |
ES2266476T3 (es) * | 2001-01-19 | 2007-03-01 | Akzo Nobel N.V. | Derivados de ester 2,6-dialcoxifenilico de alanina como hipnoticos. |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1102011A (en) * | 1964-05-21 | 1968-02-07 | Richardson Merrell Spa | Phenol esters of amino acids |
GB1160468A (en) | 1967-05-08 | 1969-08-06 | May & Baker Ltd | Morpholine Derivative |
-
1999
- 1999-07-16 US US09/744,004 patent/US6451854B1/en not_active Expired - Fee Related
- 1999-07-16 SK SK103-2001A patent/SK1032001A3/sk unknown
- 1999-07-16 CA CA002337945A patent/CA2337945A1/en not_active Abandoned
- 1999-07-16 BR BR9912291-0A patent/BR9912291A/pt not_active Application Discontinuation
- 1999-07-16 KR KR1020017000592A patent/KR100599142B1/ko not_active IP Right Cessation
- 1999-07-16 TR TR2001/00166T patent/TR200100166T2/xx unknown
- 1999-07-16 PT PT99936544T patent/PT1098871E/pt unknown
- 1999-07-16 CN CNB998091308A patent/CN1183101C/zh not_active Expired - Fee Related
- 1999-07-16 DE DE69909486T patent/DE69909486T2/de not_active Expired - Fee Related
- 1999-07-16 AU AU51602/99A patent/AU758808B2/en not_active Ceased
- 1999-07-16 IL IL14058699A patent/IL140586A/en not_active IP Right Cessation
- 1999-07-16 NZ NZ509327A patent/NZ509327A/xx unknown
- 1999-07-16 HU HU0102705A patent/HUP0102705A3/hu unknown
- 1999-07-16 AT AT99936544T patent/ATE244697T1/de not_active IP Right Cessation
- 1999-07-16 JP JP2000561153A patent/JP2002521358A/ja active Pending
- 1999-07-16 ID IDW20010160A patent/ID27261A/id unknown
- 1999-07-16 PL PL99345621A patent/PL345621A1/xx not_active IP Right Cessation
- 1999-07-16 ES ES99936544T patent/ES2203163T3/es not_active Expired - Lifetime
- 1999-07-16 DK DK99936544T patent/DK1098871T3/da active
- 1999-07-16 RU RU2001104896/04A patent/RU2223947C2/ru not_active IP Right Cessation
- 1999-07-16 WO PCT/EP1999/005051 patent/WO2000005196A1/en active IP Right Grant
- 1999-07-16 EP EP99936544A patent/EP1098871B1/en not_active Expired - Lifetime
- 1999-07-21 AR ARP990103567A patent/AR021165A1/es active IP Right Grant
- 1999-07-21 CO CO99045953A patent/CO5080742A1/es unknown
- 1999-07-21 PE PE1999000731A patent/PE20000880A1/es not_active Application Discontinuation
- 1999-07-23 TW TW088112565A patent/TW565546B/zh not_active IP Right Cessation
-
2001
- 2001-01-17 NO NO20010280A patent/NO20010280L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
RU2223947C2 (ru) | 2004-02-20 |
SK1032001A3 (en) | 2001-08-06 |
ES2203163T3 (es) | 2004-04-01 |
BR9912291A (pt) | 2001-04-17 |
AU5160299A (en) | 2000-02-14 |
HUP0102705A2 (hu) | 2001-12-28 |
EP1098871B1 (en) | 2003-07-09 |
PE20000880A1 (es) | 2000-09-12 |
AR021165A1 (es) | 2002-07-03 |
AU758808B2 (en) | 2003-03-27 |
WO2000005196A1 (en) | 2000-02-03 |
PT1098871E (pt) | 2003-11-28 |
TR200100166T2 (tr) | 2001-05-21 |
PL345621A1 (en) | 2002-01-02 |
US6451854B1 (en) | 2002-09-17 |
TW565546B (en) | 2003-12-11 |
DK1098871T3 (da) | 2003-10-27 |
HUP0102705A3 (en) | 2002-11-28 |
CN1183101C (zh) | 2005-01-05 |
NO20010280L (no) | 2001-03-08 |
IL140586A0 (en) | 2002-02-10 |
NO20010280D0 (no) | 2001-01-17 |
DE69909486T2 (de) | 2004-05-27 |
CA2337945A1 (en) | 2000-02-03 |
EP1098871A1 (en) | 2001-05-16 |
NZ509327A (en) | 2003-04-29 |
JP2002521358A (ja) | 2002-07-16 |
ID27261A (id) | 2001-03-22 |
KR20010071905A (ko) | 2001-07-31 |
CN1311770A (zh) | 2001-09-05 |
ATE244697T1 (de) | 2003-07-15 |
KR100599142B1 (ko) | 2006-07-12 |
CO5080742A1 (es) | 2001-09-25 |
DE69909486D1 (de) | 2003-08-14 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
WO1998029409A1 (fr) | Sels d'addition acides de compose de piperidine optiquement actif et procede de production associe | |
EP0116257A1 (en) | Process for preparing 4-amino-5-hexenoic acid | |
WO1997038705A1 (en) | N-formyl hydroxylamine containing compounds useful as ace inhibitors and/or nep inhibitors | |
US6451854B1 (en) | α-amino acid phenyl ester derivatives | |
IL109111A (en) | HISTORY OF MORPOLIN AND THOMORPOLIN-2 Transformed as GABA-B Antagonists, Preparation and Pharmaceutical Preparations Containing Them | |
ATE289583T1 (de) | Stereoisomere von propyl-isopropylacetamid, verfahren zu deren herstellung sowie diese enthaltende pharmazeutische zubereitungen | |
AU2002309420B2 (en) | New compounds useful in reflux disease | |
EP1853556A1 (en) | Derivatives of aminobutanoic acid inhibiting cpt | |
MXPA01000721A (en) | &agr;-AMINO ACID PHENYL ESTER DERIVATIVES | |
CZ2001269A3 (cs) | Fenylesterové deriváty alfa-aminokyselin | |
JP4043363B2 (ja) | 催眠薬としてのアラニン2,6−ジアルコキシフェニルエステル誘導体 | |
AU672315B2 (en) | Novel processes for preparing (S)-4-amino-hepta-5,6-dienoic acid and intermediates thereof | |
US20220289668A1 (en) | N-formylhydroxylamines as neprilysin (nep) inhibitors, in particular as mixed aminopeptidase n (apn) and neprilysin (nep) inhibitors | |
JP2002524443A (ja) | ピロリジン構造を有するgaba摂取阻害剤 | |
Einhorn et al. | Synthesis of a new, C 2 Symmetric α, α-Bis-(Carboxymethyl) Substituted Nitroxide |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FF | Patent granted | ||
KB | Patent renewed | ||
MM9K | Patent not in force due to non-payment of renewal fees |