HUP0001518A3 - Tricyclic erythromycin derivatives - Google Patents

Tricyclic erythromycin derivatives

Info

Publication number: HUP0001518A3
Authority: HU; Hungary
Prior art keywords: erythromycin derivatives; tricyclic; tricyclic erythromycin; derivatives; erythromycin
Prior art date: 1997-01-07

Application number

HU0001518A

Other languages

English (en)

Original Assignee

Abbott Lab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-01-07

Filing date

1997-04-07

Publication date

2001-11-28

1997-04-07 Application filed by Abbott Lab filed Critical Abbott Lab

2000-09-28 Publication of HUP0001518A2 publication Critical patent/HUP0001518A2/hu

2001-11-28 Publication of HUP0001518A3 publication Critical patent/HUP0001518A3/hu

Links

ULGZDMOVFRHVEP-RWJQBGPGSA-N Erythromycin Chemical class O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)C(=O)[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 ULGZDMOVFRHVEP-RWJQBGPGSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

HU0001518A 1997-01-07 1997-04-07 Tricyclic erythromycin derivatives HUP0001518A3 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US08/779,786 US6274715B1 (en)	1995-11-08	1997-01-07	Tricyclic erythromycin derivatives
PCT/US1997/005871 WO1998030574A1 (en)	1997-01-07	1997-04-07	Tricyclic erythromycin derivatives

Publications (2)

Publication Number	Publication Date
HUP0001518A2 HUP0001518A2 (hu)	2000-09-28
HUP0001518A3 true HUP0001518A3 (en)	2001-11-28

Family

ID=25117567

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HU0001518A HUP0001518A3 (en)	1997-01-07	1997-04-07	Tricyclic erythromycin derivatives

Country Status (15)

Country	Link
US (1)	US6274715B1 (hu)
EP (1)	EP0961776A1 (hu)
JP (1)	JP2001507714A (hu)
KR (1)	KR20000069935A (hu)
CN (1)	CN1244202A (hu)
AR (1)	AR006678A1 (hu)
AU (1)	AU2449597A (hu)
BR (1)	BR9714269A (hu)
CA (1)	CA2277116A1 (hu)
CZ (1)	CZ231599A3 (hu)
HU (1)	HUP0001518A3 (hu)
IL (1)	IL130328A0 (hu)
NZ (1)	NZ336174A (hu)
TW (1)	TW442490B (hu)
WO (1)	WO1998030574A1 (hu)

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KR100523679B1 (ko) *	1996-09-04	2005-10-26	아보트 러보러터리즈	항균 활성을 지닌 6-ｏ-치환된 케톨라이드
FR2781484B1 (fr) *	1998-07-21	2001-08-10	Hoechst Marion Roussel Inc	Nouveaux derives de la 6-deoxy erythromycine, leur procede de preparation et leur application comme medicaments
FR2784682B1 (fr) *	1998-10-15	2002-12-06	Hoechst Marion Roussel Inc	Nouveaux derives 2-halogene de 5-0-desosaminylerythronolide a, leur procede de preparation et leur application comme medicaments
US6939861B2 (en)	1999-04-16	2005-09-06	Kosan Biosciences, Inc.	Amido macrolides
US6514944B2 (en)	1999-04-16	2003-02-04	Kosan Biosciences, Inc.	Macrolide antiinfective agents
US6451768B1 (en)	1999-04-16	2002-09-17	Kosan Biosciences, Inc.	Macrolide antiinfective agents
ATE340183T1 (de)	1999-04-16	2006-10-15	Kosan Biosciences Inc	Antiinfektiöse makrolidderivate
HUP0201516A3 (en) *	1999-05-24	2003-03-28	Pfizer Prod Inc	13-methyl-erythromycin derivatives, process for their preparation and pharmaceutical compositions containing them
US6569836B2 (en)	1999-12-02	2003-05-27	Abbott Laboratories	6-O-alkyl-2-nor-2-substituted ketolide derivatives
TWI290136B (en)	2000-04-05	2007-11-21	Daiichi Seiyaku Co	Ethylenediamine derivatives
EP1146051A3 (en) *	2000-04-10	2001-10-31	Pfizer Products Inc.	Erythromycin A derivatives
WO2003000680A1 (fr)	2001-06-20	2003-01-03	Daiichi Pharmaceutical Co., Ltd.	Derives de diamine
WO2003016302A1 (fr)	2001-08-09	2003-02-27	Daiichi Pharmaceutical Co., Ltd.	Derives de diamine
WO2003000657A1 (fr)	2001-06-20	2003-01-03	Daiichi Pharmaceutical Co., Ltd.	Derives de diamine
US20040014690A1 (en) *	2002-02-13	2004-01-22	Zhenkun Ma	Macrolides with activity against methicillin-resistant staphylococcus aureus
US7910558B2 (en) *	2002-05-13	2011-03-22	Enanta Pharmaceuticals, Inc.	Bridged macrocyclic compounds and processes for the preparation thereof
US6841664B2 (en) *	2002-07-25	2005-01-11	Enanra Pharmaceuticals, Inc.	6,11-4-carbon bridged ketolides
US7273853B2 (en) *	2002-05-13	2007-09-25	Enanta Pharmaceuticals, Inc.	6-11 bicyclic ketolide derivatives
AU2003234650A1 (en) *	2002-05-31	2003-12-19	Janssen Pharmaceutica N.V.	3-descladinosyl-6-o-carbamoyl and 6-o-carbonoyl macrolide antibacterial agents
US6750204B2 (en)	2002-06-25	2004-06-15	Enanta Pharmaceuticals, Inc.	11-C-substituted ketolides
US6812216B2 (en)	2002-06-25	2004-11-02	Enanta Pharmaceuticals, Inc.	11-C-substituted derivatives of clarithromycin
US7091196B2 (en) *	2002-09-26	2006-08-15	Rib-X Pharmaceuticals, Inc.	Bifunctional heterocyclic compounds and methods of making and using same
JP2006523229A (ja) *	2003-03-05	2006-10-12	リブ−エックスファーマシューティカルズ，インコーポレイテッド	二官能性複素環式化合物ならびにその製造および使用方法
EP1638549A4 (en)	2003-03-10	2011-06-15	Optimer Pharmaceuticals Inc	NEW ANTIBACTERIAL AGENTS
US20070149463A1 (en) *	2003-10-30	2007-06-28	Oyelere Adegboyega K	Bifunctional macrolide heterocyclic compounds and methods of making and using the same
EP1699808A1 (en) *	2003-11-18	2006-09-13	Rib-X Pharmaceuticals, Inc.	Bifunctional macrolide heterocyclic compounds and methods of making and using the same
AU2003304705A1 (en)	2003-12-24	2005-08-03	Enanta Pharmaceuticals, Inc.	11-csubsituted erythromycin derivatives
US7414030B2 (en) *	2004-01-07	2008-08-19	Enanta Pharmaceuticals, Inc.	6-11 Bicyclic erythromycin derivatives
WO2005070113A2 (en) *	2004-01-09	2005-08-04	Enanta Pharmaceuticals, Inc.	9n-substituted 6-11 bicyclic erythromycin derivatives
US7384921B2 (en) *	2004-02-20	2008-06-10	Enanta Pharmaceuticals, Inc.	Polymorphic forms of 6-11 bicyclic ketolide derivatives
EP1723159B1 (en)	2004-02-27	2019-06-12	Melinta Therapeutics, Inc.	Macrocyclic compounds and methods of making and using the same
TW200635600A (en) *	2004-12-13	2006-10-16	Enanta Pharm Inc	Tetracyclic bicyclolides
US7384922B2 (en) *	2005-05-04	2008-06-10	Enanta Pharmaceuticals, Inc.	6-11 bridged oxime erythromycin derivatives
US20060252710A1 (en) *	2005-05-04	2006-11-09	Guoqiang Wang	6-11 Bridged oxime erythromycin derivatives
CN101855219B (zh) *	2007-09-17	2014-06-25	英安塔制药有限公司	6，11-桥联的联芳大环内酯类
US8354383B2 (en) *	2007-09-17	2013-01-15	Enanta Pharmaceuticals, Inc.	6,11-bridged biaryl macrolides
US8273720B2 (en) *	2007-09-17	2012-09-25	Enanta Pharmaceuticals, Inc.	6,11-bicyclolides: bridged biaryl macrolide derivatives
EP2214484A4 (en) *	2007-10-25	2013-01-02	Cempra Pharmaceuticals Inc	PROCESS FOR PREPARING ANTIBACTERIAL MAKROLIDE AGENTS
US8208698B2 (en) *	2007-12-14	2012-06-26	Mela Sciences, Inc.	Characterizing a texture of an image
TW200946109A (en) *	2008-05-09	2009-11-16	Enanta Pharm Inc	Anti-bacterial activity of 9-hydroxy derivatives 6, 11-bicyclolides
US8796232B2 (en)	2008-10-24	2014-08-05	Cempra Pharmaceuticals, Inc.	Methods for treating resistant diseases using triazole containing macrolides
US9937194B1 (en)	2009-06-12	2018-04-10	Cempra Pharmaceuticals, Inc.	Compounds and methods for treating inflammatory diseases
AU2010292010B2 (en)	2009-09-10	2016-01-07	Cempra Pharmaceuticals, Inc.	Methods for treating malaria, tuberculosis and MAC diseases
US20110064287A1 (en) *	2009-09-14	2011-03-17	Alexandru Bogdan	Characterizing a texture of an image
CN104698749B (zh) *	2010-01-25	2019-11-19	罗门哈斯电子材料有限公司	包含含氮化合物的光致抗蚀剂
CN103080122A (zh)	2010-03-22	2013-05-01	森普拉制药公司	大环内脂的结晶形式及其用途
US9051346B2 (en)	2010-05-20	2015-06-09	Cempra Pharmaceuticals, Inc.	Process for preparing triazole-containing ketolide antibiotics
JP6042334B2 (ja)	2010-09-10	2016-12-14	センプラファーマシューティカルズ，インコーポレイテッド	疾患治療のための水素結合形成フルオロケトライド
CN104470527B (zh)	2012-03-27	2019-05-28	森普拉制药公司	用于施用大环内酯抗生素的肠胃外制剂
WO2014152326A1 (en)	2013-03-14	2014-09-25	Cempra Pharmaceuticals, Inc.	Methods for treating respiratory diseases and formulations therefor
US9751908B2 (en)	2013-03-15	2017-09-05	Cempra Pharmaceuticals, Inc.	Convergent processes for preparing macrolide antibacterial agents
CN104650166B (zh) *	2014-11-17	2017-12-05	广东东阳光药业有限公司	一种大环内酯的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
KR0166096B1 (ko)	1990-11-28	1999-01-15	우에하라 아키라	6-0-메틸에리쓰로마이신 a 유도체
US5523399A (en)	1991-12-27	1996-06-04	Taisho Pharmaceutical Co., Ltd.	5-O-desosaminylerythronolide derivatives
ATE135707T1 (de)	1992-04-22	1996-04-15	Taisho Pharmaceutical Co Ltd	5-0-desosaminylerythronolid a derivate
JP3227871B2 (ja) *	1993-02-25	2001-11-12	大正製薬株式会社	６−ｏ−メチルエリスロマイシンａ誘導体
PT876388E (pt)	1995-11-08	2004-07-30	Abbott Lab	Derivados de eritromicina triciclica

1997
- 1997-01-07 US US08/779,786 patent/US6274715B1/en not_active Expired - Lifetime
- 1997-04-07 KR KR1019997006148A patent/KR20000069935A/ko not_active Application Discontinuation
- 1997-04-07 CZ CZ992315A patent/CZ231599A3/cs unknown
- 1997-04-07 JP JP53082898A patent/JP2001507714A/ja not_active Ceased
- 1997-04-07 EP EP97920261A patent/EP0961776A1/en not_active Withdrawn
- 1997-04-07 AU AU24495/97A patent/AU2449597A/en not_active Abandoned
- 1997-04-07 HU HU0001518A patent/HUP0001518A3/hu unknown
- 1997-04-07 NZ NZ336174A patent/NZ336174A/en unknown
- 1997-04-07 CA CA002277116A patent/CA2277116A1/en not_active Abandoned
- 1997-04-07 BR BR9714269-7A patent/BR9714269A/pt not_active IP Right Cessation
- 1997-04-07 IL IL13032897A patent/IL130328A0/xx unknown
- 1997-04-07 WO PCT/US1997/005871 patent/WO1998030574A1/en not_active Application Discontinuation
- 1997-04-07 CN CN97181288A patent/CN1244202A/zh active Pending
- 1997-04-14 TW TW086104775A patent/TW442490B/zh not_active IP Right Cessation
- 1997-04-16 AR ARP970101538A patent/AR006678A1/es unknown

Also Published As

Publication number	Publication date
CA2277116A1 (en)	1998-07-16
KR20000069935A (ko)	2000-11-25
CN1244202A (zh)	2000-02-09
CZ231599A3 (cs)	1999-12-15
AU2449597A (en)	1998-08-03
HUP0001518A2 (hu)	2000-09-28
IL130328A0 (en)	2000-06-01
AR006678A1 (es)	1999-09-08
TW442490B (en)	2001-06-23
EP0961776A1 (en)	1999-12-08
US6274715B1 (en)	2001-08-14
JP2001507714A (ja)	2001-06-12
NZ336174A (en)	2001-02-23
BR9714269A (pt)	2000-04-18
WO1998030574A1 (en)	1998-07-16

Publication	Publication Date	Title
IL130328A0 (en)	2000-06-01	Tricyclic erythromycin derivatives
HRP970346A2 (en)	1998-06-30	Phenylamino-substituted tricyclic derivatives
EG24081A (en)	2008-05-11	4-Substituted-9-deoxo-9a-aza-9a-homerythromycin derivatives
PL348210A1 (en)	2002-05-06	Tricyclic pyrazole derivatives
GB9702194D0 (en)	1997-03-26	Sulphonide derivatives
AU9277698A (en)	1999-05-17	9-amino-3-keto erythromycin derivatives
HUP0100566A3 (en)	2003-07-28	Novel erythromycin derivatives
IL132767A0 (en)	2001-03-19	9-Oxime erythromycin derivatives
HUP0004282A3 (en)	2001-10-29	2-halo-6-0-substituted ketolide derivatives
ZA987688B (en)	1999-02-24	6,9-bridged erythromycin derivatives
IL134996A0 (en)	2001-05-20	6,11-bridged erythromycin derivatives
AU9277398A (en)	1999-05-17	Tricyclic erythromycin derivatives
AU8925398A (en)	1999-03-22	3-descladinose 6-o-substituded erythromycin derivatives
GB9715821D0 (en)	1997-10-01	Amidino-camptothecin derivatives
GB2321457B (en)	2001-02-28	5-Aroylnaphthalene derivatives
ZA983902B (en)	1999-11-08	Erythromycin derivatives.
EP1044985A4 (en)	2001-04-18	ERYTHROMYCIN DERIVATIVES
GB9725541D0 (en)	1998-02-04	Amino-benzothiazole derivatives
GB9701628D0 (en)	1997-03-19	Imino-aza-anthracyclinone derivatives
PL337066A1 (en)	2000-07-31	Polycyclic derivatives of erythromycin
GB9700702D0 (en)	1997-03-05	Erythromycin derivatives
ZA973362B (en)	1997-11-18	Tricyclic erythromycin derivatives.
GB9706753D0 (en)	1997-05-21	Aralkoxy-morphinan derivatives
ZA951845B (en)	1996-03-15	Acid-stabile erythromycin derivatives
ZA989845B (en)	1999-04-29	2-halo-6-O-substituted ketolide derivatives