HN2001000244A - SPIROPIRIMIDIN INHIBITORS - 2, 4, 6 - TRIONA METALOPROTEINASAS. - Google Patents
SPIROPIRIMIDIN INHIBITORS - 2, 4, 6 - TRIONA METALOPROTEINASAS.Info
- Publication number
- HN2001000244A HN2001000244A HN2001000244A HN2001000244A HN2001000244A HN 2001000244 A HN2001000244 A HN 2001000244A HN 2001000244 A HN2001000244 A HN 2001000244A HN 2001000244 A HN2001000244 A HN 2001000244A HN 2001000244 A HN2001000244 A HN 2001000244A
- Authority
- HN
- Honduras
- Prior art keywords
- metaloproteinasas
- triona
- inhibitors
- spiropirimidin
- spiropririmidin
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A61P11/06—Antiasthmatics
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- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
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Abstract
LA PRESENTE INVENCION SE REFIERE A INHIBIDORES DE 5 - ESPIROPIRIMIDIN - 2, 4, 6 - TRIONA METALOPROTEINASAS Y A COMPOSICIONES FARMACEUTICAS Y PROCEDIMIENTOS DE TRATAMIENTO DE LA INFLAMACION, EL CANCER Y OTRAS DOLENCIAS.THE PRESENT INVENTION REFERS TO INHIBITORS OF 5 - SPIROPRIRIMIDIN - 2, 4, 6 - TRIONA METALOPROTEINASAS AND PHARMACEUTICAL COMPOSITIONS AND PROCEDURES OF TREATMENT OF INFLAMMATION, CANCER AND OTHER DOLENCES.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US24338900P | 2000-10-26 | 2000-10-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
HN2001000244A true HN2001000244A (en) | 2003-11-07 |
Family
ID=22918584
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HN2001000244A HN2001000244A (en) | 2000-10-26 | 2001-10-24 | SPIROPIRIMIDIN INHIBITORS - 2, 4, 6 - TRIONA METALOPROTEINASAS. |
Country Status (32)
Country | Link |
---|---|
EP (1) | EP1332146A2 (en) |
JP (1) | JP2004518635A (en) |
KR (1) | KR20040004412A (en) |
CN (1) | CN1501937A (en) |
AP (1) | AP2001002318A0 (en) |
AR (1) | AR035069A1 (en) |
AU (1) | AU2002210813A1 (en) |
BG (1) | BG107653A (en) |
BR (1) | BR0114913A (en) |
CA (1) | CA2425283A1 (en) |
CZ (1) | CZ20031083A3 (en) |
EA (1) | EA005762B1 (en) |
EC (1) | ECSP034567A (en) |
EE (1) | EE200300196A (en) |
GT (1) | GT200100213A (en) |
HN (1) | HN2001000244A (en) |
HR (1) | HRP20030332A2 (en) |
HU (1) | HUP0301577A3 (en) |
IL (1) | IL154948A0 (en) |
IS (1) | IS6762A (en) |
MA (1) | MA26957A1 (en) |
MX (1) | MXPA03003735A (en) |
NO (1) | NO20031853L (en) |
OA (1) | OA12529A (en) |
PA (1) | PA8531401A1 (en) |
PE (1) | PE20020589A1 (en) |
PL (1) | PL366201A1 (en) |
SK (1) | SK4972003A3 (en) |
SV (1) | SV2003000705A (en) |
TN (1) | TNSN01149A1 (en) |
WO (1) | WO2002034753A2 (en) |
ZA (1) | ZA200302190B (en) |
Families Citing this family (36)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DOP2002000333A (en) | 2001-02-14 | 2002-09-30 | Warner Lambert Co | DERIVATIVES OF ISOFTALIC ACID AS INHIBITORS OF METALOPROTEINASES OF THE MATRIX |
DOP2002000332A (en) | 2001-02-14 | 2002-08-30 | Warner Lambert Co | MATRIX METALOPROTEINAS PYRIDINE INHIBITORS |
DE60236851D1 (en) | 2001-02-14 | 2010-08-12 | Warner Lambert Co | Pyrimidinmatrixmetalloproteinaseinhibitoren |
PA8539501A1 (en) | 2001-02-14 | 2002-09-30 | Warner Lambert Co | TRIAZOLO COMPOUNDS AS MMP INHIBITORS |
ES2231708T3 (en) | 2001-02-14 | 2005-05-16 | Warner-Lambert Company Llc | METALOPROTEINASA MATRIX INHIBITING BENZOTIADICINES. |
US6924276B2 (en) | 2001-09-10 | 2005-08-02 | Warner-Lambert Company | Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors |
US6962922B2 (en) | 2001-10-12 | 2005-11-08 | Warner-Lambert Company Llc | Alkynylated quinazoline compounds |
WO2003032999A1 (en) | 2001-10-12 | 2003-04-24 | Warner-Lambert Company Llc | Alkyne matrix metalloproteinase inhibitors |
US6894057B2 (en) | 2002-03-08 | 2005-05-17 | Warner-Lambert Company | Oxo-azabicyclic compounds |
AU2003228701A1 (en) * | 2002-04-25 | 2003-11-10 | Bristol-Myers Squibb Company | Spirobarbituric acid derivatives useful as inhibitors of matrix metalloproteases |
CA2480092A1 (en) * | 2002-04-26 | 2003-11-06 | Pfizer Products Inc. | N-substituted-heteroaryloxy-aryl-spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors |
ATE304015T1 (en) * | 2002-04-26 | 2005-09-15 | Pfizer Prod Inc | TRIARYL-OXY-ARYL-SPIRO-PYRIMIDINE-2, 4, 6-TRION METALLOPROTEINASE INHIBITORS |
AU2003249531A1 (en) | 2002-08-13 | 2004-02-25 | Warner-Lambert Company Llc | Azaisoquinoline derivatives as matrix metalloproteinase inhibitors |
AU2003250466A1 (en) | 2002-08-13 | 2004-02-25 | Warner-Lambert Company Llc | 3-isoquinolinone derivatives as matrix metalloproteinase inhiitors |
EP1553949B1 (en) | 2002-08-13 | 2007-04-18 | Warner-Lambert Company LLC | Pyrimidine-2,4-dione derivatives as matrix metalloproteinase inhibitors |
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