HK1125631A1 - Benzazole derivatives, compositions, and methods of use as aurora kinase inhibitors - Google Patents
Benzazole derivatives, compositions, and methods of use as aurora kinase inhibitorsInfo
- Publication number
- HK1125631A1 HK1125631A1 HK09104027.0A HK09104027A HK1125631A1 HK 1125631 A1 HK1125631 A1 HK 1125631A1 HK 09104027 A HK09104027 A HK 09104027A HK 1125631 A1 HK1125631 A1 HK 1125631A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- compositions
- methods
- kinase inhibitors
- aurora kinase
- benzazole derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US77249706P | 2006-02-10 | 2006-02-10 | |
| US79118706P | 2006-04-11 | 2006-04-11 | |
| PCT/US2007/003579 WO2007095124A2 (en) | 2006-02-10 | 2007-02-09 | Benzazole derivatives, compositions, and methods of use as aurora kinase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HK1125631A1 true HK1125631A1 (en) | 2009-08-14 |
Family
ID=38157823
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HK09104027.0A HK1125631A1 (en) | 2006-02-10 | 2009-04-30 | Benzazole derivatives, compositions, and methods of use as aurora kinase inhibitors |
Country Status (10)
| Country | Link |
|---|---|
| US (2) | US7820821B2 (xx) |
| EP (2) | EP1987028A2 (xx) |
| JP (1) | JP5188988B2 (xx) |
| CN (2) | CN101379060B (xx) |
| AU (1) | AU2007215247B2 (xx) |
| BR (1) | BRPI0708034A2 (xx) |
| CA (1) | CA2641744C (xx) |
| HK (1) | HK1125631A1 (xx) |
| IL (1) | IL192580A0 (xx) |
| WO (1) | WO2007095124A2 (xx) |
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| AU2006223070B2 (en) * | 2005-03-14 | 2012-02-09 | High Point Pharmaceuticals, Llc | Benzazole derivatives, compositions, and methods of use as B-secretase inhibitors |
| JP5193876B2 (ja) * | 2005-12-02 | 2013-05-08 | バイエル・ヘルスケア・エルエルシー | オーロラキナーゼの阻害により癌を処置するために有用なピロロトリアジン誘導体 |
-
2007
- 2007-02-09 BR BRPI0708034-4A patent/BRPI0708034A2/pt not_active IP Right Cessation
- 2007-02-09 EP EP07750418A patent/EP1987028A2/en not_active Withdrawn
- 2007-02-09 CN CN2007800047858A patent/CN101379060B/zh not_active Expired - Fee Related
- 2007-02-09 US US11/704,431 patent/US7820821B2/en not_active Expired - Fee Related
- 2007-02-09 CA CA2641744A patent/CA2641744C/en not_active Expired - Fee Related
- 2007-02-09 JP JP2008554398A patent/JP5188988B2/ja not_active Expired - Fee Related
- 2007-02-09 AU AU2007215247A patent/AU2007215247B2/en not_active Ceased
- 2007-02-09 WO PCT/US2007/003579 patent/WO2007095124A2/en active Application Filing
- 2007-02-09 CN CN2012101215887A patent/CN102633783A/zh active Pending
- 2007-02-09 EP EP10194622A patent/EP2295432A1/en not_active Withdrawn
-
2008
- 2008-07-02 IL IL192580A patent/IL192580A0/en unknown
-
2009
- 2009-04-30 HK HK09104027.0A patent/HK1125631A1/xx not_active IP Right Cessation
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2010
- 2010-02-10 US US12/703,604 patent/US8377983B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| AU2007215247B2 (en) | 2012-12-13 |
| CA2641744A1 (en) | 2007-08-23 |
| CN101379060A (zh) | 2009-03-04 |
| EP2295432A1 (en) | 2011-03-16 |
| BRPI0708034A2 (pt) | 2011-05-17 |
| WO2007095124A2 (en) | 2007-08-23 |
| CN101379060B (zh) | 2012-05-23 |
| JP2009526072A (ja) | 2009-07-16 |
| US7820821B2 (en) | 2010-10-26 |
| CN102633783A (zh) | 2012-08-15 |
| IL192580A0 (en) | 2009-02-11 |
| CA2641744C (en) | 2012-09-25 |
| JP5188988B2 (ja) | 2013-04-24 |
| US8377983B2 (en) | 2013-02-19 |
| US20070219235A1 (en) | 2007-09-20 |
| US20100152170A1 (en) | 2010-06-17 |
| WO2007095124A3 (en) | 2007-11-01 |
| EP1987028A2 (en) | 2008-11-05 |
| AU2007215247A1 (en) | 2007-08-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PC | Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee) |
Effective date: 20170209 |