AU2001264872A1 - Method for synthesis of substituted azole libraries - Google Patents
Method for synthesis of substituted azole librariesInfo
- Publication number
- AU2001264872A1 AU2001264872A1 AU2001264872A AU6487201A AU2001264872A1 AU 2001264872 A1 AU2001264872 A1 AU 2001264872A1 AU 2001264872 A AU2001264872 A AU 2001264872A AU 6487201 A AU6487201 A AU 6487201A AU 2001264872 A1 AU2001264872 A1 AU 2001264872A1
- Authority
- AU
- Australia
- Prior art keywords
- libraries
- synthesis
- substituted azole
- azole
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- KAESVJOAVNADME-UHFFFAOYSA-N 1H-pyrrole Natural products C=1C=CNC=1 KAESVJOAVNADME-UHFFFAOYSA-N 0.000 title 1
- 150000003851 azoles Chemical class 0.000 title 1
- 230000015572 biosynthetic process Effects 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 238000003786 synthesis reaction Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D277/24—Radicals substituted by oxygen atoms
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US20925200P | 2000-06-05 | 2000-06-05 | |
| US60209252 | 2000-06-05 | ||
| US60/209,252 | 2000-06-05 | ||
| PCT/US2001/016727 WO2001094318A2 (en) | 2000-06-05 | 2001-05-22 | Method for synthesis of substituted azole libraries |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2001264872A1 true AU2001264872A1 (en) | 2001-12-17 |
Family
ID=22778010
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2001264872A Abandoned AU2001264872A1 (en) | 2000-06-05 | 2001-05-22 | Method for synthesis of substituted azole libraries |
Country Status (3)
| Country | Link |
|---|---|
| US (1) | US6951948B2 (en) |
| AU (1) | AU2001264872A1 (en) |
| WO (1) | WO2001094318A2 (en) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003099760A1 (en) | 2002-05-22 | 2003-12-04 | Errant Gene Therapeutics, Llc. | Histone deacetylase inhibitors based on trihalomethylcarbonyl compounds |
| AU2004251987C1 (en) * | 2003-06-30 | 2010-11-18 | Daiichi Sankyo Company, Limited | Heterocyclic methyl sulfone derivative |
| ATE443701T1 (en) * | 2004-01-16 | 2009-10-15 | Wyeth Corp | HETEROCYCLIC AZOLE-CONTAINING SULFONAMIDINE INHIBITORS OF BETA-AMYLOID PRODUCTION |
| US7541472B2 (en) | 2004-05-24 | 2009-06-02 | Cropsolution, Inc. | 3-Aryl-3-hydroxy-2-methylenepropionic acid esters as fungicides |
| NZ552510A (en) | 2004-06-18 | 2010-12-24 | Novartis Vaccines & Diagnostic | N-(1-(1-benzyl-4-phenyl-1H-imidazol-2-yl)-2,2-dimethylpropyl) benzamide derivatives and related compounds as kinesin spindle protein (KSP) inhibitors for the treatment of cancer |
| EP1757290A1 (en) | 2005-08-16 | 2007-02-28 | Zentaris GmbH | Novel triazole derivatives as ghrelin analogue ligands of growth hormone secretagogue receptors |
| US7592362B2 (en) * | 2006-01-19 | 2009-09-22 | Pfizer Limited | Substituted imidazoles |
| AU2007215247B2 (en) * | 2006-02-10 | 2012-12-13 | Transtech Pharma, Llc | Benzazole derivatives, compositions, and methods of use as Aurora kinase inhibitors |
| US7448642B2 (en) * | 2006-04-11 | 2008-11-11 | Honda Motor Co., Ltd. | Impact absorbing airbag inflator |
| MX2009007260A (en) | 2007-01-05 | 2009-07-10 | Novartis Ag | Cyclized derivatives as eg-5 inhibitors. |
| EP2431035A1 (en) | 2010-09-16 | 2012-03-21 | Æterna Zentaris GmbH | Novel Triazole Derivatives with Improved Receptor Activity and Bioavailability Properties as Ghrelin Antagonists of Growth Hormone Secretagogue Receptors |
| WO2020059841A1 (en) * | 2018-09-21 | 2020-03-26 | 国立大学法人 長崎大学 | Therapeutic agent for prion diseases |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2207088A1 (en) | 1996-06-14 | 1997-12-14 | Eli Lilly And Company | Scavenger assisted combinatorial process for preparing libraries of tertiary amine compounds |
| AU1455500A (en) * | 1998-10-29 | 2000-05-22 | Trega Biosciences, Inc. | Oxadiazole, thiadiazole and triazole derivatives and combinatorial libraries thereof |
-
2001
- 2001-05-22 AU AU2001264872A patent/AU2001264872A1/en not_active Abandoned
- 2001-05-22 US US09/862,808 patent/US6951948B2/en not_active Expired - Lifetime
- 2001-05-22 WO PCT/US2001/016727 patent/WO2001094318A2/en active Application Filing
Also Published As
| Publication number | Publication date |
|---|---|
| US20020042520A1 (en) | 2002-04-11 |
| WO2001094318A2 (en) | 2001-12-13 |
| US6951948B2 (en) | 2005-10-04 |
| WO2001094318A3 (en) | 2002-07-18 |
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