HK1112895A1 - 5-heteroaryl thiazoles and their use as pi3k inhibitors - Google Patents

5-heteroaryl thiazoles and their use as pi3k inhibitors

Info

Publication number
HK1112895A1
HK1112895A1 HK08101781.3A HK08101781A HK1112895A1 HK 1112895 A1 HK1112895 A1 HK 1112895A1 HK 08101781 A HK08101781 A HK 08101781A HK 1112895 A1 HK1112895 A1 HK 1112895A1
Authority
HK
Hong Kong
Prior art keywords
pi3k inhibitors
thiazoles
heteroaryl
heteroaryl thiazoles
pi3k
Prior art date
Application number
HK08101781.3A
Other languages
English (en)
Inventor
Malena Bengtsson
Joakim Larsson
Grigorios Nikitidis
Peter Storm
John Peter Bailey
Edward Jolyon Griffen
Jean-Claude Arnould
Thomas Geoffrey Colerick Bird
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of HK1112895A1 publication Critical patent/HK1112895A1/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
HK08101781.3A 2004-11-09 2008-02-19 5-heteroaryl thiazoles and their use as pi3k inhibitors HK1112895A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0402735A SE0402735D0 (sv) 2004-11-09 2004-11-09 Novel compounds
PCT/GB2005/004268 WO2006051270A1 (en) 2004-11-09 2005-11-07 5-heteroaryl thiazoles and their use as p13k inhibitors

Publications (1)

Publication Number Publication Date
HK1112895A1 true HK1112895A1 (en) 2008-09-19

Family

ID=33488202

Family Applications (1)

Application Number Title Priority Date Filing Date
HK08101781.3A HK1112895A1 (en) 2004-11-09 2008-02-19 5-heteroaryl thiazoles and their use as pi3k inhibitors

Country Status (21)

Country Link
US (1) US7868188B2 (xx)
EP (1) EP1841763B1 (xx)
JP (1) JP2008519021A (xx)
KR (1) KR20070085837A (xx)
CN (1) CN101098869A (xx)
AR (1) AR052232A1 (xx)
AT (1) ATE472546T1 (xx)
AU (1) AU2005303566A1 (xx)
BR (1) BRPI0517634A (xx)
CA (1) CA2585310A1 (xx)
DE (1) DE602005022116D1 (xx)
ES (1) ES2346333T3 (xx)
HK (1) HK1112895A1 (xx)
IL (1) IL182726A0 (xx)
MX (1) MX2007005546A (xx)
NO (1) NO20072259L (xx)
SE (1) SE0402735D0 (xx)
TW (1) TW200621762A (xx)
UY (1) UY29199A1 (xx)
WO (1) WO2006051270A1 (xx)
ZA (1) ZA200703714B (xx)

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BRPI0611029A2 (pt) 2005-05-24 2010-08-10 Serono Lab derivados de tiazol e uso dos mesmos
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JP5520831B2 (ja) 2007-12-19 2014-06-11 アムジエン・インコーポレーテツド Ｐｉ３キナーゼの阻害薬
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