FR2449090A1 - Nouveaux derives d'acide penicillanique utiles notamment comme antibiotiques et leurs procedes de preparation - Google Patents

Nouveaux derives d'acide penicillanique utiles notamment comme antibiotiques et leurs procedes de preparation

Info

Publication number
FR2449090A1
FR2449090A1 FR8003062A FR8003062A FR2449090A1 FR 2449090 A1 FR2449090 A1 FR 2449090A1 FR 8003062 A FR8003062 A FR 8003062A FR 8003062 A FR8003062 A FR 8003062A FR 2449090 A1 FR2449090 A1 FR 2449090A1
Authority
FR
France
Prior art keywords
penicillanic acid
antibiotics
processes
preparation
acid derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR8003062A
Other languages
English (en)
Other versions
FR2449090B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SARATH
Original Assignee
SARATH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SARATH filed Critical SARATH
Publication of FR2449090A1 publication Critical patent/FR2449090A1/fr
Application granted granted Critical
Publication of FR2449090B1 publication Critical patent/FR2449090B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D503/00—Heterocyclic compounds containing 4-oxa-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxapenicillins, clavulanic acid derivatives; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

LES NOUVEAUX COMPOSES SONT DES DERIVES D'ACIDE PENICILLANIQUE DE FORMULE GENERALE: (CF DESSIN DANS BOPI) DANS LAQUELLE R REPRESENTE UN RESTE AZACYCLOALKYLE OU AZABICYCLOALKYLE A 5-10 CHAINONS, RELIE PAR L'ATOME D'AZOTE ET FACULTATIVEMENT SUBSTITUE PAR UN OU DEUX GROUPES ALKYLE INFERIEUR IDENTIQUES OU DIFFERENTS; R REPRESENTE UN ATOME D'HYDROGENE OU UN RADICAL ALKYLE INFERIEUR, ARYLE OU ARYLALKYLE; A REPRESENTE UN RADICAL D'UN INHIBITEUR DE B-LACTAMASE CONTENANT UN NOYAU B-LACTAME AINSI QU'UN GROUPE CARBOXY, A ETANT RELIE PAR LE GROUPE CARBOXY; ET LEURS SELS D'ADDITION D'ACIDE.
FR8003062A 1979-02-13 1980-02-12 Nouveaux derives d'acide penicillanique utiles notamment comme antibiotiques et leurs procedes de preparation Granted FR2449090A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7905021 1979-02-13
GB7921342 1979-06-19

Publications (2)

Publication Number Publication Date
FR2449090A1 true FR2449090A1 (fr) 1980-09-12
FR2449090B1 FR2449090B1 (fr) 1983-07-29

Family

ID=26270553

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8003062A Granted FR2449090A1 (fr) 1979-02-13 1980-02-12 Nouveaux derives d'acide penicillanique utiles notamment comme antibiotiques et leurs procedes de preparation

Country Status (35)

Country Link
US (1) US4325960A (fr)
AR (1) AR230640A1 (fr)
AT (1) AT370106B (fr)
AU (1) AU532244B2 (fr)
CA (1) CA1144540A (fr)
CH (1) CH646176A5 (fr)
CS (1) CS236766B2 (fr)
CU (1) CU35227A (fr)
CY (1) CY1206A (fr)
DD (1) DD149528A5 (fr)
DE (1) DE3005220A1 (fr)
DK (1) DK59380A (fr)
ES (1) ES488493A0 (fr)
FI (1) FI71741C (fr)
FR (1) FR2449090A1 (fr)
GB (1) GB2045746B (fr)
GR (1) GR73697B (fr)
HK (1) HK5784A (fr)
HU (1) HU182663B (fr)
IE (1) IE49371B1 (fr)
IL (1) IL59257A (fr)
IT (1) IT1128361B (fr)
KE (1) KE3308A (fr)
LU (1) LU82163A1 (fr)
MA (1) MA18732A1 (fr)
MY (1) MY8500007A (fr)
NL (1) NL8000881A (fr)
NZ (1) NZ192776A (fr)
PH (1) PH16933A (fr)
PL (1) PL127413B1 (fr)
PT (1) PT70806A (fr)
SE (1) SE446187B (fr)
SG (1) SG43683G (fr)
SU (1) SU1015830A3 (fr)
YU (1) YU42098B (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2520362A1 (fr) * 1982-01-26 1983-07-29 Rech Applic Therapeutiq Nouveaux composes de type b-lactame, y compris leurs sels formes avec des acides ou des bases acceptables en pharmacie, procedes pour produire ces composes, medicaments les contenant et leur utilisation pour combattre les maladies infectieuses

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU77362A1 (fr) * 1977-05-17 1979-01-19
US4364957A (en) * 1979-09-26 1982-12-21 Pfizer Inc. Bis-esters of alkanediols as antibacterial agents
US4393001A (en) * 1981-03-23 1983-07-12 Pfizer Inc. Intermediates for production of 1,1-dioxopenicillanoyloxymethyl 6-(2-amino-2-phenylacetamido)penicillanates
ES2220789T3 (es) * 2000-10-30 2004-12-16 Lupin Limited Composicion de cefuroxima axetilo de liberacion lenta que se desintegra rapidamente.

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2135339A1 (fr) * 1971-05-05 1972-12-15 Sarath
FR2346355A1 (fr) * 1976-03-30 1977-10-28 Sarath Nouveaux amoxycillinates d'amidinopenicillanoyloxyalkyle et leurs procedes de preparation

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3957764A (en) * 1969-11-11 1976-05-18 Lovens Kemiske Fabrik Produktionsaktieselskab 6-aminopenicillanic acid derivatives
US4089963A (en) * 1972-03-13 1978-05-16 Astra Pharmaceutical Products, Inc. Esters of amidinopenicillanic acids, pharmaceutical preparations and method for treating infectious diseases

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2135339A1 (fr) * 1971-05-05 1972-12-15 Sarath
FR2346355A1 (fr) * 1976-03-30 1977-10-28 Sarath Nouveaux amoxycillinates d'amidinopenicillanoyloxyalkyle et leurs procedes de preparation

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2520362A1 (fr) * 1982-01-26 1983-07-29 Rech Applic Therapeutiq Nouveaux composes de type b-lactame, y compris leurs sels formes avec des acides ou des bases acceptables en pharmacie, procedes pour produire ces composes, medicaments les contenant et leur utilisation pour combattre les maladies infectieuses

Also Published As

Publication number Publication date
GB2045746B (en) 1983-05-11
DE3005220A1 (de) 1980-08-21
AU5540080A (en) 1980-08-21
CH646176A5 (de) 1984-11-15
LU82163A1 (fr) 1980-09-24
IE800170L (en) 1980-08-13
FI800412A (fi) 1980-08-14
DD149528A5 (de) 1981-07-15
GB2045746A (en) 1980-11-05
ATA61680A (de) 1982-07-15
AT370106B (de) 1983-03-10
IT8067207A0 (it) 1980-02-12
ES8101595A1 (es) 1980-12-16
FI71741C (fi) 1987-02-09
SE446187B (sv) 1986-08-18
US4325960A (en) 1982-04-20
CA1144540A (fr) 1983-04-12
NL8000881A (nl) 1980-08-15
SU1015830A3 (ru) 1983-04-30
FR2449090B1 (fr) 1983-07-29
YU35980A (en) 1983-04-30
YU42098B (en) 1988-04-30
NZ192776A (en) 1984-09-28
IL59257A (en) 1983-09-30
KE3308A (en) 1983-08-19
PH16933A (en) 1984-04-17
CS236766B2 (en) 1985-05-15
MY8500007A (en) 1985-12-31
MA18732A1 (fr) 1980-10-01
IT1128361B (it) 1986-05-28
IL59257A0 (en) 1980-05-30
FI71741B (fi) 1986-10-31
HK5784A (en) 1984-01-20
PL221963A1 (fr) 1980-12-01
SE8001100L (sv) 1980-08-14
AU532244B2 (en) 1983-09-22
GR73697B (fr) 1984-04-03
IE49371B1 (en) 1985-09-18
CU35227A (en) 1982-03-28
PT70806A (en) 1980-03-01
HU182663B (en) 1984-02-28
SG43683G (en) 1984-08-03
AR230640A1 (es) 1984-05-31
CY1206A (en) 1983-12-31
PL127413B1 (en) 1983-10-31
DK59380A (da) 1980-08-14
ES488493A0 (es) 1980-12-16

Similar Documents

Publication Publication Date Title
GB9401460D0 (en) Compositions of matter
TNSN87042A1 (fr) Procede de preparation de nouveaux steroides comportant un cycle spirannique en position 17
AU538424B2 (en) Piperazino phenylindane
FR2413369A1 (fr) Procede de preparation de derives de pyridine et nouveaux produits ainsi obtenus
FR2408584A1 (fr) Composes guanidinobenzoiques et possedant une activite antifibrinolysine et antitrypsine et leur procede de preparation
FR2449090A1 (fr) Nouveaux derives d'acide penicillanique utiles notamment comme antibiotiques et leurs procedes de preparation
FR2452486A1 (fr) Nouveaux derives d'a-(3,4-dichlorophenyl)-imidazoline ou pyrimidine-2-methane utiles notamment comme agents antisecretoires et leur procede de preparation
FR2450820A1 (fr) Nouveaux derives d'acides 1- (o-mercaptoacyl) -4,5-dihydropyrazole-5-carboxyliques, utiles notamment comme agents hypotenseurs, et leur procede de preparation
BE904646A (fr) Acide 7-amino-3-propenylcephalosporanique et ses esters.
FR2439774A1 (fr) Nouveaux derives de crysteine utiles notamment comme medicaments pour la suppression des troubles hepatiques et procedes pour leur preparation
DK45987A (da) Thianaphthenderivater, deres fremstilling og anvendelse
ES8701143A1 (es) Un procedimiento para la preparacion de nuevos aminas terciarias.
EP0066909A3 (fr) Dérivés d'imidazole, leurs compositions pharmaceutiques et procédés pour leur préparation
PT87734A (pt) Procede de preparation de nouveaux tripeptides a structure polycyclique azotee et de compositions pharmaceutiques les contenant
FR2449689A1 (fr) Nouveaux derives condenses de pyrrolidine ou de piperidine, leur procede de preparation et leurs applications en therapeutique
FR2455596A1 (fr) Nouveaux antibiotiques presentant une activite antibacterienne, leur procede de production, leur souche servant a leur obtention et les compositions pharmaceutiques les contenant
DK20886D0 (da) Imidazolderivater, deres fremstilling og terapeutiske anvendelse
ES8202332A1 (es) Un metodo para la preparacion de sales de 4'-(9-acridinila- mino)-metanosulfon-m-anisidida
FR2451363A1 (fr) (1,1-biphenyl-2-yl)-propyl- et butylamines, leur preparation et leur utilisation therapeutique
FR2453865A1 (fr) Derives de cephalosporine, leurs procedes de preparation, et medicaments antibacteriens contenant ces derives
ES8705427A1 (es) Un procedimiento para la preparacion de nuevas 3-alcoxi-2-(n-pirrolidino)-n-pirimidinil- o n-pirazinil-propilaminas
FR2456100A1 (fr) Procede pour la preparation de composes du type pyrimidine condensee a tete de pont azotee, leurs sels, hydrates et isomeres, certains representants des composes prepares et compositions pharmaceutiques les contenant
FR2450824A1 (fr) Nouveaux derives d'acides 1-(o-mercaptoacyl)-5-pyrazolidinone-3-carboxyliques, utiles notamment comme agents hypotenseurs
FR2355832A1 (fr) Sels de sulfonium d'esters d'acide acetique substitue et leur application a des compositions biocides
ES8205220A1 (es) Procedimiento para la obtencion de esteres del acido succi- nico de efecto antibacterial y antiprotozoal

Legal Events

Date Code Title Description
TP Transmission of property
ST Notification of lapse