FR2434159A1 - 2,1-benzisothiazoles, leur preparation et leur utilisation therapeutique - Google Patents
2,1-benzisothiazoles, leur preparation et leur utilisation therapeutiqueInfo
- Publication number
- FR2434159A1 FR2434159A1 FR7824614A FR7824614A FR2434159A1 FR 2434159 A1 FR2434159 A1 FR 2434159A1 FR 7824614 A FR7824614 A FR 7824614A FR 7824614 A FR7824614 A FR 7824614A FR 2434159 A1 FR2434159 A1 FR 2434159A1
- Authority
- FR
- France
- Prior art keywords
- benzisothiazoles
- preparation
- therapeutic use
- novel
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
- C07C205/49—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
- C07C205/57—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
- C07C205/58—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton the carbon skeleton being further substituted by halogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
- C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/194—Radicals derived from thio- or thiono carboxylic acids
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Abstract
L'invention concerne de nouveaux 3-(amino substitué)-2,1-benzisothiazoles de formule :
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/793,629 US4112105A (en) | 1977-05-04 | 1977-05-04 | Anti-inflammatory 3-(substituted-amino)-2,1-benzisothiazoles |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2434159A1 true FR2434159A1 (fr) | 1980-03-21 |
FR2434159B1 FR2434159B1 (fr) | 1981-03-06 |
Family
ID=25160405
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7824614A Granted FR2434159A1 (fr) | 1977-05-04 | 1978-08-24 | 2,1-benzisothiazoles, leur preparation et leur utilisation therapeutique |
Country Status (7)
Country | Link |
---|---|
US (2) | US4112105A (fr) |
BE (1) | BE869959A (fr) |
DE (1) | DE2837531A1 (fr) |
FR (1) | FR2434159A1 (fr) |
GB (1) | GB2030977B (fr) |
LU (1) | LU80161A1 (fr) |
NL (1) | NL7808844A (fr) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4452799A (en) * | 1981-12-23 | 1984-06-05 | Mead Johnson & Company | Benzisothiazole and benzisoxazole piperazine derivatives |
US4590196A (en) * | 1984-08-23 | 1986-05-20 | Bristol-Myers Company | Analgesic 1,2-benzisothiazol-3-ylpiperazine derivatives |
US5750542A (en) * | 1993-09-28 | 1998-05-12 | Pfizer | Benzisoxazole and benzisothizole derivatives as cholinesterase inhibitors |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR1435787A (fr) * | 1963-07-22 | 1966-04-22 | Parke Davis & Co | Nouveaux 2, 1-benzisothiazoles et procédés pour leur préparation |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3170955A (en) * | 1958-04-25 | 1965-02-23 | Abbott Lab | Amino and halogen substituted-n-diloweralkylamino-alkyl-benzamides |
DE1670907B2 (de) * | 1967-08-16 | 1976-07-22 | Bayer Ag, 5090 Leverkusen | N-disubstituierte 3-amino-1,2benzisothiazole und verfahren in ihrer herstellung |
-
1977
- 1977-05-04 US US05/793,629 patent/US4112105A/en not_active Expired - Lifetime
-
1978
- 1978-02-15 US US05/877,955 patent/US4152518A/en not_active Expired - Lifetime
- 1978-08-16 GB GB7833557A patent/GB2030977B/en not_active Expired
- 1978-08-24 FR FR7824614A patent/FR2434159A1/fr active Granted
- 1978-08-25 LU LU80161A patent/LU80161A1/fr unknown
- 1978-08-25 BE BE1009028A patent/BE869959A/fr unknown
- 1978-08-28 NL NL7808844A patent/NL7808844A/nl not_active Application Discontinuation
- 1978-08-28 DE DE19782837531 patent/DE2837531A1/de not_active Withdrawn
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR1435787A (fr) * | 1963-07-22 | 1966-04-22 | Parke Davis & Co | Nouveaux 2, 1-benzisothiazoles et procédés pour leur préparation |
Also Published As
Publication number | Publication date |
---|---|
LU80161A1 (fr) | 1979-05-15 |
DE2837531A1 (de) | 1980-03-20 |
NL7808844A (nl) | 1980-03-03 |
US4152518A (en) | 1979-05-01 |
US4112105A (en) | 1978-09-05 |
GB2030977B (en) | 1983-05-11 |
FR2434159B1 (fr) | 1981-03-06 |
GB2030977A (en) | 1980-04-16 |
BE869959A (fr) | 1979-02-26 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |