FR22C1024I2 - Derives de pyridazinone - Google Patents

Derives de pyridazinone

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Publication number
FR22C1024I2
FR22C1024I2 FR22C1024C FR22C1024C FR22C1024I2 FR 22C1024 I2 FR22C1024 I2 FR 22C1024I2 FR 22C1024 C FR22C1024 C FR 22C1024C FR 22C1024 C FR22C1024 C FR 22C1024C FR 22C1024 I2 FR22C1024 I2 FR 22C1024I2
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France
Prior art keywords
pyridazinone derivatives
pyridazinone
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
FR22C1024C
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English (en)
French (fr)
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Merck Patent GmbH
Original Assignee
Merck Patent GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent GmbH filed Critical Merck Patent GmbH
Publication of FR22C1024I1 publication Critical patent/FR22C1024I1/fr
Application granted granted Critical
Publication of FR22C1024I2 publication Critical patent/FR22C1024I2/fr
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50Pyridazines; Hydrogenated pyridazines
    • A61K31/501Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5355Non-condensed oxazines and containing further heterocyclic rings
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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    • A61K9/0031Rectum, anus
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    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
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    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
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    • C07D417/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
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FR22C1024C 2007-07-12 2022-06-02 Derives de pyridazinone Active FR22C1024I2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102007032507A DE102007032507A1 (de) 2007-07-12 2007-07-12 Pyridazinonderivate
PCT/EP2008/003473 WO2009006959A1 (de) 2007-07-12 2008-04-29 Pyridazinonderivate

Publications (2)

Publication Number Publication Date
FR22C1024I1 FR22C1024I1 (fr) 2022-07-22
FR22C1024I2 true FR22C1024I2 (fr) 2023-03-24

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FR22C1024C Active FR22C1024I2 (fr) 2007-07-12 2022-06-02 Derives de pyridazinone

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US (8) US8580781B2 (sl)
EP (3) EP2164843B1 (sl)
JP (2) JP5426543B2 (sl)
KR (2) KR101553418B1 (sl)
CN (2) CN101743241B (sl)
AR (2) AR066543A1 (sl)
AU (2) AU2008274670B2 (sl)
BR (2) BRPI0814616B1 (sl)
CA (2) CA2693600C (sl)
CL (1) CL2008001392A1 (sl)
CO (2) CO6170360A2 (sl)
CY (3) CY1113137T1 (sl)
DE (1) DE102007032507A1 (sl)
DK (3) DK2164843T3 (sl)
EA (2) EA016782B1 (sl)
EC (2) ECSP109953A (sl)
ES (3) ES2614283T3 (sl)
FR (1) FR22C1024I2 (sl)
HK (2) HK1142891A1 (sl)
HR (3) HRP20120661T1 (sl)
HU (2) HUE030519T2 (sl)
IL (2) IL203091A (sl)
LT (2) LT2754660T (sl)
MY (2) MY153727A (sl)
NL (1) NL301176I2 (sl)
NO (1) NO2022015I1 (sl)
NZ (1) NZ583187A (sl)
PE (1) PE20090287A1 (sl)
PL (3) PL2754660T3 (sl)
PT (3) PT2164843E (sl)
SG (1) SG183739A1 (sl)
SI (3) SI2754660T1 (sl)
TW (1) TWI501768B (sl)
UA (2) UA99621C2 (sl)
WO (2) WO2009006959A1 (sl)
ZA (1) ZA201001023B (sl)

Families Citing this family (72)

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Publication number Priority date Publication date Assignee Title
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CN101687857B (zh) 2013-07-17
HK1145265A1 (en) 2011-04-08
FR22C1024I1 (fr) 2022-07-22
AU2008274670B2 (en) 2013-03-14
CA2693600A1 (en) 2009-01-15
EA017281B1 (ru) 2012-11-30
SI2754660T1 (sl) 2017-03-31
PE20090287A1 (es) 2009-03-19
SG183739A1 (en) 2012-09-27
IL203091A (en) 2013-10-31
EP2754660B1 (de) 2016-11-02
SI2164843T1 (sl) 2015-02-27
CL2008001392A1 (es) 2009-01-23
PL2164843T3 (pl) 2015-03-31
BRPI0814616B1 (pt) 2022-04-19
ES2526352T3 (es) 2015-01-09
PL2754660T3 (pl) 2017-05-31
EP2164843B1 (de) 2014-10-29
NZ583187A (en) 2011-10-28
NO2022015I1 (no) 2022-05-13
PT2164843E (pt) 2014-12-23
EA201000094A1 (ru) 2010-06-30
AR066543A1 (es) 2009-08-26
EP2164843A1 (de) 2010-03-24
EP2164844B1 (de) 2012-06-27
ES2388883T3 (es) 2012-10-19
US8658643B2 (en) 2014-02-25
DK2754660T3 (en) 2017-02-13
ECSP109957A (es) 2010-03-31
HUE030519T2 (en) 2017-05-29
ZA201001023B (en) 2010-11-24
US8921357B2 (en) 2014-12-30
ECSP109953A (es) 2010-03-31
BRPI0813707A2 (pt) 2014-12-30
JP2010532774A (ja) 2010-10-14
UA99833C2 (en) 2012-10-10
EP2164844A1 (de) 2010-03-24
DE102007032507A1 (de) 2009-04-02
HRP20150031T1 (en) 2015-03-13
KR20100050504A (ko) 2010-05-13
LTPA2022009I1 (sl) 2022-06-10
US9062029B2 (en) 2015-06-23
BRPI0814616A2 (pt) 2015-01-27
KR101544624B1 (ko) 2015-08-17
MY153727A (en) 2015-03-13
NL301176I1 (sl) 2022-06-01
DK2164843T3 (en) 2014-12-01
JP5426544B2 (ja) 2014-02-26
AU2008274534A1 (en) 2009-01-15
US20120295908A1 (en) 2012-11-22
EA201000093A1 (ru) 2010-06-30
US20130184261A1 (en) 2013-07-18
BRPI0813707B1 (pt) 2022-02-22

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