FI950579A - The process for the preparation of 3- (2- (4- (6-fluorobenzo (N) -isoxazol-3-yl) piperidin-1-yl) ethyl) -2-methyl-6,7,8,9-tetrahydro- 4H-pyrido / 1,2-a / -pyrimidin-4-one - Google Patents

The process for the preparation of 3- (2- (4- (6-fluorobenzo (N) -isoxazol-3-yl) piperidin-1-yl) ethyl) -2-methyl-6,7,8,9-tetrahydro- 4H-pyrido / 1,2-a / -pyrimidin-4-one Download PDF

Info

Publication number: FI950579A
Authority: FI; Finland
Prior art keywords: fluorobenzo; isoxazol; pyrido; pyrimidin; piperidin
Prior art date: 1994-02-11

Application number

FI950579A

Other languages

Finnish (fi)

Swedish (sv)

Other versions

FI950579A0 (en

FI110000B (en

Inventor

Barjoan Pere Dalmases

Olondriz Francisco Marquillas

Clotet Joan Huguet

Rovira Ana Bosch

Castillo Nieto Juan Carlos Del

Ges Jose Maria Caldero

Original Assignee

Vita Invest Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-02-11

Filing date

1995-02-10

Publication date

1995-08-12

1995-02-10 Application filed by Vita Invest Sa filed Critical Vita Invest Sa

1995-02-10 Publication of FI950579A0 publication Critical patent/FI950579A0/en

1995-08-12 Publication of FI950579A publication Critical patent/FI950579A/en

2002-11-15 Application granted granted Critical

2002-11-15 Publication of FI110000B publication Critical patent/FI110000B/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

FI950579A 1994-02-11 1995-02-10 Process for obtaining 3- {2- [4- (6-fluoro-benzo [d] isoxazol-3-yl) piperidin-1-yl] -ethyl} -2-methyl-6,7,8,9-tetrahydro -4H-pyrido [1,2-a] pyrimidine-4-one FI110000B (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
ES9400252		1994-02-11
ES09400252A ES2074966B1 (en)	1994-02-11	1994-02-11	PROCEDURE FOR OBTAINING 3- (2- (4- (6-FLUORO-BENZO (D) ISOXAZOL-3-IL) PIPERIDIN-1-IL) -ETIL) -2-METHYL-6,7,8,9- TETRAHIDRO-4H-PIRIDO- (1,2-A) PIRIMIDIN-4-ONA.

Publications (3)

Publication Number	Publication Date
FI950579A0 FI950579A0 (en)	1995-02-10
FI950579A true FI950579A (en)	1995-08-12
FI110000B FI110000B (en)	2002-11-15

Family

ID=8285178

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI950579A FI110000B (en)	1994-02-11	1995-02-10	Process for obtaining 3- {2- [4- (6-fluoro-benzo [d] isoxazol-3-yl) piperidin-1-yl] -ethyl} -2-methyl-6,7,8,9-tetrahydro -4H-pyrido [1,2-a] pyrimidine-4-one

Country Status (14)

Country	Link
KR (1)	KR100221108B1 (en)
AT (1)	AT405401B (en)
CZ (1)	CZ286398B6 (en)
EG (1)	EG20877A (en)
ES (1)	ES2074966B1 (en)
FI (1)	FI110000B (en)
GR (1)	GR1002344B (en)
HU (1)	HU222110B1 (en)
IS (1)	IS1766B (en)
NO (1)	NO306022B1 (en)
PL (1)	PL181420B1 (en)
PT (1)	PT101654B (en)
RU (1)	RU2123004C1 (en)
SK (1)	SK281752B6 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2101646B1 (en) *	1995-04-12	1998-04-01	Ferrer Int	NEW COMPOUND DERIVED FROM CHROMENE.
ES2144355B1 (en) *	1997-12-30	2001-01-01	Ferrer Int	COMPOUNDS DERIVED FROM THE CHROME.
WO2001085731A1 (en) *	2000-05-05	2001-11-15	Rpg Life Sciences Limited	A PROCESS FOR THE PREPARATION OF ANTI-PSCHOTIC 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2,-a]pyrimidin-4-one
HUP0302874A2 (en)	2000-08-14	2003-12-29	Teva Pharmaceutical Industries Ltd.	Process for preparation of risperidone
KR20040034996A (en)	2002-10-18	2004-04-29	한미약품 주식회사	Improved method for the preparation of risperidone
EP1560814A1 (en)	2002-11-13	2005-08-10	Synthon B.V.	Process for making risperidone and intermediates therefor
RU2459824C2 (en) *	2007-04-19	2012-08-27	Юсинь ЛИ	New compounds for mental disorders, preparing and using them

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4352811A (en) *	1981-11-12	1982-10-05	Hoechst-Roussel Pharmaceuticals Inc.	3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles
US4804663A (en) *	1985-03-27	1989-02-14	Janssen Pharmaceutica N.V.	3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
US4980365A (en) *	1987-07-13	1990-12-25	Hoechst-Roussel Pharmaceuticals Inc.	N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents

1994
- 1994-02-11 ES ES09400252A patent/ES2074966B1/en not_active Expired - Fee Related
1995
- 1995-02-01 GR GR950100035A patent/GR1002344B/en not_active IP Right Cessation
- 1995-02-07 SK SK156-95A patent/SK281752B6/en not_active IP Right Cessation
- 1995-02-08 IS IS4259A patent/IS1766B/en unknown
- 1995-02-08 CZ CZ1995329A patent/CZ286398B6/en not_active IP Right Cessation
- 1995-02-09 EG EG11595A patent/EG20877A/en active
- 1995-02-09 NO NO950501A patent/NO306022B1/en not_active IP Right Cessation
- 1995-02-09 PT PT101654A patent/PT101654B/en active IP Right Grant
- 1995-02-10 FI FI950579A patent/FI110000B/en not_active IP Right Cessation
- 1995-02-10 AT AT0024995A patent/AT405401B/en not_active IP Right Cessation
- 1995-02-10 HU HU9500418A patent/HU222110B1/en not_active IP Right Cessation
- 1995-02-10 RU RU95101859/04A patent/RU2123004C1/en not_active IP Right Cessation
- 1995-02-10 PL PL95307200A patent/PL181420B1/en not_active IP Right Cessation
- 1995-02-11 KR KR1019950002516A patent/KR100221108B1/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
PL181420B1 (en)	2001-07-31
PT101654B (en)	2002-01-30
EG20877A (en)	2000-05-31
CZ286398B6 (en)	2000-04-12
FI950579A0 (en)	1995-02-10
GR1002344B (en)	1996-05-24
HUT70169A (en)	1995-09-28
RU95101859A (en)	1997-03-20
NO950501L (en)	1995-08-14
AT405401B (en)	1999-08-25
HU222110B1 (en)	2003-04-28
PL307200A1 (en)	1995-08-21
CZ32995A3 (en)	1995-09-13
KR950032196A (en)	1995-12-20
ATA24995A (en)	1998-12-15
KR100221108B1 (en)	1999-09-15
IS4259A (en)	1995-08-12
ES2074966B1 (en)	1996-06-16
HU9500418D0 (en)	1995-03-28
NO306022B1 (en)	1999-09-06
ES2074966A1 (en)	1995-09-16
SK15695A3 (en)	1995-10-11
NO950501D0 (en)	1995-02-09
FI110000B (en)	2002-11-15
SK281752B6 (en)	2001-07-10
RU2123004C1 (en)	1998-12-10
PT101654A (en)	1995-09-12
IS1766B (en)	2001-03-15

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Legal Events

Date

Code

Title

Description

2005-05-11

PC

Transfer of assignment of patent

Owner name: VITA CIENTIFICA

Free format text: VITA CIENTIFICA

2007-11-29

PC

Transfer of assignment of patent

Owner name: INKE, S.A.

Free format text: INKE, S.A.

2011-09-28

MM

Patent lapsed