FI931901A - Azolfoereningar, deras framstaellning och anvaendning - Google Patents

Azolfoereningar, deras framstaellning och anvaendning Download PDF

Info

Publication number: FI931901A
Authority: FI; Finland
Prior art keywords: group; following; independently; deras framstaellning; framstaellning och
Prior art date: 1992-04-28

Application number

FI931901A

Other languages

English (en)

Other versions

FI931901A0 (fi

Inventor

Katsumi Itoh

Kenji Okonogi

Norikazu Tamura

Original Assignee

Takeda Chemical Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-04-28

Filing date

1993-04-27

Publication date

1993-10-29

1993-04-27 Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd

1993-04-27 Publication of FI931901A0 publication Critical patent/FI931901A0/fi

1993-10-29 Publication of FI931901A publication Critical patent/FI931901A/fi

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Lubricants (AREA)
Adhesives Or Adhesive Processes (AREA)
Polymerization Catalysts (AREA)
Coloring (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Steroid Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

FI931901A 1992-04-28 1993-04-27 Azolfoereningar, deras framstaellning och anvaendning FI931901A (fi)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP11040092		1992-04-28
JP2262393		1993-02-10

Publications (2)

Publication Number	Publication Date
FI931901A0 FI931901A0 (fi)	1993-04-27
FI931901A true FI931901A (fi)	1993-10-29

Family

ID=26359882

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI931901A FI931901A (fi)	1992-04-28	1993-04-27	Azolfoereningar, deras framstaellning och anvaendning

Country Status (18)

Country	Link
US (2)	US5371101A (fi)
EP (1)	EP0567982B1 (fi)
JP (1)	JP2818097B2 (fi)
KR (1)	KR100257619B1 (fi)
CN (1)	CN1040433C (fi)
AT (1)	ATE167857T1 (fi)
AU (1)	AU655544B2 (fi)
CA (1)	CA2094962A1 (fi)
DE (1)	DE69319380T2 (fi)
DK (1)	DK0567982T3 (fi)
ES (1)	ES2118160T3 (fi)
FI (1)	FI931901A (fi)
HU (2)	HUT64327A (fi)
NO (1)	NO303284B1 (fi)
NZ (1)	NZ247488A (fi)
PH (1)	PH31082A (fi)
SG (1)	SG48939A1 (fi)
TW (1)	TW218017B (fi)

Families Citing this family (52)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
HU212458B (en) *	1993-09-23	1996-06-28	Richter Gedeon Vegyeszet	New silyloxypropane derivatives substituted with triazole or imidazole pharmaceutical compositions containing them and process for producing them
TW297813B (fi) *	1993-09-24	1997-02-11	Takeda Pharm Industry Co Ltd
CA2134417A1 (en) *	1993-12-22	1995-06-23	Katsumi Itoh	Optically active azole derivatives, their production and use
NZ270418A (en) *	1994-02-07	1997-09-22	Eisai Co Ltd	Polycyclic triazole & imidazole derivatives, antifungal compositions
AU682580B2 (en) *	1994-02-25	1997-10-09	Takeda Chemical Industries Ltd.	Injectable emulsions containing antifungal triazole derivatives
US5677464A (en) *	1994-05-31	1997-10-14	Takeda Chemical Industries, Ltd.	Production of optically active triazole compounds and their intermediates
US5639754A (en) *	1994-07-12	1997-06-17	Janssen Pharmaceutica N.V.	Urea and thiourea derivatives of azolones
US5637592A (en) *	1994-07-12	1997-06-10	Janssen Pharmaceutica N.V.	Acyl derivatives of azolones
CA2211458A1 (en) *	1995-02-17	1996-08-22	Kenji Okonogi	Azole compounds, their production and use
TW318841B (fi) *	1995-02-17	1997-11-01	Takeda Pharm Industry Co Ltd
US6060604A (en) *	1995-03-31	2000-05-09	Florida State University	Pharmaceutical compounds comprising polyamines substituted with electron-affinic groups
US5700825A (en) *	1995-03-31	1997-12-23	Florida State University	Radiosensitizing diamines and their pharmaceutical preparations
DE19520597A1 (de) *	1995-06-06	1996-12-12	Bayer Ag	Mercapto-bis-triazole
KR970705560A (ko) *	1995-08-02	1997-10-09	호아껭 우리아치 토렐로	항진균 활성을 갖는 신규한 카르복사미드(new carboxamides with antifungal activity)
PT783501E (pt) *	1995-08-02	2001-04-30	Uriach & Cia Sa J	Derivados de pirimidona com actividade antifungica
ES2120885B1 (es) *	1996-03-15	1999-06-16	Uriach & Cia Sa J	Nuevas tienopirimidonas con actividad antifungica.
ES2107376B1 (es) *	1995-08-02	1998-07-01	Uriach & Cia Sa J	Nuevos derivados de pirimidona con actividad antifungica.
GB9602080D0 (en) *	1996-02-02	1996-04-03	Pfizer Ltd	Pharmaceutical compounds
US6001835A (en) *	1996-04-03	1999-12-14	Merck & Co., Inc.	Inhibitors of farnesyl-protein transferase
JP2000507585A (ja) *	1996-04-03	2000-06-20	メルクエンドカンパニーインコーポレーテッド	ファルネシルタンパク質トランスフェラーゼの阻害剤
WO1998039305A1 (en) *	1997-03-05	1998-09-11	Takeda Chemical Industries, Ltd.	Crystalline form of a bis 1,2,4-triazole compound
US6407129B1 (en)	1997-03-31	2002-06-18	Takeda Chemical Industries, Ltd.	Azole compounds, their production and their use
EP0884311A3 (en) *	1997-06-06	1999-01-27	Takeda Chemical Industries, Ltd.	Triazole Derivatives and their production
US6133485A (en) *	1998-04-15	2000-10-17	Synphar Laboratories, Inc.	Asymmetric synthesis of 2-(2,4-difluorophenyl)-1-heterocycl-1-yl butan-2,3-diols
WO2000018401A1 (fr) *	1998-09-29	2000-04-06	Takeda Chemical Industries, Ltd.	Composition de medicament antimycotique
IN191188B (fi)	2000-03-07	2003-10-04	Ranbaxy Lab Ltd
ES2159488B1 (es) *	2000-03-07	2002-04-16	Uriach & Cia Sa J	Procedimiento para la preparacion de derivados de pirimidona con actividad antifungica.
NZ521241A (en) *	2000-03-07	2004-02-27	Ranbaxy Lab Ltd	Azole compounds as therapeutic agents for fungal infections
US6710049B2 (en)	2000-12-26	2004-03-23	Ranbaxy Laboratories Limited	Azole compounds as anti-fungal agents
CA2439310C (en) *	2001-03-23	2009-09-29	Richter Gedeon Vegyeszeti Gyar Rt.	Process for preparing fluconazole and its crystal modifications
IN191819B (fi) *	2001-07-19	2004-01-03	Ranbaxy Lab Ltd
IN192526B (fi) *	2001-09-25	2004-04-24	Ranbaxy Lab
US7028055B2 (en) *	2002-03-22	2006-04-11	Sun Microsystems, Inc.	Method and apparatus for improving transaction specification by marking application states
CN1628119A (zh) *	2002-04-12	2005-06-15	兰贝克赛实验室有限公司	作为抗真菌剂的2,2,4－三取代的四氢呋喃衍生物
EP1537868B1 (en)	2002-06-18	2011-08-24	Pola Pharma Inc.	Antifungal medicinal compositions
AU2002328176A1 (en) *	2002-08-26	2004-03-11	Ranbaxy Laboratories Limited	Azole derivatives as antifungal agents
KR100572996B1 (ko) *	2003-08-12	2006-04-25	한국화학연구원	불소화 비닐 에테르 측쇄기를 갖는 아졸계 살균제 화합물및 그의 제조방법
JP4954083B2 (ja) *	2004-11-18	2012-06-13	シンタファーマスーティカルズコーポレイション	Ｈｓｐ９０活性を調節するトリアゾール化合物
CN1304376C (zh) *	2005-03-04	2007-03-14	清华大学	一种卤化烷基咪唑型离子液体的制备方法
AU2006279794B2 (en) *	2005-08-12	2011-04-07	Synta Pharmaceuticals Corp.	Pyrazole compounds that modulate HSP90 activity
CA2618628C (en) *	2005-08-18	2014-11-18	Synta Pharmaceuticals Corp.	Triazole compounds that modulate hsp90 activity
EP2034996A2 (en) *	2006-05-25	2009-03-18	Synta Pharmaceuticals Corporation	Triazole compounds that modulate hsp90 activity
EP2032545A2 (en) *	2006-05-25	2009-03-11	Synta Pharmaceuticals Corporation	Compounds that modulate hsp90 activity and methods for identifying same
WO2007139967A2 (en)	2006-05-25	2007-12-06	Synta Pharmaceuticals Corp.	Triazole compounds that modulate hsp90 activity
EP2038262B1 (en) *	2006-05-25	2014-11-12	Synta Pharmaceuticals Corp.	Triazole compounds that modulate hsp90 activity
RU2500679C2 (ru)	2006-08-07	2013-12-10	Палау Фарма, С.А.	Кристаллические противогрибковые соединения
KR20110079776A (ko) *	2006-10-19	2011-07-07	에프. 호프만-라 로슈 아게	당뇨병을 위한 11베타-에이치에스디1 억제제로서의 이미다졸론 및 이미다졸리딘온 유도체
EP2560640A1 (en)	2010-04-19	2013-02-27	Synta Pharmaceuticals Corp.	Cancer therapy using a combination of a hsp90 inhibitory compounds and a egfr inhibitor
CN102824342B (zh) *	2011-06-17	2016-03-30	全哲山	一类用作抗癫痫药的化合物及其可药用盐
CA2853799A1 (en)	2011-11-02	2013-05-10	Synta Pharmaceuticals Corp.	Cancer therapy using a combination of hsp90 inhibitors with topoisomerase i inhibitors
CA2853806C (en)	2011-11-02	2020-07-14	Synta Pharmaceuticals Corp.	Combination therapy of hsp90 inhibitors with platinum-containing agents
CA2854188A1 (en)	2011-11-14	2013-05-23	Synta Pharmaceuticals Corp.	Combination therapy of hsp90 inhibitors with braf inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8306351D0 (en) *	1983-03-08	1983-04-13	Ici Plc	Azole fungicides
DK159205C (da) *	1983-03-16	1991-03-04	Pfizer	Bis(triazol)alkanol-forbindelser, anvendelse af disse, farmaceutiske praeparater og landbrugsfungicider indeholdende disse og fremgangsmaade til behandling af planter eller froe, som har en svampeinfektion
IE58738B1 (en) *	1984-09-05	1993-11-03	Ici Plc	Antifungal azole compounds
NZ223799A (en) *	1987-03-25	1989-12-21	Janssen Pharmaceutica Nv	Azolylmethyl-dioxolanylmethoxyphenyl-piperazinyl-phenyl-triazolones and antimicrobial compositions
NO171272C (no) *	1988-03-04	1993-02-17	Sankyo Co	Analogifremgangsmaate til fremstilling av terapeutisk aktive 1,2,4-triazolforbindelser
DE3837463A1 (de) *	1988-11-04	1990-05-10	Bayer Ag	Substituierte bisazole, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel

1993
- 1993-04-24 TW TW082103176A patent/TW218017B/zh active
- 1993-04-26 NZ NZ247488A patent/NZ247488A/en unknown
- 1993-04-27 DK DK93106772T patent/DK0567982T3/da active
- 1993-04-27 NO NO931533A patent/NO303284B1/no not_active IP Right Cessation
- 1993-04-27 FI FI931901A patent/FI931901A/fi unknown
- 1993-04-27 CA CA002094962A patent/CA2094962A1/en not_active Abandoned
- 1993-04-27 AU AU38221/93A patent/AU655544B2/en not_active Ceased
- 1993-04-27 SG SG1996003901A patent/SG48939A1/en unknown
- 1993-04-27 ES ES93106772T patent/ES2118160T3/es not_active Expired - Lifetime
- 1993-04-27 EP EP93106772A patent/EP0567982B1/en not_active Expired - Lifetime
- 1993-04-27 JP JP5101216A patent/JP2818097B2/ja not_active Expired - Fee Related
- 1993-04-27 AT AT93106772T patent/ATE167857T1/de not_active IP Right Cessation
- 1993-04-27 DE DE69319380T patent/DE69319380T2/de not_active Expired - Fee Related
- 1993-04-28 CN CN93105239A patent/CN1040433C/zh not_active Expired - Fee Related
- 1993-04-28 HU HU9301226A patent/HUT64327A/hu unknown
- 1993-04-28 KR KR1019930007244A patent/KR100257619B1/ko not_active IP Right Cessation
- 1993-04-28 US US08/053,239 patent/US5371101A/en not_active Expired - Fee Related
- 1993-08-30 PH PH46773A patent/PH31082A/en unknown
1994
- 1994-08-19 US US08/293,066 patent/US5466820A/en not_active Expired - Fee Related
1995
- 1995-06-16 HU HU95P/P00243P patent/HU211474A9/hu unknown

Also Published As

Publication number	Publication date
AU655544B2 (en)	1994-12-22
HU211474A9 (en)	1995-11-28
DE69319380T2 (de)	1998-10-29
JP2818097B2 (ja)	1998-10-30
CA2094962A1 (en)	1993-10-29
SG48939A1 (en)	1998-05-18
DE69319380D1 (de)	1998-08-06
US5466820A (en)	1995-11-14
ATE167857T1 (de)	1998-07-15
DK0567982T3 (da)	1999-04-12
TW218017B (fi)	1993-12-21
HUT64327A (en)	1993-12-28
AU3822193A (en)	1993-11-04
HU9301226D0 (en)	1993-07-28
JPH06293740A (ja)	1994-10-21
ES2118160T3 (es)	1998-09-16
CN1040433C (zh)	1998-10-28
NO931533L (no)	1993-10-29
EP0567982A1 (en)	1993-11-03
US5371101A (en)	1994-12-06
NZ247488A (en)	1995-02-24
PH31082A (en)	1998-02-05
EP0567982B1 (en)	1998-07-01
KR940005616A (ko)	1994-03-21
NO931533D0 (no)	1993-04-27
NO303284B1 (no)	1998-06-22
KR100257619B1 (en)	2000-07-01
FI931901A0 (fi)	1993-04-27
CN1079467A (zh)	1993-12-15

Publication	Publication Date	Title
FI931901A0 (fi)	1993-04-27	Azolfoereningar, deras framstaellning och anvaendning
FI944417A (fi)	1995-03-25	Atsoliyhdisteet, niiden valmistus ja käyttö
ES2123873T3 (es)	1999-01-16	Pirrolocarbazol.
AU546388B2 (en)	1985-08-29	;het;-substituted-3-triazolylpropanes
ATE39923T1 (de)	1989-01-15	Triazol-antifungal-mittel.
MX9206930A (es)	1993-06-01	Nuevos compuestos
DK0594329T3 (da)	1998-04-14	Antimikrobielle midler, der omfatter polykvaternære ammoniumforbindelser
MY109672A (en)	1997-04-30	Azole compounds, their production and use
ATE105565T1 (de)	1994-05-15	Pradimicinderivate.
RU93005133A (ru)	1996-02-27	Производные азола, способ их получения, фармацевтическая композиция