ES464642A1 - Procedimiento para la preparacion de formas de preparados deacido 3-n-pirrolidino-4-fenoxi-5-sulfamibenzoico. - Google Patents
Procedimiento para la preparacion de formas de preparados deacido 3-n-pirrolidino-4-fenoxi-5-sulfamibenzoico.Info
- Publication number
- ES464642A1 ES464642A1 ES464642A ES464642A ES464642A1 ES 464642 A1 ES464642 A1 ES 464642A1 ES 464642 A ES464642 A ES 464642A ES 464642 A ES464642 A ES 464642A ES 464642 A1 ES464642 A1 ES 464642A1
- Authority
- ES
- Spain
- Prior art keywords
- pyrrolidino
- phenoxy
- preparations
- active substance
- sulphamyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
Procedimiento para la preparación de formas de preparados de ácido 3-N-pirrolidino-4-fenoxi-5-sulfamilbenzoicocon retardo de liberación dirigidocaracterizado porque se dota a partículas que contienen sustancia activa de recubrimientos que se disuelven en un medio débilmente ácidolos cuales conducen a la liberación de sustancia activa in Vitroen el elemento de paso según Dibbernal cabo de 75 minutos en una solución tampón de pH 55a no más de 25% del contenido de sustancia activa.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19762655331 DE2655331A1 (de) | 1976-12-07 | 1976-12-07 | Zubereitungsformen von 3-n-pyrrolidino-4-phenoxy-5-sulfamyl-benzoesaeure und verfahren zu ihrer herstellung |
Publications (1)
Publication Number | Publication Date |
---|---|
ES464642A1 true ES464642A1 (es) | 1978-09-01 |
Family
ID=5994862
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES464642A Expired ES464642A1 (es) | 1976-12-07 | 1977-12-01 | Procedimiento para la preparacion de formas de preparados deacido 3-n-pirrolidino-4-fenoxi-5-sulfamibenzoico. |
Country Status (15)
Country | Link |
---|---|
JP (1) | JPS5372815A (es) |
AT (1) | AT355216B (es) |
AU (1) | AU513409B2 (es) |
BE (1) | BE861608A (es) |
DE (1) | DE2655331A1 (es) |
DK (1) | DK542877A (es) |
ES (1) | ES464642A1 (es) |
FR (1) | FR2373280A1 (es) |
GB (1) | GB1569018A (es) |
IE (1) | IE46005B1 (es) |
IL (1) | IL53539A0 (es) |
NL (1) | NL7713392A (es) |
NZ (1) | NZ185855A (es) |
PT (1) | PT67370B (es) |
ZA (1) | ZA777204B (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3772091D1 (de) * | 1986-04-29 | 1991-09-19 | Hoechst Roussel Pharma | Schichtenstruktur fuer die verabreichung von chemikalien mit kontrollierter abgaberate. |
SE460947B (sv) * | 1986-08-26 | 1989-12-11 | Lejus Medical Ab | En multiple-unit-dos komposition av l-dopa |
PT812320E (pt) * | 1995-02-22 | 2000-12-29 | Aventis Pharma Ltd | Firetanido amorfo piretanido polimorfo processo para a sua preparacao e sua utilizacao |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IE33874B1 (en) * | 1968-12-24 | 1974-11-27 | Leo Pharm Prod Ltd | New sulphamyl-benzoic acid derivatives |
-
1976
- 1976-12-07 DE DE19762655331 patent/DE2655331A1/de active Pending
-
1977
- 1977-12-01 ES ES464642A patent/ES464642A1/es not_active Expired
- 1977-12-02 NL NL7713392A patent/NL7713392A/xx not_active Application Discontinuation
- 1977-12-05 IL IL53539A patent/IL53539A0/xx unknown
- 1977-12-05 ZA ZA00777204A patent/ZA777204B/xx unknown
- 1977-12-05 NZ NZ185855A patent/NZ185855A/xx unknown
- 1977-12-06 AU AU31274/77A patent/AU513409B2/en not_active Expired
- 1977-12-06 IE IE2474/77A patent/IE46005B1/en unknown
- 1977-12-06 PT PT67370A patent/PT67370B/pt unknown
- 1977-12-06 DK DK542877A patent/DK542877A/da not_active Application Discontinuation
- 1977-12-06 AT AT873777A patent/AT355216B/de not_active IP Right Cessation
- 1977-12-07 BE BE183258A patent/BE861608A/xx unknown
- 1977-12-07 GB GB50915/77A patent/GB1569018A/en not_active Expired
- 1977-12-07 JP JP14619077A patent/JPS5372815A/ja active Pending
- 1977-12-07 FR FR7736876A patent/FR2373280A1/fr active Granted
Also Published As
Publication number | Publication date |
---|---|
NZ185855A (en) | 1979-10-25 |
FR2373280B1 (es) | 1980-06-20 |
PT67370B (de) | 1979-09-20 |
GB1569018A (en) | 1980-06-11 |
NL7713392A (nl) | 1978-06-09 |
ATA873777A (de) | 1979-07-15 |
IE46005B1 (en) | 1983-01-26 |
JPS5372815A (en) | 1978-06-28 |
PT67370A (de) | 1978-01-01 |
AU3127477A (en) | 1979-06-14 |
AT355216B (de) | 1980-02-25 |
FR2373280A1 (fr) | 1978-07-07 |
DE2655331A1 (de) | 1978-06-08 |
AU513409B2 (en) | 1980-11-27 |
BE861608A (fr) | 1978-06-07 |
DK542877A (da) | 1978-06-08 |
ZA777204B (en) | 1978-10-25 |
IE46005L (en) | 1978-06-07 |
IL53539A0 (en) | 1978-03-10 |
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