ES2058351T3 - Un procedimiento para producir una formulacion de liberacion sostenida que es adecuada para el uso humano y veterinario. - Google Patents

Un procedimiento para producir una formulacion de liberacion sostenida que es adecuada para el uso humano y veterinario.

Info

Publication number
ES2058351T3
ES2058351T3 ES89101428T ES89101428T ES2058351T3 ES 2058351 T3 ES2058351 T3 ES 2058351T3 ES 89101428 T ES89101428 T ES 89101428T ES 89101428 T ES89101428 T ES 89101428T ES 2058351 T3 ES2058351 T3 ES 2058351T3
Authority
ES
Spain
Prior art keywords
producing
human
procedure
release formulation
sustained release
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES89101428T
Other languages
English (en)
Inventor
Keiji Sumitomo Pharmac Fujioka
Shigeji Sumitomo Pharmace Sato
Nobuhiko Sumitomo Pharm Tamura
Yoshihiro Sumitomo Phar Takada
Yoshio C O Sumitomo Pha Sasaki
Miho C O Sumitomo Pharma Maeda
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Koken Co Ltd
Sumitomo Pharmaceuticals Co Ltd
Original Assignee
Koken Co Ltd
Sumitomo Pharmaceuticals Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Koken Co Ltd, Sumitomo Pharmaceuticals Co Ltd filed Critical Koken Co Ltd
Application granted granted Critical
Publication of ES2058351T3 publication Critical patent/ES2058351T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2063Proteins, e.g. gelatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12Carboxylic acids; Salts or anhydrides thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183Amino acids, e.g. glycine, EDTA or aspartame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/42Proteins; Polypeptides; Degradation products thereof; Derivatives thereof, e.g. albumin, gelatin or zein
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats

Abstract

FORMULACION DE LIBERACION CONTROLADA QUE CONTIENE UN COMPUESTO ORGANICO ACIDO O UN ANHIDRIDO DE ACIDO O UN ESTER CAPAZ DE GENERAR UNO DE LOS COMPUESTOS ORGANICOSA ACIDOS POR HIDROLISIS, JUNTO CON UN INGREDIENTE ACTIVO Y COLAGENO COMO VEHICULO, SIENDO DICHA FORMULACION CAPAZ DE EXHIBIR UN PERFIL DE LIBERACION PREDETERMINADO DEL INGREDIENTE ACTIVO. SE INCLUYE UN PROCESO PARA PRODUCIR DICHA FORMULACION.
ES89101428T 1988-01-29 1989-01-27 Un procedimiento para producir una formulacion de liberacion sostenida que es adecuada para el uso humano y veterinario. Expired - Lifetime ES2058351T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2045988 1988-01-29

Publications (1)

Publication Number Publication Date
ES2058351T3 true ES2058351T3 (es) 1994-11-01

Family

ID=12027662

Family Applications (1)

Application Number Title Priority Date Filing Date
ES89101428T Expired - Lifetime ES2058351T3 (es) 1988-01-29 1989-01-27 Un procedimiento para producir una formulacion de liberacion sostenida que es adecuada para el uso humano y veterinario.

Country Status (6)

Country Link
US (1) US5236704A (es)
EP (1) EP0326151B1 (es)
AT (1) ATE90570T1 (es)
CA (1) CA1338839C (es)
DE (1) DE68907066T2 (es)
ES (1) ES2058351T3 (es)

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US20030211095A1 (en) * 2002-05-08 2003-11-13 Abd. Al-Roof Higazi Peptide for regulation of urokinase plasminogen activator and method of optimizing therapeutic efficacy
WO2003066083A1 (fr) * 2002-02-04 2003-08-14 Sumitomo Pharmaceuticals Company, Limited Preparations pour le traitement de fracture osseuse de deperdition osseuse ou d'augmentation la densite osseuse
US7772188B2 (en) 2003-01-28 2010-08-10 Ironwood Pharmaceuticals, Inc. Methods and compositions for the treatment of gastrointestinal disorders
PL1684782T3 (pl) 2003-10-03 2016-03-31 Thorn Bioscience Llc Sposób synchronizacji owulacji dla zsynchronizowanego rozmnażania bez wykrywania rui
EP1682537B1 (en) 2003-11-05 2012-03-28 SARcode Bioscience Inc. Modulators of cellular adhesion
EP1874334A4 (en) * 2005-04-15 2011-03-30 Vascular Biogenics Ltd COMPOSITIONS WITH BETA 2-GLYCOPROTEIN I-PEPTIDES FOR THE PREVENTION AND / OR TREATMENT OF VASCULAR DISEASES
PL2444079T3 (pl) 2005-05-17 2017-07-31 Sarcode Bioscience Inc. Kompozycje i sposoby leczenia chorób oczu
US7718616B2 (en) 2006-12-21 2010-05-18 Zimmer Orthobiologics, Inc. Bone growth particles and osteoinductive composition thereof
US8969514B2 (en) 2007-06-04 2015-03-03 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
CA2688161C (en) 2007-06-04 2020-10-20 Kunwar Shailubhai Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
US20090155176A1 (en) 2007-10-19 2009-06-18 Sarcode Corporation Compositions and methods for treatment of diabetic retinopathy
US20090258069A1 (en) * 2008-04-15 2009-10-15 John Burnier Delivery of LFA-1 antagonists to the gastrointestinal system
WO2009139817A2 (en) 2008-04-15 2009-11-19 Sarcode Corporation Crystalline pharmaceutical and methods of preparation and use thereof
ES2522968T3 (es) 2008-06-04 2014-11-19 Synergy Pharmaceuticals Inc. Agonistas de guanilato ciclasa útiles para el tratamiento de trastornos gastrointestinales, inflamación, cáncer y otros trastornos
ES2624828T3 (es) 2008-07-16 2017-07-17 Synergy Pharmaceuticals Inc. Agonistas de la guanilato ciclasa útiles para el tratamiento de trastornos gastrointestinales, inflamación, cáncer y otros
BRPI1014362A2 (pt) 2009-04-23 2016-04-05 Pennatek Llc método e composição para sincronizar o tempo de inseminação
WO2011050175A1 (en) 2009-10-21 2011-04-28 Sarcode Corporation Crystalline pharmaceutical and methods of preparation and use thereof
US9616097B2 (en) 2010-09-15 2017-04-11 Synergy Pharmaceuticals, Inc. Formulations of guanylate cyclase C agonists and methods of use
JP2013542837A (ja) 2010-11-15 2013-11-28 ジンマー オーソバイオロジクス,インコーポレイティド 骨空隙充填剤
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Also Published As

Publication number Publication date
ATE90570T1 (de) 1993-07-15
EP0326151A3 (en) 1991-03-13
DE68907066T2 (de) 1993-12-16
CA1338839C (en) 1997-01-14
US5236704A (en) 1993-08-17
EP0326151A2 (en) 1989-08-02
EP0326151B1 (en) 1993-06-16
DE68907066D1 (de) 1993-07-22

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