GT199600098A - Formulaciones de quinolona inyectables. - Google Patents
Formulaciones de quinolona inyectables.Info
- Publication number
- GT199600098A GT199600098A GT199600098A GT199600098A GT199600098A GT 199600098 A GT199600098 A GT 199600098A GT 199600098 A GT199600098 A GT 199600098A GT 199600098 A GT199600098 A GT 199600098A GT 199600098 A GT199600098 A GT 199600098A
- Authority
- GT
- Guatemala
- Prior art keywords
- injectable
- complementary
- quinolone
- formulations
- injection
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4995—Pyrazines or piperazines forming part of bridged ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/22—Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Inorganic Chemistry (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Dermatology (AREA)
- Engineering & Computer Science (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Communicable Diseases (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
UNA SOLUCION FARMACEUTICA ACUOSA QUE ES ADECUADA PARA INYECCION EN UN HUESPED, QUE COMPRENDE DANOFLOXACINA O UNA DE SUS SALES FARMACEUTICAMENTE ACEPTABLES EN UNA CANTIDAD SUFICIENTE PARA EL TRATAMIENTO DE INFECCIONES BACTERIANAS Y, (1) UN COMPUESTO DE MAGNESIO O, (2) UN COMPUESTO DE CINC MEZCLADO CON UN DISOLVENTE COMPLEMENTARIO, ESTANDO PRESENTES DICHOS COMPUESTOS Y DICHOS DISOLVENTES COMPLEMENTARIOS EN CANTIDADES QUE SON SUFICIENTES PARA MEJORAR LA TOLERANCIA EN EL SITIO DE LA INYECCION. LA DANOFLOXACINA ES EL ACIDO 1CICLOPROPIL6FLUORO7{(1S, 4S)5METIL2.5DIAZABICICLO [2.2.1] HEPT2IL} 4OXO3QUINOLIN CARBOXILICO.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US905295P | 1995-12-21 | 1995-12-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
GT199600098A true GT199600098A (es) | 1998-06-12 |
Family
ID=21735307
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GT199600098A GT199600098A (es) | 1995-12-21 | 1996-12-19 | Formulaciones de quinolona inyectables. |
Country Status (42)
Country | Link |
---|---|
US (1) | US5811130A (es) |
EP (1) | EP0868183B1 (es) |
JP (1) | JP3416145B2 (es) |
KR (1) | KR100402570B1 (es) |
CN (1) | CN1104899C (es) |
AP (1) | AP706A (es) |
AR (1) | AR005147A1 (es) |
AT (1) | ATE212551T1 (es) |
AU (1) | AU709474B2 (es) |
BG (1) | BG63933B1 (es) |
BR (1) | BR9612230A (es) |
CA (1) | CA2239352C (es) |
CO (1) | CO4480098A1 (es) |
CZ (1) | CZ293747B6 (es) |
DE (1) | DE69618987T2 (es) |
DK (1) | DK0868183T3 (es) |
DZ (1) | DZ2146A1 (es) |
EG (1) | EG24071A (es) |
ES (1) | ES2167609T3 (es) |
GT (1) | GT199600098A (es) |
HR (1) | HRP960607B1 (es) |
HU (1) | HU227918B1 (es) |
IL (1) | IL124454A (es) |
IS (1) | IS2010B (es) |
MA (1) | MA24035A1 (es) |
MX (1) | MX9805026A (es) |
MY (1) | MY117109A (es) |
NO (1) | NO315734B1 (es) |
NZ (2) | NZ320545A (es) |
OA (1) | OA10697A (es) |
PE (1) | PE25798A1 (es) |
PL (1) | PL186795B1 (es) |
PT (1) | PT868183E (es) |
RS (1) | RS49523B (es) |
RU (1) | RU2141827C1 (es) |
SI (1) | SI0868183T1 (es) |
SK (1) | SK284412B6 (es) |
TN (1) | TNSN96163A1 (es) |
TW (1) | TW449475B (es) |
UA (1) | UA56151C2 (es) |
WO (1) | WO1997023217A1 (es) |
ZA (1) | ZA9610780B (es) |
Families Citing this family (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ID21415A (id) * | 1997-12-05 | 1999-06-10 | Upjohn Co | Senyawa-senyawa antibiotik magnesium quinolon |
US6017948A (en) * | 1998-10-30 | 2000-01-25 | Supergen, Inc. | Water-miscible pharmaceutical compositions |
DE19937115A1 (de) | 1999-08-06 | 2001-02-08 | Bayer Ag | Wäßrige Arzneimittelformulierung von Moxifloxacin oder Salzen davon |
DE19937116A1 (de) * | 1999-08-06 | 2001-02-08 | Bayer Ag | Moxifloxacin Kochsalzformulierung |
WO2001051089A1 (de) * | 2000-01-13 | 2001-07-19 | Merck Patent Gmbh | Pharmazeutische zubereitungen enthaltend 2-pyrrolidon als lösungsvermittler |
US8637077B2 (en) | 2000-12-28 | 2014-01-28 | Takeda Pharmaceutical Company Limited | Sustained-release preparation |
AU2003247793A1 (en) * | 2002-06-26 | 2004-01-19 | Pharmacia Corporation | Stable liquid parenteral parecoxib formulation |
EP1764102A4 (en) * | 2004-07-02 | 2010-08-25 | Daiichi Seiyaku Co | MEDICINAL COMPOSITION CONTAINING QUINOLONE |
US8546423B2 (en) | 2005-05-18 | 2013-10-01 | Mpex Pharmaceuticals, Inc. | Aerosolized fluoroquinolones and uses thereof |
HUE038814T2 (hu) * | 2005-05-18 | 2018-11-28 | Horizon Orphan Llc | Aeroszolizált fluor-kinolonok és alkalmazásaik |
FR2896416B1 (fr) | 2006-01-24 | 2010-08-13 | Vetoquinol | Composition anti-infectieuse comprenant un compose de type pyrido (3,2,1-ij)-benzoxadiazine |
LT1991201T (lt) * | 2006-02-10 | 2018-07-25 | Pari Pharma Gmbh | Puškiami antibiotikai inhaliaciniam gydymui |
US20070197548A1 (en) | 2006-02-17 | 2007-08-23 | Murthy Yerramilli V S | Fluoroquinolone compositions |
DE102006010643A1 (de) * | 2006-03-08 | 2007-09-13 | Bayer Healthcare Aktiengesellschaft | Arzneimittel enthaltend Fluorchinolone |
DE102006010642A1 (de) * | 2006-03-08 | 2007-09-27 | Bayer Healthcare Aktiengesellschaft | Arzneimittelformulierungen, enthaltend Fluorchinolone |
MX2007009796A (es) | 2007-08-14 | 2009-02-25 | Cell Therapy And Technology S | Gel conteniendo pirfenidona. |
JP2012505223A (ja) | 2008-10-07 | 2012-03-01 | エムペックス・ファーマシューティカルズ・インコーポレーテッド | 薬物動態の改善のためのエアゾールフルオロキノロン配合物 |
CN102325532B (zh) | 2008-10-07 | 2015-06-17 | Mpex医药有限公司 | 用于减轻肺部炎症的左氧氟沙星吸入剂 |
LT2473170T (lt) | 2009-09-04 | 2019-10-10 | Horizon Orphan Llc | Aerozolizuoto levofloksacino panaudojimas cistinės fibrozės gydymui |
MX2011007675A (es) | 2011-07-19 | 2012-07-11 | Cell Therapy And Technology S A De C V | Procedimiento para la fabricacion de una composicion farmaceutica en forma de tabletas de liberacion prolongada conteniendo pirfenidona y su aplicacion en la regresion de la insuficiencia renal cronica, contractura capsular mamaria y fibrosis hepatica humanas. |
MX346763B (es) | 2012-03-28 | 2017-03-31 | Cell Therapy And Tech S A De C V | Composición tópica semisólida conteniendo pirfenidona y dialil óxido de disulfuro modificado (odd-m) para eliminar o prevenir el acné. |
MX356551B (es) | 2012-08-23 | 2018-06-04 | Grupo Medifarma S A De C V Star | Composición antiséptica, antiseborreica y exfoliante para eliminar o prevenir el acné. |
JP6675396B2 (ja) | 2015-06-02 | 2020-04-01 | 杏林製薬株式会社 | 水性液剤 |
EP3305296A4 (en) | 2015-06-02 | 2019-02-13 | Kyorin Pharmaceutical Co., Ltd. | AQUEOUS LIQUID FORMULATION |
US10617684B2 (en) | 2015-06-02 | 2020-04-14 | Kyorin Pharmaceutical Co., Ltd. | Aqueous drug |
MX2019009572A (es) * | 2017-02-13 | 2019-10-02 | Bayer Animal Health Gmbh | Composicion liquida que contiene pradofloxacina. |
MX366086B (es) | 2017-08-15 | 2019-06-27 | Cell Therapy And Tech S A De C V | Composicion topica semisolida conteniendo un agente antimicrobiano y pirfenidona para el tratamiento de daños cronicos de la piel. |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3517709A1 (de) * | 1985-01-05 | 1986-07-10 | Bayer Ag | Basische zubereitungen von chinoloncarbonsaeuren |
JPS63188626A (ja) * | 1987-01-30 | 1988-08-04 | Dainippon Pharmaceut Co Ltd | ピリドンカルボン酸の可溶化方法 |
DE3902079A1 (de) * | 1988-04-15 | 1989-10-26 | Bayer Ag | I.m. injektionsformen von gyrase-inhibitoren |
DK0507851T3 (da) * | 1989-12-29 | 1997-08-25 | Abbott Lab | Quinoloncarboxylsyre-matalion-syrekomplekser |
US5084276A (en) * | 1990-01-05 | 1992-01-28 | Abbott Laboratories | Quinolone carboxylic acid compositions with polymeric additive to reduce vein irritation |
ATE108649T1 (de) * | 1990-02-14 | 1994-08-15 | Takeda Chemical Industries Ltd | Brausemischung, deren herstellung sowie verwendung. |
FR2665635A1 (fr) * | 1990-08-10 | 1992-02-14 | Merck Sharp & Dohme | Composition pharmaceutique fluide a base d'un complexe metallique et son procede de preparation. |
US5082863A (en) * | 1990-08-29 | 1992-01-21 | Schering Corporation | Pharmaceutical composition of florfenicol |
US5235054A (en) * | 1992-07-15 | 1993-08-10 | Pfizer Inc. | 3-carboxaldehyde substituted quinolines and naphthyridines |
JPH0782141A (ja) * | 1993-09-17 | 1995-03-28 | Tanabe Seiyaku Co Ltd | 動物用注射剤 |
-
1996
- 1996-11-13 SK SK807-98A patent/SK284412B6/sk not_active IP Right Cessation
- 1996-11-13 HU HU9903726A patent/HU227918B1/hu unknown
- 1996-11-13 SI SI9630422T patent/SI0868183T1/xx unknown
- 1996-11-13 IL IL12445496A patent/IL124454A/xx not_active IP Right Cessation
- 1996-11-13 DE DE69618987T patent/DE69618987T2/de not_active Expired - Lifetime
- 1996-11-13 EP EP96935251A patent/EP0868183B1/en not_active Expired - Lifetime
- 1996-11-13 BR BR9612230A patent/BR9612230A/pt active IP Right Grant
- 1996-11-13 NZ NZ320545A patent/NZ320545A/xx not_active IP Right Cessation
- 1996-11-13 CZ CZ19981930A patent/CZ293747B6/cs not_active IP Right Cessation
- 1996-11-13 ES ES96935251T patent/ES2167609T3/es not_active Expired - Lifetime
- 1996-11-13 CA CA002239352A patent/CA2239352C/en not_active Expired - Lifetime
- 1996-11-13 UA UA98063226A patent/UA56151C2/uk unknown
- 1996-11-13 JP JP52344797A patent/JP3416145B2/ja not_active Expired - Lifetime
- 1996-11-13 PT PT96935251T patent/PT868183E/pt unknown
- 1996-11-13 AU AU73289/96A patent/AU709474B2/en not_active Expired
- 1996-11-13 NZ NZ501160A patent/NZ501160A/en not_active IP Right Cessation
- 1996-11-13 CN CN96199249A patent/CN1104899C/zh not_active Expired - Lifetime
- 1996-11-13 AT AT96935251T patent/ATE212551T1/de active
- 1996-11-13 DK DK96935251T patent/DK0868183T3/da active
- 1996-11-13 WO PCT/IB1996/001217 patent/WO1997023217A1/en active IP Right Grant
- 1996-11-13 KR KR10-1998-0704719A patent/KR100402570B1/ko not_active IP Right Cessation
- 1996-11-13 PL PL96328001A patent/PL186795B1/pl unknown
- 1996-11-13 RU RU98111831A patent/RU2141827C1/ru active
- 1996-11-15 TW TW085114021A patent/TW449475B/zh not_active IP Right Cessation
- 1996-12-10 PE PE1996000892A patent/PE25798A1/es not_active Application Discontinuation
- 1996-12-17 EG EG113496A patent/EG24071A/xx active
- 1996-12-18 MA MA24427A patent/MA24035A1/fr unknown
- 1996-12-18 DZ DZ960191A patent/DZ2146A1/fr active
- 1996-12-18 TN TNTNSN96163A patent/TNSN96163A1/fr unknown
- 1996-12-19 US US08/769,809 patent/US5811130A/en not_active Expired - Lifetime
- 1996-12-19 AR ARP960105774A patent/AR005147A1/es active IP Right Grant
- 1996-12-19 AP APAP/P/1996/000898A patent/AP706A/en active
- 1996-12-19 HR HR960607A patent/HRP960607B1/xx not_active IP Right Cessation
- 1996-12-19 GT GT199600098A patent/GT199600098A/es unknown
- 1996-12-20 RS YU69096A patent/RS49523B/sr unknown
- 1996-12-20 CO CO96066993A patent/CO4480098A1/es unknown
- 1996-12-20 MY MYPI96005411A patent/MY117109A/en unknown
- 1996-12-20 ZA ZA9610780A patent/ZA9610780B/xx unknown
-
1998
- 1998-05-25 IS IS4755A patent/IS2010B/is unknown
- 1998-06-12 OA OA9800082A patent/OA10697A/en unknown
- 1998-06-15 BG BG102542A patent/BG63933B1/bg unknown
- 1998-06-19 NO NO19982842A patent/NO315734B1/no not_active IP Right Cessation
- 1998-06-19 MX MX9805026A patent/MX9805026A/es unknown
Also Published As
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