EA200601515A1 - Пиразолопиримидины для борьбы с нежелательными микроорганизмами - Google Patents

Пиразолопиримидины для борьбы с нежелательными микроорганизмами

Info

Publication number
EA200601515A1
EA200601515A1 EA200601515A EA200601515A EA200601515A1 EA 200601515 A1 EA200601515 A1 EA 200601515A1 EA 200601515 A EA200601515 A EA 200601515A EA 200601515 A EA200601515 A EA 200601515A EA 200601515 A1 EA200601515 A1 EA 200601515A1
Authority
EA
Eurasian Patent Office
Prior art keywords
pyrazolopyrimidines
microoranisms
against undesirable
struggle against
struggle
Prior art date
Application number
EA200601515A
Other languages
English (en)
Inventor
Олаф Гебауер
Херберт Гайер
Ульрих Хайнеманн
Штефан Херрманн
Штефан Хиллебранд
Ханс-Людвиг Эльбе
Рональд Эбберт
Ульрике Вахендорфф-Нойманн
Петер Дамен
Карл-Хайнц Кук
Маморау Хатазава
Original Assignee
Байер Кропсайенс Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Байер Кропсайенс Аг filed Critical Байер Кропсайенс Аг
Publication of EA200601515A1 publication Critical patent/EA200601515A1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Изобретение относится к пиразолопиримидинам формулыгдеR, R, R, R, Rи Х имеют значения, приведенные в описании.Приведен способ получения этих соединений и описано их применение для борьбы с нежелательными микроорганизмами.
EA200601515A 2004-02-20 2005-02-18 Пиразолопиримидины для борьбы с нежелательными микроорганизмами EA200601515A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004008807A DE102004008807A1 (de) 2004-02-20 2004-02-20 Pyrazolopyrimidine
PCT/EP2005/001694 WO2005082907A2 (de) 2004-02-20 2005-02-18 Pyrazolopyrimidine zur bekämpfung unerwünschter mikroorganismen

Publications (1)

Publication Number Publication Date
EA200601515A1 true EA200601515A1 (ru) 2006-12-29

Family

ID=34832976

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200601515A EA200601515A1 (ru) 2004-02-20 2005-02-18 Пиразолопиримидины для борьбы с нежелательными микроорганизмами

Country Status (15)

Country Link
US (1) US7629294B2 (ru)
EP (1) EP1718652A2 (ru)
JP (1) JP2007524691A (ru)
KR (1) KR20070015386A (ru)
CN (1) CN1946293A (ru)
AR (1) AR048857A1 (ru)
BR (1) BRPI0507894A (ru)
CA (1) CA2556798A1 (ru)
CR (1) CR8559A (ru)
DE (1) DE102004008807A1 (ru)
EA (1) EA200601515A1 (ru)
IL (1) IL177510A0 (ru)
MX (1) MXPA06009311A (ru)
TW (1) TW200538044A (ru)
WO (1) WO2005082907A2 (ru)

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RU2805476C2 (ru) * 2017-07-28 2023-10-17 Нимбус Лакшми, Инк. Ингибиторы tyk2 и их применения

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DE102005007534A1 (de) * 2005-02-17 2006-08-31 Bayer Cropscience Ag Pyrazolopyrimidine
US8188097B2 (en) 2005-10-21 2012-05-29 Mitsubishi Tanabe Pharma Corporation Pyrazolo[1,5-A]pyrimidine compounds
JP4847275B2 (ja) * 2005-10-21 2011-12-28 田辺三菱製薬株式会社 ピラゾロ［１，５−ａ］ピリミジン化合物
AR061793A1 (es) 2006-07-05 2008-09-24 Mitsubishi Tanabe Pharma Corp Compuesto de pirazolo[1,5-a] pirimidina y composicion farmaceutica
TWI419889B (zh) * 2006-07-05 2013-12-21 Mitsubishi Tanabe Pharma Corp 吡唑并〔１，５-ａ〕嘧啶化合物
DE102006039255A1 (de) * 2006-08-17 2008-02-21 Bayer Cropscience Ag Insektizide heterocyclische Carbonsäurederivate
WO2008046856A2 (de) * 2006-10-18 2008-04-24 Basf Se Fungizide zusammensetzungen
JP4837701B2 (ja) * 2007-04-20 2011-12-14 田辺三菱製薬株式会社 医薬組成物
EP2014661A1 (de) * 2007-06-13 2009-01-14 Bayer CropScience AG Heterocyclisch substituierte Heterocyclyl-carbonsäurederivate
US8507673B2 (en) * 2008-12-11 2013-08-13 Emory University Process for preparing 5,7 diaminopyrazolo [1,5-A] pyrimidine compounds
US9133189B2 (en) 2013-03-14 2015-09-15 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
EP2970137A1 (en) 2013-03-14 2016-01-20 Epizyme, Inc. Pyrazole derivatives as arginine methyltransferase inhibitors and uses thereof
US9120757B2 (en) 2013-03-14 2015-09-01 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
US9023883B2 (en) 2013-03-14 2015-05-05 Epizyme, Inc. PRMT1 inhibitors and uses thereof
WO2014153208A1 (en) 2013-03-14 2014-09-25 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
BR112015022785A2 (pt) 2013-03-14 2017-07-18 Epizyme Inc composto; composição farmacêutica; kit ou artigo farmacêutico embalado; método de inibição de uma arginina metil transferase (rmt); método de modulação da expressão genética; método de modulação da transcrição; e método de tratamento de um distúrbio mediado por rmt
EP2970134B1 (en) 2013-03-14 2018-02-28 Epizyme, Inc. Pyrazole derivatives as prmt1 inhibitors and uses thereof
US9447079B2 (en) 2013-03-14 2016-09-20 Epizyme, Inc. PRMT1 inhibitors and uses thereof
EP3363434A1 (en) 2013-03-14 2018-08-22 Epizyme Inc Arginine methyltransferase inhibitors and uses thereof
US9394258B2 (en) 2013-03-14 2016-07-19 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
CN117946114A (zh) 2017-07-28 2024-04-30 武田药品工业株式会社 Tyk2抑制剂与其用途
EP3866789A4 (en) * 2018-10-15 2022-07-06 Nimbus Lakshmi, Inc. TYK2 INHIBITORS AND USES THEREOF

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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2805476C2 (ru) * 2017-07-28 2023-10-17 Нимбус Лакшми, Инк. Ингибиторы tyk2 и их применения

Also Published As

Publication number Publication date
AR048857A1 (es) 2006-06-07
MXPA06009311A (es) 2007-03-01
KR20070015386A (ko) 2007-02-02
WO2005082907A2 (de) 2005-09-09
TW200538044A (en) 2005-12-01
CN1946293A (zh) 2007-04-11
EP1718652A2 (de) 2006-11-08
DE102004008807A1 (de) 2005-09-08
US7629294B2 (en) 2009-12-08
US20050187224A1 (en) 2005-08-25
BRPI0507894A (pt) 2007-07-24
CR8559A (es) 2006-11-23
JP2007524691A (ja) 2007-08-30
WO2005082907A3 (de) 2006-06-29
CA2556798A1 (en) 2005-09-09
IL177510A0 (en) 2006-12-10

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