EA200500703A1 - Новые трициклические соединения для лечения воспалительных и аллергических нарушений, способ их приготовления и содержащие их фармацевтические составы - Google Patents
Новые трициклические соединения для лечения воспалительных и аллергических нарушений, способ их приготовления и содержащие их фармацевтические составыInfo
- Publication number
- EA200500703A1 EA200500703A1 EA200500703A EA200500703A EA200500703A1 EA 200500703 A1 EA200500703 A1 EA 200500703A1 EA 200500703 A EA200500703 A EA 200500703A EA 200500703 A EA200500703 A EA 200500703A EA 200500703 A1 EA200500703 A1 EA 200500703A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- treatment
- inflammatory
- tricyclic compounds
- preparation
- allergic disorders
- Prior art date
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/91—Dibenzofurans; Hydrogenated dibenzofurans
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/80—[b, c]- or [b, d]-condensed
- C07D209/82—Carbazoles; Hydrogenated carbazoles
- C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/76—Dibenzothiophenes
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Abstract
Настоящее изобретение относится к новым трициклическим соединениям, применимым для лечения воспалительных состояний, заболеваний центральной нервной системы и инсулин-резистентного диабета.Международная заявка была опубликована вместе с отчетом о международном поиске.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN922MU2002 | 2002-10-23 | ||
PCT/IB2003/004442 WO2004037805A1 (en) | 2002-10-23 | 2003-10-08 | Novel tricyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200500703A1 true EA200500703A1 (ru) | 2005-12-29 |
EA010408B1 EA010408B1 (ru) | 2008-08-29 |
Family
ID=32170663
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200500703A EA010408B1 (ru) | 2002-10-23 | 2003-10-08 | Трициклические соединения для лечения воспалительных и аллергических нарушений, способы их приготовления и содержащие их фармацевтические составы |
Country Status (20)
Country | Link |
---|---|
US (2) | US7238725B2 (ru) |
EP (1) | EP1554262B1 (ru) |
JP (1) | JP2006506379A (ru) |
KR (1) | KR20050065624A (ru) |
CN (1) | CN100532374C (ru) |
AP (1) | AP2021A (ru) |
AR (1) | AR041661A1 (ru) |
AT (1) | ATE380185T1 (ru) |
AU (1) | AU2003269317B2 (ru) |
BR (1) | BR0314721A (ru) |
CA (1) | CA2503015A1 (ru) |
CO (1) | CO5690638A2 (ru) |
DE (1) | DE60317918T2 (ru) |
EA (1) | EA010408B1 (ru) |
ES (1) | ES2298552T3 (ru) |
MX (1) | MXPA05004432A (ru) |
MY (1) | MY140187A (ru) |
PL (1) | PL376769A1 (ru) |
WO (1) | WO2004037805A1 (ru) |
ZA (1) | ZA200502969B (ru) |
Families Citing this family (77)
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CA2503015A1 (en) * | 2002-10-23 | 2004-05-06 | Glenmark Pharmaceuticals Ltd. | Novel tricyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them |
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GB0401334D0 (en) | 2004-01-21 | 2004-02-25 | Novartis Ag | Organic compounds |
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GT200500281A (es) | 2004-10-22 | 2006-04-24 | Novartis Ag | Compuestos organicos. |
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WO2006051390A1 (en) * | 2004-11-10 | 2006-05-18 | Glenmark Pharmaceuticals S.A. | Heterocyclic compounds useful for the treatment of inflammatory and allergic disorders, pharmaceutical compositions containing them, and methods of preparing them |
GB0426164D0 (en) | 2004-11-29 | 2004-12-29 | Novartis Ag | Organic compounds |
NZ555809A (en) | 2004-12-17 | 2010-07-30 | Glenmark Pharmaceuticals Sa | Novel heterocyclic compounds useful for the treatment of inflammatory and allergic disorders |
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GB0507577D0 (en) | 2005-04-14 | 2005-05-18 | Novartis Ag | Organic compounds |
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- 2003-10-08 BR BR0314721-5A patent/BR0314721A/pt not_active IP Right Cessation
- 2003-10-08 AU AU2003269317A patent/AU2003269317B2/en not_active Ceased
- 2003-10-08 AP AP2005003302A patent/AP2021A/xx active
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- 2003-10-08 JP JP2004546246A patent/JP2006506379A/ja active Pending
- 2003-10-08 KR KR1020057006974A patent/KR20050065624A/ko not_active Application Discontinuation
- 2003-10-08 US US10/532,273 patent/US7238725B2/en not_active Expired - Fee Related
- 2003-10-08 EA EA200500703A patent/EA010408B1/ru not_active IP Right Cessation
- 2003-10-08 WO PCT/IB2003/004442 patent/WO2004037805A1/en active IP Right Grant
- 2003-10-08 PL PL376769A patent/PL376769A1/pl not_active Application Discontinuation
- 2003-10-08 CN CNB2003801072469A patent/CN100532374C/zh not_active Expired - Fee Related
- 2003-10-08 ES ES03751096T patent/ES2298552T3/es not_active Expired - Lifetime
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- 2003-10-08 MX MXPA05004432A patent/MXPA05004432A/es active IP Right Grant
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- 2005-04-13 ZA ZA200502969A patent/ZA200502969B/en unknown
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AP2005003302A0 (en) | 2005-06-30 |
ES2298552T3 (es) | 2008-05-16 |
CO5690638A2 (es) | 2006-10-31 |
US20060178418A1 (en) | 2006-08-10 |
AP2021A (en) | 2009-08-03 |
CN1729181A (zh) | 2006-02-01 |
MXPA05004432A (es) | 2005-11-23 |
EP1554262A1 (en) | 2005-07-20 |
PL376769A1 (pl) | 2006-01-09 |
AU2003269317B2 (en) | 2009-10-29 |
US20080146810A1 (en) | 2008-06-19 |
US7238725B2 (en) | 2007-07-03 |
BR0314721A (pt) | 2005-08-02 |
KR20050065624A (ko) | 2005-06-29 |
CN100532374C (zh) | 2009-08-26 |
JP2006506379A (ja) | 2006-02-23 |
CA2503015A1 (en) | 2004-05-06 |
ATE380185T1 (de) | 2007-12-15 |
DE60317918D1 (de) | 2008-01-17 |
EA010408B1 (ru) | 2008-08-29 |
AR041661A1 (es) | 2005-05-26 |
ZA200502969B (en) | 2006-02-22 |
AU2003269317A1 (en) | 2004-05-13 |
EP1554262B1 (en) | 2007-12-05 |
MY140187A (en) | 2009-11-30 |
DE60317918T2 (de) | 2009-01-29 |
WO2004037805A1 (en) | 2004-05-06 |
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