EA200201247A1 - Соединения для лечения болезни альцгеймера - Google Patents

Соединения для лечения болезни альцгеймера

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Publication number
EA200201247A1
EA200201247A1 EA200201247A EA200201247A EA200201247A1 EA 200201247 A1 EA200201247 A1 EA 200201247A1 EA 200201247 A EA200201247 A EA 200201247A EA 200201247 A EA200201247 A EA 200201247A EA 200201247 A1 EA200201247 A1 EA 200201247A1
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EA
Eurasian Patent Office
Prior art keywords
disease
alzheimer
connections
treatment
formula
Prior art date
Application number
EA200201247A
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English (en)
Other versions
EA007337B1 (ru
Inventor
Мишель Мэйлард
Рой Хом
Андреа Гэйлунас
Барбара Ягоджинска
Лоренс И. Фанг
Варгезе Джон
Джон Н. Фрескос
Шон Р. Пулли
Джеймс П. Бек
Рут Е. Тенбринк
Original Assignee
Элан Фармасьютикалз, Инк.
Фармация Энд Апджон Компани
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Application filed by Элан Фармасьютикалз, Инк., Фармация Энд Апджон Компани filed Critical Элан Фармасьютикалз, Инк.
Publication of EA200201247A1 publication Critical patent/EA200201247A1/ru
Publication of EA007337B1 publication Critical patent/EA007337B1/ru

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    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/26—Sulfur atoms
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    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
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    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
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Abstract

Данное изобретение касается замещенных аминов формулы (X)использующихся для лечения болезни Альцгеймера и других похожих заболеваний.
EA200201247A 2000-06-30 2001-06-29 Соединения для лечения болезни альцгеймера EA007337B1 (ru)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US21532300P 2000-06-30 2000-06-30
US25273600P 2000-11-22 2000-11-22
US25595600P 2000-12-15 2000-12-15
US26849701P 2001-02-13 2001-02-13
US27977901P 2001-03-29 2001-03-29
US29558901P 2001-06-04 2001-06-04
PCT/US2001/021012 WO2002002512A2 (en) 2000-06-30 2001-06-29 Compounds to treat alzheimer's disease

Publications (2)

Publication Number Publication Date
EA200201247A1 true EA200201247A1 (ru) 2003-10-30
EA007337B1 EA007337B1 (ru) 2006-08-25

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EA200201247A EA007337B1 (ru) 2000-06-30 2001-06-29 Соединения для лечения болезни альцгеймера

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US (1) US7214715B2 (ru)
EP (1) EP1353898A2 (ru)
JP (1) JP2004502669A (ru)
KR (1) KR20030058960A (ru)
CN (1) CN100366605C (ru)
AR (1) AR031852A1 (ru)
AU (1) AU2001273137A1 (ru)
BR (1) BR0112000A (ru)
CA (1) CA2410651A1 (ru)
CZ (1) CZ20024194A3 (ru)
EA (1) EA007337B1 (ru)
EE (1) EE200200716A (ru)
HU (1) HUP0303037A3 (ru)
IL (1) IL153214A0 (ru)
MX (1) MXPA02012608A (ru)
NO (1) NO20026199L (ru)
NZ (3) NZ547529A (ru)
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HUP0303037A2 (hu) 2004-03-01
CA2410651A1 (en) 2002-01-10
AU2001273137A1 (en) 2002-01-14
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