DOP2018000083A - NUEVOS DERIVADOS DE IMIDAZO[4,5-b]PIRIDINA, UN PROCESO PARA SU PREPARACIÓN Y COMPOSICIONES FARMACÉUTICAS QUE LOS CONTIENEN - Google Patents
NUEVOS DERIVADOS DE IMIDAZO[4,5-b]PIRIDINA, UN PROCESO PARA SU PREPARACIÓN Y COMPOSICIONES FARMACÉUTICAS QUE LOS CONTIENENInfo
- Publication number
- DOP2018000083A DOP2018000083A DO2018000083A DO2018000083A DOP2018000083A DO P2018000083 A DOP2018000083 A DO P2018000083A DO 2018000083 A DO2018000083 A DO 2018000083A DO 2018000083 A DO2018000083 A DO 2018000083A DO P2018000083 A DOP2018000083 A DO P2018000083A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- piridina
- imidazo
- preparation
- pharmaceutical compositions
- compositions containing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Abstract
Compuestos de fórmula (I): en la que R1, R2, R3, R4, y R5 son como se definen en la descripción. Medicamentos.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR1559252A FR3041639B1 (fr) | 2015-09-30 | 2015-09-30 | NOUVEAUX DERIVES D'IMIDAZO[4,5-b]PYRIDINE, PROCEDE POUR LES PREPARER ET COMPOSITIONS PHARMACEUTIQUES LES CONTENANT |
Publications (1)
Publication Number | Publication Date |
---|---|
DOP2018000083A true DOP2018000083A (es) | 2018-10-15 |
Family
ID=54979755
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DO2018000083A DOP2018000083A (es) | 2015-09-30 | 2018-03-27 | NUEVOS DERIVADOS DE IMIDAZO[4,5-b]PIRIDINA, UN PROCESO PARA SU PREPARACIÓN Y COMPOSICIONES FARMACÉUTICAS QUE LOS CONTIENEN |
Country Status (26)
Country | Link |
---|---|
US (1) | US20180273528A1 (es) |
EP (1) | EP3356363A1 (es) |
JP (1) | JP2018535931A (es) |
KR (1) | KR20180054858A (es) |
CN (1) | CN108137581A (es) |
AU (1) | AU2016333505A1 (es) |
BR (1) | BR112018006157A2 (es) |
CA (1) | CA2999935A1 (es) |
CL (1) | CL2018000783A1 (es) |
CO (1) | CO2018003473A2 (es) |
CR (1) | CR20180181A (es) |
CU (1) | CU20180028A7 (es) |
DO (1) | DOP2018000083A (es) |
EA (1) | EA201890821A1 (es) |
EC (1) | ECSP18023253A (es) |
FR (1) | FR3041639B1 (es) |
HK (1) | HK1255804A1 (es) |
IL (1) | IL258341A (es) |
MA (1) | MA43020A (es) |
MX (1) | MX2018003860A (es) |
NI (1) | NI201800043A (es) |
PE (1) | PE20181331A1 (es) |
PH (1) | PH12018500650A1 (es) |
SV (1) | SV2018005657A (es) |
TN (1) | TN2018000090A1 (es) |
WO (1) | WO2017055530A1 (es) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN108822103A (zh) * | 2018-07-28 | 2018-11-16 | 刘凤娟 | 一种咪唑并[4,5-b]吡啶化合物及其制备方法和应用 |
CA3118093A1 (en) * | 2018-09-28 | 2020-04-02 | Arizona Board Of Regents On Behalf Of The University Of Arizona | Small molecule inhibitors of dyrk1/clk and uses thereof |
CA3116347A1 (en) | 2018-10-31 | 2020-05-07 | Gilead Sciences, Inc. | Substituted 6-azabenzimidazole compounds having hpk1 inhibitory activity |
JP7460644B2 (ja) | 2018-10-31 | 2024-04-02 | ギリアード サイエンシーズ, インコーポレイテッド | Hpk1阻害剤としての置換6-アザベンゾイミダゾール化合物 |
US11453681B2 (en) | 2019-05-23 | 2022-09-27 | Gilead Sciences, Inc. | Substituted eneoxindoles and uses thereof |
KR20220079851A (ko) * | 2019-09-11 | 2022-06-14 | 프렐루드 테라퓨틱스, 인코포레이티드 | Cdk 억제제 및 약제로서의 이의 용도 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2016516710A (ja) * | 2013-03-13 | 2016-06-09 | アッヴィ・インコーポレイテッド | ピリジン系cdk9キナーゼ阻害薬 |
-
2015
- 2015-09-30 FR FR1559252A patent/FR3041639B1/fr not_active Expired - Fee Related
-
2016
- 2016-09-30 KR KR1020187012175A patent/KR20180054858A/ko unknown
- 2016-09-30 JP JP2018516194A patent/JP2018535931A/ja active Pending
- 2016-09-30 BR BR112018006157A patent/BR112018006157A2/pt not_active Application Discontinuation
- 2016-09-30 CR CR20180181A patent/CR20180181A/es unknown
- 2016-09-30 WO PCT/EP2016/073395 patent/WO2017055530A1/en active Application Filing
- 2016-09-30 AU AU2016333505A patent/AU2016333505A1/en not_active Abandoned
- 2016-09-30 EP EP16774682.5A patent/EP3356363A1/en not_active Withdrawn
- 2016-09-30 MA MA043020A patent/MA43020A/fr unknown
- 2016-09-30 CU CUP2018000028A patent/CU20180028A7/es unknown
- 2016-09-30 TN TNP/2018/000090A patent/TN2018000090A1/en unknown
- 2016-09-30 CN CN201680058054.0A patent/CN108137581A/zh not_active Withdrawn
- 2016-09-30 MX MX2018003860A patent/MX2018003860A/es unknown
- 2016-09-30 CA CA2999935A patent/CA2999935A1/en not_active Abandoned
- 2016-09-30 PE PE2018000443A patent/PE20181331A1/es unknown
- 2016-09-30 US US15/763,248 patent/US20180273528A1/en not_active Abandoned
- 2016-09-30 EA EA201890821A patent/EA201890821A1/ru unknown
-
2018
- 2018-03-22 SV SV2018005657A patent/SV2018005657A/es unknown
- 2018-03-23 NI NI201800043A patent/NI201800043A/es unknown
- 2018-03-23 PH PH12018500650A patent/PH12018500650A1/en unknown
- 2018-03-25 IL IL258341A patent/IL258341A/en unknown
- 2018-03-26 EC ECIEPI201823253A patent/ECSP18023253A/es unknown
- 2018-03-26 CL CL2018000783A patent/CL2018000783A1/es unknown
- 2018-03-27 DO DO2018000083A patent/DOP2018000083A/es unknown
- 2018-03-28 CO CONC2018/0003473A patent/CO2018003473A2/es unknown
- 2018-11-15 HK HK18114643.2A patent/HK1255804A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
KR20180054858A (ko) | 2018-05-24 |
EA201890821A1 (ru) | 2018-10-31 |
US20180273528A1 (en) | 2018-09-27 |
TN2018000090A1 (en) | 2019-07-08 |
BR112018006157A2 (pt) | 2018-10-09 |
CA2999935A1 (en) | 2017-04-06 |
AU2016333505A1 (en) | 2018-04-19 |
SV2018005657A (es) | 2018-07-31 |
ECSP18023253A (es) | 2018-04-30 |
MX2018003860A (es) | 2018-08-16 |
PE20181331A1 (es) | 2018-08-20 |
JP2018535931A (ja) | 2018-12-06 |
WO2017055530A1 (en) | 2017-04-06 |
FR3041639B1 (fr) | 2019-01-25 |
MA43020A (fr) | 2018-08-08 |
CL2018000783A1 (es) | 2018-09-21 |
FR3041639A1 (es) | 2017-03-31 |
EP3356363A1 (en) | 2018-08-08 |
HK1255804A1 (zh) | 2019-08-23 |
NI201800043A (es) | 2018-06-21 |
PH12018500650A1 (en) | 2018-10-01 |
CO2018003473A2 (es) | 2018-07-10 |
IL258341A (en) | 2018-05-31 |
CR20180181A (es) | 2018-06-22 |
CU20180028A7 (es) | 2018-07-05 |
CN108137581A (zh) | 2018-06-08 |
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