DK92880A - 6-beta-substituerede penicillansyrer fremgangsmaade til deres fremstilling samt deres anvendelse - Google Patents

6-beta-substituerede penicillansyrer fremgangsmaade til deres fremstilling samt deres anvendelse

Info

Publication number: DK92880A
Authority: DK; Denmark
Prior art keywords: beta; preparation; penicillanic acid; acid procedure; substituted penicillanic
Prior art date: 1979-03-05

Application number

DK92880A

Other languages

English (en)

Other versions

DK157136C (da

DK157136B (da

Inventor

M S Kellogg

E S Hamanaka

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-03-05

Filing date

1980-03-04

Publication date

1980-09-06

1980-03-04 Application filed by Pfizer filed Critical Pfizer

1980-09-06 Publication of DK92880A publication Critical patent/DK92880A/da

1989-11-13 Publication of DK157136B publication Critical patent/DK157136B/da

1990-04-16 Application granted granted Critical

1990-04-16 Publication of DK157136C publication Critical patent/DK157136C/da

Links

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
- A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
- A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)

DK092880A 1979-03-05 1980-03-04 Fremgangsmaade til fremstilling af 6-beta-iodpenicillansyre og estre heraf DK157136C (da)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US1780979A	1979-03-05	1979-03-05
US1780979		1979-03-05
US06/096,832 US4397783A (en)	1979-03-05	1979-11-23	Process for converting 6,6-disubstituted penicillanic acid derivatives to the 6-β-congeners
US9683279		1979-11-23

Publications (3)

Publication Number	Publication Date
DK92880A true DK92880A (da)	1980-09-06
DK157136B DK157136B (da)	1989-11-13
DK157136C DK157136C (da)	1990-04-16

Family

ID=26690341

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK092880A DK157136C (da)	1979-03-05	1980-03-04	Fremgangsmaade til fremstilling af 6-beta-iodpenicillansyre og estre heraf

Country Status (29)

Country	Link
US (1)	US4397783A (da)
KR (1)	KR840000589B1 (da)
AR (1)	AR225758A1 (da)
AT (1)	AT369744B (da)
AU (1)	AU518472B2 (da)
CA (1)	CA1154011A (da)
CH (1)	CH648850A5 (da)
DD (1)	DD149366A5 (da)
DE (1)	DE3008316C2 (da)
DK (1)	DK157136C (da)
ES (1)	ES489186A0 (da)
FI (1)	FI71739C (da)
FR (1)	FR2450837A1 (da)
GB (1)	GB2047684B (da)
GR (1)	GR67697B (da)
HK (1)	HK66687A (da)
IE (1)	IE51931B1 (da)
IL (1)	IL59514A (da)
IT (1)	IT1130301B (da)
KE (1)	KE3456A (da)
LU (1)	LU82219A1 (da)
MY (1)	MY8500320A (da)
NL (1)	NL8001286A (da)
NO (1)	NO800617L (da)
OA (1)	OA06496A (da)
PH (2)	PH18550A (da)
PT (1)	PT70898A (da)
SE (1)	SE451329B (da)
SG (1)	SG56484G (da)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4518530A (en) *	1979-03-05	1985-05-21	Pfizer Inc.	6-β-Substituted penicillanic acids as β-lactamase inhibitors
IL59948A0 (en) *	1979-05-21	1980-06-30	Rech Applications Therap	Penicillanic acid derivatives,their production and pharmaceutical compositions containing them
US4511512A (en) *	1980-05-01	1985-04-16	Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Produktionsaktiensel skab)	Substantially pure dicyclohexyl ammonium 6-β-bromo-penicillanate
IE51846B1 (en) *	1980-11-17	1987-04-15	Leo Pharm Prod Ltd	Pharmaceutical preparation for veterinary use and an appliance containing it
EP0139047A1 (en) *	1983-10-18	1985-05-02	Gist-Brocades N.V.	Process for the preparation of 6,6-dibromopenicillanic acid 1,1-dioxide
GB8522156D0 (en) *	1985-09-06	1985-10-09	Leo Pharm Prod Ltd	Producing chemical compounds
US4816580A (en) *	1986-04-10	1989-03-28	Leo Pharmaceutical Products Ltd. A/S	Improved method for preparing penicillanic acid derivatives
PA8579701A1 (es) *	2002-08-23	2005-05-24	Pfizer Prod Inc	Profarmaco inhibidor de beta-lactamasa
BRPI0410936A (pt) *	2003-06-05	2006-06-27	Pfizer Prod Inc	pró-fármaco inibidor da beta-lactamase

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS5749555B2 (da) *	1973-04-04	1982-10-22
US4093625A (en) *	1976-08-09	1978-06-06	Massachusetts Institute Of Technology	6-Sulfur analogs of penicillins and cephalosporins
US4180506A (en) *	1978-01-18	1979-12-25	Rex Pratt	6β-Bromo penicillanic acid
CA1158639A (en) *	1978-12-11	1983-12-13	Eric M. Gordon	6-bromopenicillanic acid sulfone
US4203992A (en) *	1978-12-11	1980-05-20	E. R. Squibb & Sons, Inc.	β-Bromopenicillanic acid sulfone
DE3068390D1 (en) *	1979-01-10	1984-08-09	Beecham Group Plc	Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
IL59081A0 (en) *	1979-01-10	1980-05-30	Schering Corp	2-penem compounds and a method for preparing them

1979
- 1979-11-23 US US06/096,832 patent/US4397783A/en not_active Expired - Lifetime
1980
- 1980-03-03 LU LU82219A patent/LU82219A1/fr unknown
- 1980-03-03 PH PH23716A patent/PH18550A/en unknown
- 1980-03-03 IL IL59514A patent/IL59514A/xx not_active IP Right Cessation
- 1980-03-03 GB GB8007142A patent/GB2047684B/en not_active Expired
- 1980-03-03 GR GR61335A patent/GR67697B/el unknown
- 1980-03-04 FR FR8004765A patent/FR2450837A1/fr active Granted
- 1980-03-04 IE IE428/80A patent/IE51931B1/en not_active IP Right Cessation
- 1980-03-04 CH CH1715/80A patent/CH648850A5/de not_active IP Right Cessation
- 1980-03-04 ES ES489186A patent/ES489186A0/es active Granted
- 1980-03-04 SE SE8001689A patent/SE451329B/sv not_active IP Right Cessation
- 1980-03-04 AR AR225758A patent/AR225758A1/es active
- 1980-03-04 PT PT70898A patent/PT70898A/pt unknown
- 1980-03-04 CA CA000346906A patent/CA1154011A/en not_active Expired
- 1980-03-04 NO NO800617A patent/NO800617L/no unknown
- 1980-03-04 DE DE3008316A patent/DE3008316C2/de not_active Expired
- 1980-03-04 AT AT0118980A patent/AT369744B/de not_active IP Right Cessation
- 1980-03-04 FI FI800662A patent/FI71739C/fi not_active IP Right Cessation
- 1980-03-04 DD DD80219434A patent/DD149366A5/de unknown
- 1980-03-04 AU AU56105/80A patent/AU518472B2/en not_active Ceased
- 1980-03-04 KR KR1019800000921A patent/KR840000589B1/ko active
- 1980-03-04 DK DK092880A patent/DK157136C/da not_active IP Right Cessation
- 1980-03-04 NL NL8001286A patent/NL8001286A/nl not_active Application Discontinuation
- 1980-03-05 IT IT20368/80A patent/IT1130301B/it active
- 1980-03-27 OA OA57065A patent/OA06496A/xx unknown
- 1980-09-12 PH PH24569A patent/PH17879A/en unknown
1984
- 1984-08-13 SG SG564/84A patent/SG56484G/en unknown
- 1984-09-24 KE KE3456A patent/KE3456A/xx unknown
1985
- 1985-12-30 MY MY320/85A patent/MY8500320A/xx unknown
1987
- 1987-09-17 HK HK666/87A patent/HK66687A/xx unknown

Also Published As

Publication number	Publication date
SG56484G (en)	1985-03-08
IL59514A (en)	1984-01-31
IT1130301B (it)	1986-06-11
PH17879A (en)	1985-01-14
IT8020368A0 (it)	1980-03-05
HK66687A (en)	1987-09-25
KR840000589B1 (ko)	1984-04-24
ES8103095A1 (es)	1981-02-16
AR225758A1 (es)	1982-04-30
FI800662A (fi)	1980-09-06
CH648850A5 (de)	1985-04-15
DD149366A5 (de)	1981-07-08
DE3008316A1 (de)	1980-09-25
FI71739C (fi)	1987-02-09
GR67697B (da)	1981-09-07
IE800428L (en)	1980-09-05
ES489186A0 (es)	1981-02-16
FI71739B (fi)	1986-10-31
ATA118980A (de)	1982-06-15
LU82219A1 (fr)	1980-09-24
AU5610580A (en)	1980-09-18
OA06496A (fr)	1981-07-31
IL59514A0 (en)	1980-06-30
KR830001941A (ko)	1983-05-19
CA1154011A (en)	1983-09-20
GB2047684A (en)	1980-12-03
MY8500320A (en)	1985-12-31
PH18550A (en)	1985-08-09
SE8001689L (sv)	1980-09-06
DK157136C (da)	1990-04-16
SE451329B (sv)	1987-09-28
DK157136B (da)	1989-11-13
US4397783A (en)	1983-08-09
GB2047684B (en)	1983-09-28
IE51931B1 (en)	1987-04-29
NO800617L (no)	1980-09-08
AU518472B2 (en)	1981-10-01
PT70898A (en)	1980-04-01
AT369744B (de)	1983-01-25
KE3456A (en)	1984-10-12
DE3008316C2 (de)	1982-12-16
NL8001286A (nl)	1980-09-09
FR2450837B1 (da)	1984-01-13
FR2450837A1 (fr)	1980-10-03

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Legal Events

Date	Code	Title	Description
1996-11-18	PBP	Patent lapsed