DK2010538T3 - Fremgangsmåde til fremstilling af [(1R), 2S]-2-aminopropionsyre 2-[4-(4-fluor-2-methyl-1H-indol-5-yloxy)-5-methylpyrrol]2,1-f-[1,2,4-triazin-6-yloxy]-1-methylethylester - Google Patents

Fremgangsmåde til fremstilling af [(1R), 2S]-2-aminopropionsyre 2-[4-(4-fluor-2-methyl-1H-indol-5-yloxy)-5-methylpyrrol]2,1-f-[1,2,4-triazin-6-yloxy]-1-methylethylester

Info

Publication number: DK2010538T3
Authority: DK; Denmark
Prior art keywords: yloxy; methylpyrrole; triazin; indol; fluoro
Prior art date: 2006-04-21

Application number

DK07760872.7T

Other languages

English (en)

Inventor

Gerard A Crispino

Mourad Hamedi

Thomas L Laporte

John E Thornton

Jaan A Pesti

Zhongmin Xu

Paul C Lobben

David K Leahy

Jale Muslehiddinoglu

Chiajen Lai

Robert P Discordia

Lori Ann Spangler

Original Assignee

Bristol Myers Squibb Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-04-21

Filing date

2007-04-19

Publication date

2013-03-18

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38357966&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK2010538(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2007-04-19 Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co

2013-03-18 Application granted granted Critical

2013-03-18 Publication of DK2010538T3 publication Critical patent/DK2010538T3/da

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

DK07760872.7T 2006-04-21 2007-04-19 Fremgangsmåde til fremstilling af [(1R), 2S]-2-aminopropionsyre 2-[4-(4-fluor-2-methyl-1H-indol-5-yloxy)-5-methylpyrrol]2,1-f-[1,2,4-triazin-6-yloxy]-1-methylethylester DK2010538T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US74530006P	2006-04-21	2006-04-21
PCT/US2007/066911 WO2007124332A1 (en)	2006-04-21	2007-04-19	PROCESS FOR THE PREPARATION OF [(1R), 2S]-2-AMINOPROPIONIC ACID 2-[4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLO[2,1-f][1,2,4]TRIAZIN-6-YLOXY]-1-METHYLETHYL ESTER

Publications (1)

Publication Number	Publication Date
DK2010538T3 true DK2010538T3 (da)	2013-03-18

Family

ID=38357966

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK07760872.7T DK2010538T3 (da)	2006-04-21	2007-04-19	Fremgangsmåde til fremstilling af [(1R), 2S]-2-aminopropionsyre 2-[4-(4-fluor-2-methyl-1H-indol-5-yloxy)-5-methylpyrrol]2,1-f-[1,2,4-triazin-6-yloxy]-1-methylethylester

Country Status (23)

Country	Link
US (1)	US7671199B2 (da)
EP (1)	EP2010538B1 (da)
JP (1)	JP5203353B2 (da)
KR (1)	KR101423789B1 (da)
CN (1)	CN101472927B (da)
AR (1)	AR060622A1 (da)
AU (1)	AU2007240453B2 (da)
BR (1)	BRPI0710691A2 (da)
CA (1)	CA2650059A1 (da)
CL (2)	CL2007001141A1 (da)
DK (1)	DK2010538T3 (da)
EA (1)	EA019693B1 (da)
ES (1)	ES2399379T3 (da)
HR (1)	HRP20130099T1 (da)
IL (1)	IL194715A (da)
MX (1)	MX2008013232A (da)
NO (1)	NO20084326L (da)
PE (1)	PE20080193A1 (da)
PL (1)	PL2010538T3 (da)
PT (1)	PT2010538E (da)
SI (1)	SI2010538T1 (da)
TW (1)	TWI378100B (da)
WO (1)	WO2007124332A1 (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2007038648A1 (en) *	2005-09-27	2007-04-05	Bristol-Myers Squibb Company	Crystalline forms of [(1r), 2s]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1h-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy]-1-methylethyl ester
US20120135875A1 (en) *	2008-02-29	2012-05-31	Bristol-Myers Squibb Company	Methods for determining sensitivity to vascular endothelial growth factor receptor-2 modulators
AR074830A1 (es)	2008-12-19	2011-02-16	Cephalon Inc	Pirrolotriazinas como inhibidores de alk y jak2
EP3864418A1 (en)	2018-10-08	2021-08-18	Applied Photophysics Limited	System and method for analysing the composition of a quenched flow reaction liquid

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6982265B1 (en) *	1999-05-21	2006-01-03	Bristol Myers Squibb Company	Pyrrolotriazine inhibitors of kinases
TWI329112B (en) *	2002-07-19	2010-08-21	Bristol Myers Squibb Co	Novel inhibitors of kinases
TWI272271B (en) *	2002-07-19	2007-02-01	Bristol Myers Squibb Co	Process for preparing certain pyrrolotriazine compounds
US7173031B2 (en) *	2004-06-28	2007-02-06	Bristol-Myers Squibb Company	Pyrrolotriazine kinase inhibitors
US7432373B2 (en) *	2004-06-28	2008-10-07	Bristol-Meyers Squibb Company	Processes and intermediates useful for preparing fused heterocyclic kinase inhibitors
WO2006130657A2 (en) *	2005-05-31	2006-12-07	Bristol-Myers Squibb Company	Stereoselective reduction process for the preparation of pyrrolotriazine compounds
WO2007038648A1 (en) *	2005-09-27	2007-04-05	Bristol-Myers Squibb Company	Crystalline forms of [(1r), 2s]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1h-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy]-1-methylethyl ester

2007
- 2007-04-19 PT PT77608727T patent/PT2010538E/pt unknown
- 2007-04-19 ES ES07760872T patent/ES2399379T3/es active Active
- 2007-04-19 DK DK07760872.7T patent/DK2010538T3/da active
- 2007-04-19 EA EA200802171A patent/EA019693B1/ru not_active IP Right Cessation
- 2007-04-19 EP EP07760872A patent/EP2010538B1/en active Active
- 2007-04-19 KR KR1020087025577A patent/KR101423789B1/ko active IP Right Grant
- 2007-04-19 MX MX2008013232A patent/MX2008013232A/es active IP Right Grant
- 2007-04-19 BR BRPI0710691-2A patent/BRPI0710691A2/pt not_active IP Right Cessation
- 2007-04-19 CA CA002650059A patent/CA2650059A1/en not_active Abandoned
- 2007-04-19 SI SI200731167T patent/SI2010538T1/sl unknown
- 2007-04-19 JP JP2009506761A patent/JP5203353B2/ja not_active Expired - Fee Related
- 2007-04-19 CN CN2007800232897A patent/CN101472927B/zh active Active
- 2007-04-19 PL PL07760872T patent/PL2010538T3/pl unknown
- 2007-04-19 WO PCT/US2007/066911 patent/WO2007124332A1/en active Application Filing
- 2007-04-19 AU AU2007240453A patent/AU2007240453B2/en not_active Ceased
- 2007-04-20 PE PE2007000492A patent/PE20080193A1/es not_active Application Discontinuation
- 2007-04-20 TW TW096114144A patent/TWI378100B/zh not_active IP Right Cessation
- 2007-04-20 US US11/737,787 patent/US7671199B2/en active Active
- 2007-04-20 CL CL2007001141A patent/CL2007001141A1/es unknown
- 2007-04-20 AR ARP070101727A patent/AR060622A1/es unknown
2008
- 2008-10-12 IL IL194715A patent/IL194715A/en not_active IP Right Cessation
- 2008-10-16 NO NO20084326A patent/NO20084326L/no not_active Application Discontinuation
2010
- 2010-05-28 CL CL2010000554A patent/CL2010000554A1/es unknown
2013
- 2013-02-05 HR HRP20130099TT patent/HRP20130099T1/hr unknown

Also Published As

Publication number	Publication date
AU2007240453B2 (en)	2012-04-12
HRP20130099T1 (hr)	2013-03-31
MX2008013232A (es)	2008-10-21
TWI378100B (en)	2012-12-01
EP2010538A1 (en)	2009-01-07
WO2007124332A1 (en)	2007-11-01
PT2010538E (pt)	2013-02-22
CN101472927A (zh)	2009-07-01
AU2007240453A1 (en)	2007-11-01
AR060622A1 (es)	2008-07-02
US7671199B2 (en)	2010-03-02
JP2009534413A (ja)	2009-09-24
BRPI0710691A2 (pt)	2011-08-23
TW200808799A (en)	2008-02-16
CL2007001141A1 (es)	2008-01-18
JP5203353B2 (ja)	2013-06-05
CN101472927B (zh)	2012-07-04
PL2010538T3 (pl)	2013-04-30
PE20080193A1 (es)	2008-03-10
KR101423789B1 (ko)	2014-07-30
IL194715A (en)	2013-10-31
KR20090008246A (ko)	2009-01-21
EA200802171A1 (ru)	2009-08-28
EA019693B1 (ru)	2014-05-30
CL2010000554A1 (es)	2010-10-15
NO20084326L (no)	2008-11-18
CA2650059A1 (en)	2007-11-01
ES2399379T3 (es)	2013-04-01
US20070249610A1 (en)	2007-10-25
SI2010538T1 (sl)	2013-06-28
EP2010538B1 (en)	2012-12-05

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