DK0714395T3 - Substituerede dihydropyranopyridiner med vasokonstriktoraktivitet - Google Patents

Substituerede dihydropyranopyridiner med vasokonstriktoraktivitet

Info

Publication number
DK0714395T3
DK0714395T3 DK94924873T DK94924873T DK0714395T3 DK 0714395 T3 DK0714395 T3 DK 0714395T3 DK 94924873 T DK94924873 T DK 94924873T DK 94924873 T DK94924873 T DK 94924873T DK 0714395 T3 DK0714395 T3 DK 0714395T3
Authority
DK
Denmark
Prior art keywords
6alkyl
hydrogen
pct
formula
radical
Prior art date
Application number
DK94924873T
Other languages
English (en)
Inventor
Lommen Guy Rosalia Eugene Van
Francisco Javi Fernandez-Gadea
Jose Ignacio Vesubi Andres-Gil
Maria Enc Matesanz-Ballesteros
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Application granted granted Critical
Publication of DK0714395T3 publication Critical patent/DK0714395T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/02Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyridine Compounds (AREA)
DK94924873T 1993-08-19 1994-08-12 Substituerede dihydropyranopyridiner med vasokonstriktoraktivitet DK0714395T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP93202440 1993-08-19
PCT/EP1994/002700 WO1995005381A1 (en) 1993-08-19 1994-08-12 Vasoconstrictive substituted dihydropyranopyridines

Publications (1)

Publication Number Publication Date
DK0714395T3 true DK0714395T3 (da) 1999-10-11

Family

ID=8214053

Family Applications (1)

Application Number Title Priority Date Filing Date
DK94924873T DK0714395T3 (da) 1993-08-19 1994-08-12 Substituerede dihydropyranopyridiner med vasokonstriktoraktivitet

Country Status (27)

Country Link
US (1) US5691344A (da)
EP (1) EP0714395B1 (da)
JP (1) JP3650398B2 (da)
KR (1) KR100330697B1 (da)
CN (1) CN1051085C (da)
AT (1) ATE178330T1 (da)
AU (1) AU684819B2 (da)
BR (1) BR9407298A (da)
CA (1) CA2168022C (da)
CZ (1) CZ286645B6 (da)
DE (1) DE69417560T2 (da)
DK (1) DK0714395T3 (da)
ES (1) ES2132424T3 (da)
FI (1) FI113773B (da)
GR (1) GR3029924T3 (da)
HU (1) HU228673B1 (da)
IL (1) IL110688A (da)
MY (1) MY111419A (da)
NO (1) NO315001B1 (da)
NZ (1) NZ271383A (da)
PL (1) PL177516B1 (da)
RO (1) RO116729B1 (da)
RU (1) RU2135501C1 (da)
SI (1) SI0714395T1 (da)
SK (1) SK282108B6 (da)
WO (1) WO1995005381A1 (da)
ZA (1) ZA946268B (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6818659B2 (en) 2001-11-06 2004-11-16 Bristol-Myers Squibb Pharma, Inc. (2S)-2-amino-4-(2-amino-(3,4,5,6-tetrahydropyrimidin-4-yl) butanoyl and its use in cyclic and acyclic peptides
JP7171444B2 (ja) * 2016-07-01 2022-11-15 ヤンセン・サイエンシズ・アイルランド・アンリミテッド・カンパニー ウイルス感染治療用のジヒドロピラノピリミジン

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU576868B2 (en) * 1984-06-11 1988-09-08 E.I. Du Pont De Nemours And Company Thiophene and pyridine sulfonamides
CH674984A5 (da) * 1987-05-16 1990-08-15 Sandoz Ag
DE3901814A1 (de) * 1988-07-28 1990-02-01 Bayer Ag Substituierte aminomethylzetraline sowie ihre heterocyclischen analoga
US5140031A (en) * 1989-05-31 1992-08-18 E. R. Squibb & Sons, Inc. Pyranyl cyanoguanidine derivatives
US5250450A (en) * 1991-04-08 1993-10-05 Micron Technology, Inc. Insulated-gate vertical field-effect transistor with high current drive and minimum overlap capacitance
DE4120322A1 (de) * 1991-06-20 1992-12-24 Bayer Ag Aminomethyl-substituierte 2,3-dihydropyrano(2,3-b)pyridine, verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln
SI9300097B (en) * 1992-02-27 2001-12-31 Janssen Pharmaceutica Nv (benzodioxan, benzofuran or benzopyran) alkylamino) alkyl substituted guanidines

Also Published As

Publication number Publication date
IL110688A (en) 1998-10-30
MY111419A (en) 2000-04-29
GR3029924T3 (en) 1999-07-30
FI113773B (fi) 2004-06-15
KR100330697B1 (ko) 2002-10-04
CZ37396A3 (en) 1996-05-15
RU2135501C1 (ru) 1999-08-27
SK19496A3 (en) 1997-02-05
NZ271383A (en) 1997-05-26
PL177516B1 (pl) 1999-12-31
CA2168022C (en) 2006-11-21
IL110688A0 (en) 1994-11-11
NO960647L (no) 1996-02-19
HU9600374D0 (en) 1996-04-29
US5691344A (en) 1997-11-25
SI0714395T1 (en) 1999-08-31
AU7499594A (en) 1995-03-14
ZA946268B (en) 1996-02-19
JP3650398B2 (ja) 2005-05-18
PL313080A1 (en) 1996-05-27
ATE178330T1 (de) 1999-04-15
NO315001B1 (no) 2003-06-23
NO960647D0 (no) 1996-02-19
FI960721A (fi) 1996-02-16
CA2168022A1 (en) 1995-02-23
RO116729B1 (ro) 2001-05-30
SK282108B6 (sk) 2001-11-06
EP0714395A1 (en) 1996-06-05
CN1129943A (zh) 1996-08-28
HU228673B1 (en) 2013-05-28
HUT74676A (en) 1997-01-28
WO1995005381A1 (en) 1995-02-23
DE69417560T2 (de) 1999-11-11
FI960721A0 (fi) 1996-02-16
ES2132424T3 (es) 1999-08-16
AU684819B2 (en) 1998-01-08
JPH09501669A (ja) 1997-02-18
DE69417560D1 (de) 1999-05-06
EP0714395B1 (en) 1999-03-31
CN1051085C (zh) 2000-04-05
BR9407298A (pt) 1996-10-01
CZ286645B6 (cs) 2000-05-17

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