DE69910186D1 - Pharmazeutische zusammensetzung von topiramate - Google Patents

Pharmazeutische zusammensetzung von topiramate

Info

Publication number
DE69910186D1
DE69910186D1 DE69910186T DE69910186T DE69910186D1 DE 69910186 D1 DE69910186 D1 DE 69910186D1 DE 69910186 T DE69910186 T DE 69910186T DE 69910186 T DE69910186 T DE 69910186T DE 69910186 D1 DE69910186 D1 DE 69910186D1
Authority
DE
Germany
Prior art keywords
topiramate
pharmaceutical composition
pharmaceutical
composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Revoked
Application number
DE69910186T
Other languages
English (en)
Other versions
DE69910186T2 (de
Inventor
S Thakur
M Kotwal
S Gibbs
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Janssen Pharmaceuticals Inc
Original Assignee
Ortho McNeil Pharmaceutical Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22134079&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE69910186(D1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ortho McNeil Pharmaceutical Inc filed Critical Ortho McNeil Pharmaceutical Inc
Application granted granted Critical
Publication of DE69910186D1 publication Critical patent/DE69910186D1/de
Publication of DE69910186T2 publication Critical patent/DE69910186T2/de
Anticipated expiration legal-status Critical
Revoked legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
    • A61K9/1676—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface having a drug-free core with discrete complete coating layer containing drug
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846—Poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Molecular Biology (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DE69910186T 1998-03-04 1999-03-01 Pharmazeutische zusammensetzung von topiramate Revoked DE69910186T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US7677098P 1998-03-04 1998-03-04
US76770P 1998-03-04
PCT/US1999/004449 WO1999044581A2 (en) 1998-03-04 1999-03-01 Pharmaceutical composition of topiramate

Publications (2)

Publication Number Publication Date
DE69910186D1 true DE69910186D1 (de) 2003-09-11
DE69910186T2 DE69910186T2 (de) 2004-07-29

Family

ID=22134079

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69910186T Revoked DE69910186T2 (de) 1998-03-04 1999-03-01 Pharmazeutische zusammensetzung von topiramate

Country Status (32)

Country Link
US (4) US6696091B2 (de)
EP (1) EP1066027B1 (de)
JP (1) JP2003530295A (de)
KR (1) KR20010041592A (de)
CN (1) CN100364501C (de)
AR (3) AR017984A1 (de)
AT (1) ATE246490T1 (de)
AU (1) AU763643B2 (de)
BG (1) BG64885B1 (de)
BR (1) BR9908488A (de)
CA (1) CA2322644C (de)
DE (1) DE69910186T2 (de)
DK (1) DK1066027T3 (de)
EA (1) EA200000814A1 (de)
EE (1) EE04175B1 (de)
ES (1) ES2204109T3 (de)
HK (1) HK1032009A1 (de)
HR (1) HRP20000563B1 (de)
HU (1) HUP0301192A3 (de)
ID (1) ID26982A (de)
IL (2) IL138032A0 (de)
MY (1) MY125821A (de)
NO (1) NO20004311L (de)
NZ (1) NZ506532A (de)
PL (1) PL194559B1 (de)
PT (1) PT1066027E (de)
SK (1) SK285440B6 (de)
TR (1) TR200002541T2 (de)
TW (1) TW590778B (de)
UA (1) UA65607C2 (de)
WO (1) WO1999044581A2 (de)
ZA (1) ZA991716B (de)

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CA2322644C (en) 2005-07-26
AU763643B2 (en) 2003-07-31
WO1999044581A2 (en) 1999-09-10
KR20010041592A (ko) 2001-05-25
IL138032A0 (en) 2001-10-31
ATE246490T1 (de) 2003-08-15
HRP20000563A2 (en) 2001-04-30
PT1066027E (pt) 2003-12-31
TR200002541T2 (tr) 2001-03-21
CA2322644A1 (en) 1999-09-10
PL194559B1 (pl) 2007-06-29
US7125560B2 (en) 2006-10-24
DK1066027T3 (da) 2003-11-10
AR017984A1 (es) 2001-10-24
AU2798999A (en) 1999-09-20
UA65607C2 (uk) 2004-04-15
NO20004311D0 (no) 2000-08-30
AR048456A2 (es) 2006-04-26
IL138032A (en) 2007-09-20
BR9908488A (pt) 2000-12-05
EE200000503A (et) 2002-02-15
MY125821A (en) 2006-08-30
CN1419444A (zh) 2003-05-21
NO20004311L (no) 2000-10-25
HUP0301192A3 (en) 2004-03-01
TW590778B (en) 2004-06-11
SK13062000A3 (sk) 2001-04-09
BG64885B1 (bg) 2006-08-31
US20080260813A1 (en) 2008-10-23
EP1066027B1 (de) 2003-08-06
EA200000814A1 (ru) 2001-02-26
US20020064563A1 (en) 2002-05-30
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AR048457A2 (es) 2006-04-26
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EP1066027A1 (de) 2001-01-10
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ES2204109T3 (es) 2004-04-16
US6696091B2 (en) 2004-02-24
US20060286163A1 (en) 2006-12-21
US20040156901A1 (en) 2004-08-12
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