DE69328975T2 - Aminomethylen substituierte heterocyclische verbindungen und ihre verwendung alssubstanz p antagonisten - Google Patents

Aminomethylen substituierte heterocyclische verbindungen und ihre verwendung alssubstanz p antagonisten

Info

Publication number
DE69328975T2
DE69328975T2 DE69328975T DE69328975T DE69328975T2 DE 69328975 T2 DE69328975 T2 DE 69328975T2 DE 69328975 T DE69328975 T DE 69328975T DE 69328975 T DE69328975 T DE 69328975T DE 69328975 T2 DE69328975 T2 DE 69328975T2
Authority
DE
Germany
Prior art keywords
antagonists
substance
substituted heterocyclic
heterocyclic compounds
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69328975T
Other languages
English (en)
Other versions
DE69328975D1 (de
Inventor
R Howard
T O'neill
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Application granted granted Critical
Publication of DE69328975D1 publication Critical patent/DE69328975D1/de
Publication of DE69328975T2 publication Critical patent/DE69328975T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, ***e
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
DE69328975T 1992-12-10 1993-10-07 Aminomethylen substituierte heterocyclische verbindungen und ihre verwendung alssubstanz p antagonisten Expired - Fee Related DE69328975T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US98865392A 1992-12-10 1992-12-10
PCT/US1993/009407 WO1994013663A1 (en) 1992-12-10 1993-10-07 Aminomethylene substituted non-aromatic heterocycles and use as substance p antagonists

Publications (2)

Publication Number Publication Date
DE69328975D1 DE69328975D1 (de) 2000-08-10
DE69328975T2 true DE69328975T2 (de) 2000-11-09

Family

ID=25534364

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69328975T Expired - Fee Related DE69328975T2 (de) 1992-12-10 1993-10-07 Aminomethylen substituierte heterocyclische verbindungen und ihre verwendung alssubstanz p antagonisten

Country Status (15)

Country Link
EP (2) EP0806423A1 (de)
JP (2) JP2722279B2 (de)
CN (1) CN1092771A (de)
AT (1) ATE194340T1 (de)
AU (1) AU5169693A (de)
CA (1) CA2150123C (de)
DE (1) DE69328975T2 (de)
DK (1) DK0675886T3 (de)
ES (1) ES2147759T3 (de)
FI (1) FI935529A (de)
GR (1) GR3034329T3 (de)
IL (1) IL107843A0 (de)
MX (1) MX9307810A (de)
PT (1) PT675886E (de)
WO (1) WO1994013663A1 (de)

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Also Published As

Publication number Publication date
FI935529A (fi) 1994-06-11
PT675886E (pt) 2000-12-29
JPH07509490A (ja) 1995-10-19
ATE194340T1 (de) 2000-07-15
DK0675886T3 (da) 2000-09-18
CA2150123C (en) 2004-12-07
ES2147759T3 (es) 2000-10-01
EP0806423A1 (de) 1997-11-12
EP0675886B1 (de) 2000-07-05
FI935529A0 (fi) 1993-12-09
IL107843A0 (en) 1994-04-12
MX9307810A (es) 1994-07-29
DE69328975D1 (de) 2000-08-10
JP3165401B2 (ja) 2001-05-14
WO1994013663A1 (en) 1994-06-23
CA2150123A1 (en) 1994-06-23
JP2722279B2 (ja) 1998-03-04
JPH1095780A (ja) 1998-04-14
EP0675886A1 (de) 1995-10-11
CN1092771A (zh) 1994-09-28
GR3034329T3 (en) 2000-12-29
AU5169693A (en) 1994-07-04

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