DE602004014640D1 - Tricyclische modulatoren von nuklearen steroidhormonrezeptoren - Google Patents

Tricyclische modulatoren von nuklearen steroidhormonrezeptoren

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Publication number
DE602004014640D1
DE602004014640D1 DE602004014640T DE602004014640T DE602004014640D1 DE 602004014640 D1 DE602004014640 D1 DE 602004014640D1 DE 602004014640 T DE602004014640 T DE 602004014640T DE 602004014640 T DE602004014640 T DE 602004014640T DE 602004014640 D1 DE602004014640 D1 DE 602004014640D1
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DE
Germany
Prior art keywords
tricyclic
modulators
steroid hormone
hormone receptors
nuclear steroid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
DE602004014640T
Other languages
English (en)
Inventor
Konstantinos Gavardinas
Jonathan Edward Green
Prabhakar Kondaji Jadhav
Donald P Matthews
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of DE602004014640D1 publication Critical patent/DE602004014640D1/de
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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    • C07—ORGANIC CHEMISTRY
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    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/26—Oxygen atoms
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DE602004014640T 2003-12-19 2004-12-08 Tricyclische modulatoren von nuklearen steroidhormonrezeptoren Active DE602004014640D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US53128303P 2003-12-19 2003-12-19
PCT/US2004/038233 WO2005066161A1 (en) 2003-12-19 2004-12-08 Tricyclic steroid hormone nuclear receptor modulators

Publications (1)

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DE602004014640D1 true DE602004014640D1 (de) 2008-08-07

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DE602004014640T Active DE602004014640D1 (de) 2003-12-19 2004-12-08 Tricyclische modulatoren von nuklearen steroidhormonrezeptoren

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US (1) US7803814B2 (de)
EP (1) EP1697350B1 (de)
JP (1) JP4846596B2 (de)
CN (1) CN1918151A (de)
AR (1) AR046951A1 (de)
AT (1) ATE399163T1 (de)
AU (1) AU2004312293A1 (de)
BR (1) BRPI0416882A (de)
CA (1) CA2549053C (de)
CY (1) CY1108309T1 (de)
DE (1) DE602004014640D1 (de)
DK (1) DK1697350T3 (de)
ES (1) ES2308296T3 (de)
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DK1697350T3 (da) 2008-10-13
CA2549053C (en) 2012-08-28
CA2549053A1 (en) 2005-07-21
EP1697350B1 (de) 2008-06-25
JP2007515431A (ja) 2007-06-14
EP1697350A1 (de) 2006-09-06
IL175996A0 (en) 2006-10-05
ES2308296T3 (es) 2008-12-01
PT1697350E (pt) 2008-09-18
NO20063329L (no) 2006-09-14
US20070037788A1 (en) 2007-02-15
WO2005066161A1 (en) 2005-07-21
ZA200604889B (en) 2007-11-28
BRPI0416882A (pt) 2007-02-27
CN1918151A (zh) 2007-02-21
SI1697350T1 (sl) 2008-12-31
CY1108309T1 (el) 2014-02-12
PL1697350T3 (pl) 2008-11-28
JP4846596B2 (ja) 2011-12-28
ATE399163T1 (de) 2008-07-15
US7803814B2 (en) 2010-09-28
AU2004312293A1 (en) 2005-07-21
MXPA06007055A (es) 2007-01-30

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