NO20063329L - Tricykliske steroidhormone nukleaer reseptormodulatorer - Google Patents

Tricykliske steroidhormone nukleaer reseptormodulatorer

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Publication number
NO20063329L
NO20063329L NO20063329A NO20063329A NO20063329L NO 20063329 L NO20063329 L NO 20063329L NO 20063329 A NO20063329 A NO 20063329A NO 20063329 A NO20063329 A NO 20063329A NO 20063329 L NO20063329 L NO 20063329L
Authority
NO
Norway
Prior art keywords
receptor modulators
nuclear receptor
steroid hormone
compound
formula
Prior art date
Application number
NO20063329A
Other languages
English (en)
Inventor
Donald Paul Matthews
Jonathan Edward Green
Prabhakar Kondaji Jadhav
Konstantinos Gavardinas
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of NO20063329L publication Critical patent/NO20063329L/no

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/26—Oxygen atoms
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Abstract

Foreliggende oppfinnelse tilveiebringer en forbindelse med Formel (I): eller et farmasøytisk akseptabelt salt derav; farmasøytiske sammensetninger som innbefatter en effektiv mengde av en forbindelse med Formel (I) i kombinasjon med en egnet bærer, fortynningsmiddel eller eksipient; fremgangsmåter for behandling av fysiologiske forstyrrelser, særlig kongestiv hjertesvikt, hypertensjon, reumatoid artritt eller inflammasjon, som innbefatter administrering til en pasient som trenger det av en effektiv mengde av en forbindelse med Formel (I).
NO20063329A 2003-12-19 2006-07-18 Tricykliske steroidhormone nukleaer reseptormodulatorer NO20063329L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US53128303P 2003-12-19 2003-12-19
PCT/US2004/038233 WO2005066161A1 (en) 2003-12-19 2004-12-08 Tricyclic steroid hormone nuclear receptor modulators

Publications (1)

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NO20063329L true NO20063329L (no) 2006-09-14

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ID=34748755

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20063329A NO20063329L (no) 2003-12-19 2006-07-18 Tricykliske steroidhormone nukleaer reseptormodulatorer

Country Status (21)

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US (1) US7803814B2 (no)
EP (1) EP1697350B1 (no)
JP (1) JP4846596B2 (no)
CN (1) CN1918151A (no)
AR (1) AR046951A1 (no)
AT (1) ATE399163T1 (no)
AU (1) AU2004312293A1 (no)
BR (1) BRPI0416882A (no)
CA (1) CA2549053C (no)
CY (1) CY1108309T1 (no)
DE (1) DE602004014640D1 (no)
DK (1) DK1697350T3 (no)
ES (1) ES2308296T3 (no)
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EP1697350B1 (en) 2008-06-25
JP4846596B2 (ja) 2011-12-28
WO2005066161A1 (en) 2005-07-21
EP1697350A1 (en) 2006-09-06
PT1697350E (pt) 2008-09-18
CA2549053A1 (en) 2005-07-21
PL1697350T3 (pl) 2008-11-28
DK1697350T3 (da) 2008-10-13
DE602004014640D1 (de) 2008-08-07
CN1918151A (zh) 2007-02-21
MXPA06007055A (es) 2007-01-30
CY1108309T1 (el) 2014-02-12
CA2549053C (en) 2012-08-28
IL175996A0 (en) 2006-10-05
AR046951A1 (es) 2006-01-04
ATE399163T1 (de) 2008-07-15
SI1697350T1 (sl) 2008-12-31
AU2004312293A1 (en) 2005-07-21
ZA200604889B (en) 2007-11-28
ES2308296T3 (es) 2008-12-01
BRPI0416882A (pt) 2007-02-27
US20070037788A1 (en) 2007-02-15
US7803814B2 (en) 2010-09-28

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