NO20063329L - Tricykliske steroidhormone nukleaer reseptormodulatorer - Google Patents
Tricykliske steroidhormone nukleaer reseptormodulatorerInfo
- Publication number
- NO20063329L NO20063329L NO20063329A NO20063329A NO20063329L NO 20063329 L NO20063329 L NO 20063329L NO 20063329 A NO20063329 A NO 20063329A NO 20063329 A NO20063329 A NO 20063329A NO 20063329 L NO20063329 L NO 20063329L
- Authority
- NO
- Norway
- Prior art keywords
- receptor modulators
- nuclear receptor
- steroid hormone
- compound
- formula
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/26—Oxygen atoms
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Diabetes (AREA)
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- Neurosurgery (AREA)
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- Obesity (AREA)
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Abstract
Foreliggende oppfinnelse tilveiebringer en forbindelse med Formel (I): eller et farmasøytisk akseptabelt salt derav; farmasøytiske sammensetninger som innbefatter en effektiv mengde av en forbindelse med Formel (I) i kombinasjon med en egnet bærer, fortynningsmiddel eller eksipient; fremgangsmåter for behandling av fysiologiske forstyrrelser, særlig kongestiv hjertesvikt, hypertensjon, reumatoid artritt eller inflammasjon, som innbefatter administrering til en pasient som trenger det av en effektiv mengde av en forbindelse med Formel (I).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US53128303P | 2003-12-19 | 2003-12-19 | |
PCT/US2004/038233 WO2005066161A1 (en) | 2003-12-19 | 2004-12-08 | Tricyclic steroid hormone nuclear receptor modulators |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20063329L true NO20063329L (no) | 2006-09-14 |
Family
ID=34748755
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20063329A NO20063329L (no) | 2003-12-19 | 2006-07-18 | Tricykliske steroidhormone nukleaer reseptormodulatorer |
Country Status (21)
Country | Link |
---|---|
US (1) | US7803814B2 (no) |
EP (1) | EP1697350B1 (no) |
JP (1) | JP4846596B2 (no) |
CN (1) | CN1918151A (no) |
AR (1) | AR046951A1 (no) |
AT (1) | ATE399163T1 (no) |
AU (1) | AU2004312293A1 (no) |
BR (1) | BRPI0416882A (no) |
CA (1) | CA2549053C (no) |
CY (1) | CY1108309T1 (no) |
DE (1) | DE602004014640D1 (no) |
DK (1) | DK1697350T3 (no) |
ES (1) | ES2308296T3 (no) |
IL (1) | IL175996A0 (no) |
MX (1) | MXPA06007055A (no) |
NO (1) | NO20063329L (no) |
PL (1) | PL1697350T3 (no) |
PT (1) | PT1697350E (no) |
SI (1) | SI1697350T1 (no) |
WO (1) | WO2005066161A1 (no) |
ZA (1) | ZA200604889B (no) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200400816A (en) * | 2002-06-26 | 2004-01-16 | Lilly Co Eli | Tricyclic steroid hormone nuclear receptor modulators |
WO2006071750A1 (en) * | 2004-12-23 | 2006-07-06 | Athersys, Inc. | 4-piperidinol tertiary amines as histamine 3 receptor inhibitors for the treatment of obesity and other cns disorders |
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2004
- 2004-12-08 US US10/576,761 patent/US7803814B2/en not_active Expired - Fee Related
- 2004-12-08 AT AT04811084T patent/ATE399163T1/de not_active IP Right Cessation
- 2004-12-08 EP EP04811084A patent/EP1697350B1/en not_active Not-in-force
- 2004-12-08 CN CNA2004800418534A patent/CN1918151A/zh active Pending
- 2004-12-08 WO PCT/US2004/038233 patent/WO2005066161A1/en active Application Filing
- 2004-12-08 AU AU2004312293A patent/AU2004312293A1/en not_active Abandoned
- 2004-12-08 BR BRPI0416882-8A patent/BRPI0416882A/pt not_active Application Discontinuation
- 2004-12-08 SI SI200430840T patent/SI1697350T1/sl unknown
- 2004-12-08 MX MXPA06007055A patent/MXPA06007055A/es unknown
- 2004-12-08 CA CA2549053A patent/CA2549053C/en not_active Expired - Fee Related
- 2004-12-08 DK DK04811084T patent/DK1697350T3/da active
- 2004-12-08 JP JP2006545655A patent/JP4846596B2/ja not_active Expired - Fee Related
- 2004-12-08 PT PT04811084T patent/PT1697350E/pt unknown
- 2004-12-08 DE DE602004014640T patent/DE602004014640D1/de active Active
- 2004-12-08 ES ES04811084T patent/ES2308296T3/es active Active
- 2004-12-08 PL PL04811084T patent/PL1697350T3/pl unknown
- 2004-12-17 AR ARP040104730A patent/AR046951A1/es unknown
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2006
- 2006-05-29 IL IL175996A patent/IL175996A0/en unknown
- 2006-06-13 ZA ZA200604889A patent/ZA200604889B/en unknown
- 2006-07-18 NO NO20063329A patent/NO20063329L/no not_active Application Discontinuation
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Also Published As
Publication number | Publication date |
---|---|
JP2007515431A (ja) | 2007-06-14 |
EP1697350B1 (en) | 2008-06-25 |
JP4846596B2 (ja) | 2011-12-28 |
WO2005066161A1 (en) | 2005-07-21 |
EP1697350A1 (en) | 2006-09-06 |
PT1697350E (pt) | 2008-09-18 |
CA2549053A1 (en) | 2005-07-21 |
PL1697350T3 (pl) | 2008-11-28 |
DK1697350T3 (da) | 2008-10-13 |
DE602004014640D1 (de) | 2008-08-07 |
CN1918151A (zh) | 2007-02-21 |
MXPA06007055A (es) | 2007-01-30 |
CY1108309T1 (el) | 2014-02-12 |
CA2549053C (en) | 2012-08-28 |
IL175996A0 (en) | 2006-10-05 |
AR046951A1 (es) | 2006-01-04 |
ATE399163T1 (de) | 2008-07-15 |
SI1697350T1 (sl) | 2008-12-31 |
AU2004312293A1 (en) | 2005-07-21 |
ZA200604889B (en) | 2007-11-28 |
ES2308296T3 (es) | 2008-12-01 |
BRPI0416882A (pt) | 2007-02-27 |
US20070037788A1 (en) | 2007-02-15 |
US7803814B2 (en) | 2010-09-28 |
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