DE2661014C2 - - Google Patents
Info
- Publication number
- DE2661014C2 DE2661014C2 DE2661014A DE2661014A DE2661014C2 DE 2661014 C2 DE2661014 C2 DE 2661014C2 DE 2661014 A DE2661014 A DE 2661014A DE 2661014 A DE2661014 A DE 2661014A DE 2661014 C2 DE2661014 C2 DE 2661014C2
- Authority
- DE
- Germany
- Prior art keywords
- pyrrolo
- cyan
- benzazepin
- water
- acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/325—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
- C07D207/327—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/38—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to acyclic carbon atoms and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/24—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US59243675A | 1975-07-02 | 1975-07-02 |
Publications (2)
Publication Number | Publication Date |
---|---|
DE2661014A1 DE2661014A1 (sv) | 1985-07-04 |
DE2661014C2 true DE2661014C2 (sv) | 1989-01-05 |
Family
ID=24370639
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE2661014A Expired DE2661014C2 (sv) | 1975-07-02 | 1976-07-02 | |
DE19762629877 Granted DE2629877A1 (de) | 1975-07-02 | 1976-07-02 | Pyrrolo eckige klammer auf 2,1-b eckige klammer zu eckige klammer auf 3 eckige klammer zu benzazepine |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE19762629877 Granted DE2629877A1 (de) | 1975-07-02 | 1976-07-02 | Pyrrolo eckige klammer auf 2,1-b eckige klammer zu eckige klammer auf 3 eckige klammer zu benzazepine |
Country Status (18)
Country | Link |
---|---|
JP (1) | JPS527996A (sv) |
AU (1) | AU499122B2 (sv) |
BE (1) | BE843678A (sv) |
CA (1) | CA1092105A (sv) |
CH (5) | CH626366A5 (sv) |
CY (1) | CY1091A (sv) |
DE (2) | DE2661014C2 (sv) |
ES (1) | ES449432A1 (sv) |
FR (1) | FR2315935A1 (sv) |
GB (1) | GB1499047A (sv) |
GR (1) | GR60851B (sv) |
HK (1) | HK60580A (sv) |
HU (1) | HU177866B (sv) |
MY (1) | MY8100227A (sv) |
NL (1) | NL188287C (sv) |
PT (1) | PT65295B (sv) |
SE (1) | SE424076B (sv) |
ZA (1) | ZA763990B (sv) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4148903A (en) * | 1977-07-28 | 1979-04-10 | Merck & Co., Inc. | Antipsychotic, antiserotonin and antihistaminic pyrrolo[2,1-b][3]benzazepines |
JPH0487401U (sv) * | 1990-12-06 | 1992-07-29 | ||
US6271392B1 (en) | 1994-10-07 | 2001-08-07 | Rhone-Poulenc Inc. | Intermediates useful for the synthesis of 1-arylpyrrole pesticides |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3428677A (en) * | 1962-09-24 | 1969-02-18 | Merck & Co Inc | Chemical compounds and methods of preparing same |
US3499037A (en) * | 1966-05-31 | 1970-03-03 | Merck & Co Inc | Preparation of trifluoromethyl substituted dibenzocycloheptenes |
-
1976
- 1976-06-30 CA CA256,080A patent/CA1092105A/en not_active Expired
- 1976-06-30 PT PT65295A patent/PT65295B/pt unknown
- 1976-06-30 FR FR7619897A patent/FR2315935A1/fr active Granted
- 1976-07-01 ES ES449432A patent/ES449432A1/es not_active Expired
- 1976-07-01 GB GB27487/76A patent/GB1499047A/en not_active Expired
- 1976-07-01 AU AU15488/76A patent/AU499122B2/en not_active Expired
- 1976-07-01 BE BE168549A patent/BE843678A/xx not_active IP Right Cessation
- 1976-07-01 GR GR51162A patent/GR60851B/el unknown
- 1976-07-01 SE SE7607534A patent/SE424076B/sv not_active IP Right Cessation
- 1976-07-01 CY CY1091A patent/CY1091A/xx unknown
- 1976-07-01 CH CH844376A patent/CH626366A5/de not_active IP Right Cessation
- 1976-07-02 NL NLAANVRAGE7607347,A patent/NL188287C/xx not_active IP Right Cessation
- 1976-07-02 ZA ZA00763990A patent/ZA763990B/xx unknown
- 1976-07-02 HU HU76ME2001A patent/HU177866B/hu unknown
- 1976-07-02 DE DE2661014A patent/DE2661014C2/de not_active Expired
- 1976-07-02 JP JP51077992A patent/JPS527996A/ja active Granted
- 1976-07-02 DE DE19762629877 patent/DE2629877A1/de active Granted
-
1980
- 1980-05-16 CH CH386080A patent/CH626616A5/de not_active IP Right Cessation
- 1980-05-16 CH CH386180A patent/CH626617A5/de not_active IP Right Cessation
- 1980-05-16 CH CH386280A patent/CH626618A5/de not_active IP Right Cessation
- 1980-05-16 CH CH385980A patent/CH626893A5/de not_active IP Right Cessation
- 1980-10-30 HK HK605/80A patent/HK60580A/xx unknown
-
1981
- 1981-12-30 MY MY227/81A patent/MY8100227A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
DE2629877A1 (de) | 1977-01-20 |
NL7607347A (nl) | 1977-01-04 |
CA1092105A (en) | 1980-12-23 |
GB1499047A (en) | 1978-01-25 |
JPS527996A (en) | 1977-01-21 |
DE2661014A1 (sv) | 1985-07-04 |
GR60851B (en) | 1978-08-31 |
MY8100227A (en) | 1981-12-31 |
FR2315935A1 (fr) | 1977-01-28 |
CH626366A5 (en) | 1981-11-13 |
CY1091A (en) | 1980-12-27 |
AU499122B2 (en) | 1979-04-05 |
AU1548876A (en) | 1978-01-05 |
FR2315935B1 (sv) | 1978-11-17 |
JPH0132225B2 (sv) | 1989-06-29 |
BE843678A (fr) | 1977-01-03 |
PT65295A (en) | 1976-07-01 |
HK60580A (en) | 1980-11-07 |
SE424076B (sv) | 1982-06-28 |
CH626617A5 (en) | 1981-11-30 |
CH626616A5 (en) | 1981-11-30 |
NL188287B (nl) | 1991-12-16 |
DE2629877C2 (sv) | 1989-01-05 |
ZA763990B (en) | 1978-02-22 |
CH626893A5 (en) | 1981-12-15 |
HU177866B (en) | 1982-01-28 |
SE7607534L (sv) | 1977-01-03 |
CH626618A5 (en) | 1981-11-30 |
ES449432A1 (es) | 1977-12-16 |
PT65295B (en) | 1978-05-10 |
NL188287C (nl) | 1992-05-18 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
Q172 | Divided out of (supplement): |
Ref country code: DE Ref document number: 2629877 |
|
8110 | Request for examination paragraph 44 | ||
8181 | Inventor (new situation) |
Free format text: ROKACH, JOSHUA, CHOMEDEY LAVAL, QUEBEC, CA ATKINSON, JOSEPH GEORGE, MONTREAL, QUEBEC, CA ROONEY, CLARENCE STANLEY, BEACONSFIELD, QUEBEC, CA |
|
AC | Divided out of |
Ref country code: DE Ref document number: 2629877 Format of ref document f/p: P |
|
D2 | Grant after examination | ||
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |