CZ20011394A3 - Derivát bicyklických, dusík obsahujících heterocyklických sloučenin, způsob jeho přípravy a farmaceutický prostředek, který ho obsahuje - Google Patents

Derivát bicyklických, dusík obsahujících heterocyklických sloučenin, způsob jeho přípravy a farmaceutický prostředek, který ho obsahuje

Info

Publication number
CZ20011394A3
CZ20011394A3 CZ20011394A CZ20011394A CZ20011394A3 CZ 20011394 A3 CZ20011394 A3 CZ 20011394A3 CZ 20011394 A CZ20011394 A CZ 20011394A CZ 20011394 A CZ20011394 A CZ 20011394A CZ 20011394 A3 CZ20011394 A3 CZ 20011394A3
Authority
CZ
Czechia
Prior art keywords
lower alkyl
heteroaryl
aryl
cycloalkyl
preparation
Prior art date
Application number
CZ20011394A
Other languages
English (en)
Inventor
William Harris
Christopher Huw Hill
Ian Edward David Smith
Original Assignee
F. Hoffmann-La Roche Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26314565&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CZ20011394(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9823277.0A external-priority patent/GB9823277D0/en
Application filed by F. Hoffmann-La Roche Ag filed Critical F. Hoffmann-La Roche Ag
Publication of CZ20011394A3 publication Critical patent/CZ20011394A3/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Neurology (AREA)
  • Immunology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Inorganic Insulating Materials (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CZ20011394A 1998-10-23 1999-10-13 Derivát bicyklických, dusík obsahujících heterocyklických sloučenin, způsob jeho přípravy a farmaceutický prostředek, který ho obsahuje CZ20011394A3 (cs)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9823277.0A GB9823277D0 (en) 1998-10-23 1998-10-23 Bicycle nitrogen heterocycles
GBGB9920044.6A GB9920044D0 (en) 1998-10-23 1999-08-24 Biciclic nitrogen heterocycles

Publications (1)

Publication Number Publication Date
CZ20011394A3 true CZ20011394A3 (cs) 2001-12-12

Family

ID=26314565

Family Applications (1)

Application Number Title Priority Date Filing Date
CZ20011394A CZ20011394A3 (cs) 1998-10-23 1999-10-13 Derivát bicyklických, dusík obsahujících heterocyklických sloučenin, způsob jeho přípravy a farmaceutický prostředek, který ho obsahuje

Country Status (25)

Country Link
US (1) US6150373A (cs)
EP (1) EP1123295B1 (cs)
JP (1) JP3593035B2 (cs)
CN (1) CN1150195C (cs)
AT (1) ATE277931T1 (cs)
AU (1) AU769989B2 (cs)
BR (1) BR9914677A (cs)
CA (1) CA2347474C (cs)
CZ (1) CZ20011394A3 (cs)
DE (1) DE69920732T2 (cs)
ES (1) ES2228123T3 (cs)
HK (1) HK1041483B (cs)
HR (1) HRP20010274A2 (cs)
HU (1) HUP0104199A3 (cs)
ID (1) ID28276A (cs)
MA (1) MA27678A1 (cs)
MY (1) MY126478A (cs)
NO (1) NO318802B1 (cs)
NZ (1) NZ510760A (cs)
PL (1) PL347432A1 (cs)
PT (1) PT1123295E (cs)
RU (1) RU2256662C2 (cs)
TR (1) TR200101102T2 (cs)
TW (1) TWI227235B (cs)
WO (1) WO2000024744A1 (cs)

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US6759410B1 (en) 1999-11-23 2004-07-06 Smithline Beecham Corporation 3,4-dihydro-(1H)-quinazolin-2-ones and their use as CSBP/p38 kinase inhibitors
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Also Published As

Publication number Publication date
ATE277931T1 (de) 2004-10-15
NO318802B1 (no) 2005-05-09
MA27678A1 (fr) 2006-01-02
NZ510760A (en) 2003-08-29
CN1324360A (zh) 2001-11-28
JP2002528455A (ja) 2002-09-03
TWI227235B (en) 2005-02-01
WO2000024744A1 (en) 2000-05-04
ES2228123T3 (es) 2005-04-01
DE69920732T2 (de) 2006-02-23
CA2347474A1 (en) 2000-05-04
CN1150195C (zh) 2004-05-19
HUP0104199A3 (en) 2002-12-28
NO20011929L (no) 2001-04-19
BR9914677A (pt) 2001-07-17
ID28276A (id) 2001-05-10
EP1123295B1 (en) 2004-09-29
MY126478A (en) 2006-10-31
HRP20010274A2 (en) 2002-06-30
NO20011929D0 (no) 2001-04-19
HK1041483B (zh) 2004-12-24
TR200101102T2 (tr) 2002-01-21
PT1123295E (pt) 2005-01-31
EP1123295A1 (en) 2001-08-16
RU2256662C2 (ru) 2005-07-20
HK1041483A1 (en) 2002-07-12
DE69920732D1 (de) 2004-11-04
AU769989B2 (en) 2004-02-12
JP3593035B2 (ja) 2004-11-24
CA2347474C (en) 2008-08-26
US6150373A (en) 2000-11-21
HUP0104199A2 (hu) 2002-04-29
PL347432A1 (en) 2002-04-08
AU1036300A (en) 2000-05-15

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