CS262417B2 - Process for preparing new 1h,3h-pyrrolo/1,2-c/-thiazoles - Google Patents

Process for preparing new 1h,3h-pyrrolo/1,2-c/-thiazoles Download PDF

Info

Publication number: CS262417B2
Authority: CS; Czechoslovakia
Prior art keywords: pyridyl; solution; pyrrolo; total; reduced pressure
Prior art date: 1983-01-13

Application number

CS84197A

Other languages

Czech (cs)

English (en)

Other versions

CS19784A2 (en

Inventor

Jean-Louis Fabre

Daniel Farge

Claude James

Daniel Lave

Original Assignee

Rhone Poulenc Sante

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1983-01-13

Filing date

1984-01-10

Publication date

1989-03-14

1984-01-10 Application filed by Rhone Poulenc Sante filed Critical Rhone Poulenc Sante

1987-01-08 Priority to CS87172A priority Critical patent/CS262445B2/cs

1987-01-08 Priority to CS87171A priority patent/CS262444B2/cs

1988-08-16 Publication of CS19784A2 publication Critical patent/CS19784A2/cs

1989-03-14 Publication of CS262417B2 publication Critical patent/CS262417B2/cs

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pain & Pain Management (AREA)
Immunology (AREA)
Diabetes (AREA)
Hematology (AREA)
Pulmonology (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pyrrole Compounds (AREA)

CS84197A 1983-01-13 1984-01-10 Process for preparing new 1h,3h-pyrrolo/1,2-c/-thiazoles CS262417B2 (en)

Priority Applications (2)

Application Number	Priority Date	Filing Date	Title
CS87172A CS262445B2 (cs)	1984-01-10	1987-01-08	Způsob výroby nového lH,3H-pyrrolo[l,2-c]thiazolového derivátu
CS87171A CS262444B2 (cs)	1983-01-13	1987-01-08	Způsub výroby nového 1H,3H pyrrolo[l,2-c]thiazolového derivátu

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR8300453A FR2541280B1 (fr)	1983-01-13	1983-01-13	Nouveaux derives du 1h, 3h-pyrrolo (1,2c) thiazolecarboxamide-7, leur preparation et les medicaments qui les contiennent

Publications (2)

Publication Number	Publication Date
CS19784A2 CS19784A2 (en)	1988-08-16
CS262417B2 true CS262417B2 (en)	1989-03-14

Family

ID=9284898

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CS84197A CS262417B2 (en)	1983-01-13	1984-01-10	Process for preparing new 1h,3h-pyrrolo/1,2-c/-thiazoles

Country Status (28)

Country	Link
US (1)	US4529728A (ko)
EP (1)	EP0115979B1 (ko)
JP (2)	JPH0653748B2 (ko)
KR (1)	KR910001482B1 (ko)
AR (1)	AR240828A1 (ko)
AT (1)	ATE21248T1 (ko)
AU (1)	AU562795B2 (ko)
BG (2)	BG40145A3 (ko)
CA (1)	CA1229603A (ko)
CS (1)	CS262417B2 (ko)
DD (1)	DD218362A5 (ko)
DE (1)	DE3460401D1 (ko)
DK (1)	DK13984A (ko)
ES (2)	ES8407058A1 (ko)
FI (1)	FI76577C (ko)
FR (1)	FR2541280B1 (ko)
GR (1)	GR81679B (ko)
HU (1)	HU193277B (ko)
IE (1)	IE56839B1 (ko)
IL (1)	IL70664A (ko)
MA (1)	MA20001A1 (ko)
MX (5)	MX160610A (ko)
NO (1)	NO167031C (ko)
NZ (1)	NZ206807A (ko)
PL (2)	PL141846B1 (ko)
PT (1)	PT77952B (ko)
SU (3)	SU1245263A3 (ko)
ZA (2)	ZA84233B (ko)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2557111B1 (fr) *	1983-12-21	1986-04-11	Rhone Poulenc Sante	Nouveaux derives ortho-condenses du pyrrole, leur preparation et les medicaments qui les contiennent
FR2601016B1 (fr) *	1986-07-04	1988-10-07	Rhone Poulenc Sante	Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2601015B1 (fr) *	1986-07-04	1988-08-05	Rhone Poulenc Sante	Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent
CN1030415A (zh)	1987-02-20	1989-01-18	山之内制药株式会社	饱和的杂环碳酰胺衍生物和它的制备方法
FR2617484B1 (fr) *	1987-07-02	1989-10-20	Rhone Poulenc Sante	Procede de preparation de l'acide (pyridyl-3)-3 1h-3h-pyrrolo (1,2-c) thiazolecarboxylique-7 dextrogyre
FR2626004B1 (fr) *	1988-01-20	1991-08-02	Rhone Poulenc Sante	Procede de preparation du (pyridyl-3)-3 1h, 3h-pyrrolo (1,2-c) thiazolecarbonitrile-7
FR2644456B1 (fr) *	1989-03-17	1991-07-05	Rhone Poulenc Sante	Nouveaux derives du 1h, 3h-pyrrolo(1,2-c)thiazolecarboxamide-7, leur preparation et les compositions pharmaceutiques qui les contiennent
EP0479951A4 (en) *	1989-06-26	1992-12-09	The Research Foundation Of State University Of New York	Bis-acyloxymethyl derivatives
FR2678834A1 (fr) *	1991-07-09	1993-01-15	Rhone Poulenc Rorer Sa	Nouvelle application therapeutique du pyridylpyrrolothiazole carboxamide.
EP0595924B1 (en) *	1991-07-17	1999-04-14	Abbott Laboratories	Platelet activating factor antagonists
HU230518B1 (hu) *	2005-12-20	2016-10-28	Richter Gedeon Nyrt.	Bradykinin B1 receptor szelektív antagonista hatással rendelkező új fenatridin származékok, eljárás előállításukra, és az ezeket tartalmazó gyógyszerkészítmények

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3544590A (en) *	1967-04-28	1970-12-01	Exxon Research Engineering Co	Cyclic amines and the process for their formation
US3865839A (en) *	1973-03-01	1975-02-11	Hoechst Co American	Thiopyranopyrrolylsalicyclic acids and derivatives thereof

1983
- 1983-01-13 FR FR8300453A patent/FR2541280B1/fr not_active Expired
1984
- 1984-01-10 BG BG8465204A patent/BG40145A3/xx unknown
- 1984-01-10 CS CS84197A patent/CS262417B2/cs unknown
- 1984-01-10 BG BG8465203A patent/BG40144A3/xx unknown
- 1984-01-11 GR GR73491A patent/GR81679B/el unknown
- 1984-01-11 MA MA20222A patent/MA20001A1/fr unknown
- 1984-01-11 AU AU23202/84A patent/AU562795B2/en not_active Ceased
- 1984-01-11 ZA ZA84233A patent/ZA84233B/xx unknown
- 1984-01-11 DD DD84259351A patent/DD218362A5/de not_active IP Right Cessation
- 1984-01-11 ZA ZA84235A patent/ZA84235B/xx unknown
- 1984-01-11 IL IL70664A patent/IL70664A/xx unknown
- 1984-01-11 US US06/569,908 patent/US4529728A/en not_active Expired - Fee Related
- 1984-01-11 NZ NZ206807A patent/NZ206807A/en unknown
- 1984-01-12 CA CA000445146A patent/CA1229603A/fr not_active Expired
- 1984-01-12 IE IE64/84A patent/IE56839B1/en not_active IP Right Cessation
- 1984-01-12 DK DK13984A patent/DK13984A/da not_active Application Discontinuation
- 1984-01-12 HU HU8480A patent/HU193277B/hu unknown
- 1984-01-12 MX MX6146A patent/MX160610A/es unknown
- 1984-01-12 EP EP84400057A patent/EP0115979B1/fr not_active Expired
- 1984-01-12 PT PT77952A patent/PT77952B/pt not_active IP Right Cessation
- 1984-01-12 SU SU843692013A patent/SU1245263A3/ru active
- 1984-01-12 KR KR8400095A patent/KR910001482B1/ko not_active IP Right Cessation
- 1984-01-12 AT AT84400057T patent/ATE21248T1/de not_active IP Right Cessation
- 1984-01-12 DE DE8484400057T patent/DE3460401D1/de not_active Expired
- 1984-01-12 NO NO840106A patent/NO167031C/no unknown
- 1984-01-12 FI FI840106A patent/FI76577C/fi not_active IP Right Cessation
- 1984-01-13 JP JP59003686A patent/JPH0653748B2/ja not_active Expired - Lifetime
- 1984-01-13 JP JP59003687A patent/JPS59137490A/ja active Granted
- 1984-01-13 ES ES528873A patent/ES8407058A1/es not_active Expired
- 1984-01-13 PL PL1984245701A patent/PL141846B1/pl unknown
- 1984-01-13 PL PL1984251304A patent/PL140595B1/pl unknown
- 1984-01-13 AR AR295414A patent/AR240828A1/es active
- 1984-04-11 ES ES531518A patent/ES8502123A1/es not_active Expired
- 1984-10-17 SU SU843799806A patent/SU1284459A3/ru active
- 1984-10-17 SU SU843801005A patent/SU1266472A3/ru active
1988
- 1988-10-05 MX MX1329288A patent/MX13292A/es unknown
- 1988-10-05 MX MX1329188A patent/MX13291A/es unknown
- 1988-10-18 MX MX1346388A patent/MX13463A/es unknown
- 1988-10-18 MX MX1346288A patent/MX13462A/es unknown

Also Published As

Publication number	Publication date
JPH0653748B2 (ja)	1994-07-20
MX13291A (es)	1993-11-01
MX13463A (es)	1993-10-01
US4529728A (en)	1985-07-16
BG40144A3 (en)	1986-10-15
ES531518A0 (es)	1984-12-16
FI76577B (fi)	1988-07-29
SU1245263A3 (ru)	1986-07-15
SU1284459A3 (ru)	1987-01-15
EP0115979B1 (fr)	1986-08-06
FI840106A (fi)	1984-07-14
ATE21248T1 (de)	1986-08-15
PT77952B (fr)	1986-07-14
JPS59137490A (ja)	1984-08-07
PL140595B1 (en)	1987-05-30
GR81679B (ko)	1984-12-12
NO840106L (no)	1984-07-16
ES528873A0 (es)	1984-08-16
AU2320284A (en)	1984-07-19
NO167031C (no)	1991-09-25
PT77952A (fr)	1984-02-01
MX13292A (es)	1993-11-01
DK13984D0 (da)	1984-01-12
MX160610A (es)	1990-03-28
FR2541280A1 (fr)	1984-08-24
ZA84235B (en)	1984-09-26
AR240828A2 (es)	1991-02-28
NO167031B (no)	1991-06-17
BG40145A3 (en)	1986-10-15
PL251304A1 (en)	1985-09-24
KR840007419A (ko)	1984-12-07
PL141846B1 (en)	1987-08-31
HU193277B (en)	1987-09-28
DE3460401D1 (en)	1986-09-11
FI840106A0 (fi)	1984-01-12
MX13462A (es)	1993-08-01
CS19784A2 (en)	1988-08-16
NZ206807A (en)	1985-12-13
IE56839B1 (en)	1992-01-01
SU1266472A3 (ru)	1986-10-23
FR2541280B1 (fr)	1985-06-21
AR240828A1 (es)	1991-02-28
ZA84233B (en)	1984-09-26
MA20001A1 (fr)	1984-10-01
HUT34986A (en)	1985-05-28
JPS59134798A (ja)	1984-08-02
IL70664A (en)	1986-10-31
DK13984A (da)	1984-07-14
PL245701A1 (en)	1985-05-07
ES8502123A1 (es)	1984-12-16
AU562795B2 (en)	1987-06-18
IL70664A0 (en)	1984-04-30
IE840064L (en)	1984-07-13
JPH0547548B2 (ko)	1993-07-19
ES8407058A1 (es)	1984-08-16
CA1229603A (fr)	1987-11-24
EP0115979A1 (fr)	1984-08-15
DD218362A5 (de)	1985-02-06
FI76577C (fi)	1988-11-10
KR910001482B1 (ko)	1991-03-09

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