ATE21248T1 - Derivate von 1h,3h-pyrrolo(1,2-c)thiazol, ihre herstellung und sie enthaltende pharmazeutische zusammensetzungen. - Google Patents

Derivate von 1h,3h-pyrrolo(1,2-c)thiazol, ihre herstellung und sie enthaltende pharmazeutische zusammensetzungen.

Info

Publication number: ATE21248T1
Authority: AT; Austria
Prior art keywords: pyrrolo; thiazole; derivatives; preparation; pharmaceutical compositions
Prior art date: 1983-01-13

Application number

AT84400057T

Other languages

English (en)

Inventor

Jean-Louis Fabre

Daniel Farge

Claude James

Daniel Lave

Original Assignee

Rhone Poulenc Sante

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1983-01-13

Filing date

1984-01-12

Publication date

1986-08-15

1984-01-12 Application filed by Rhone Poulenc Sante filed Critical Rhone Poulenc Sante

1986-08-15 Application granted granted Critical

1986-08-15 Publication of ATE21248T1 publication Critical patent/ATE21248T1/de

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Immunology (AREA)
Pulmonology (AREA)
Diabetes (AREA)
Hematology (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pyrrole Compounds (AREA)

AT84400057T 1983-01-13 1984-01-12 Derivate von 1h,3h-pyrrolo(1,2-c)thiazol, ihre herstellung und sie enthaltende pharmazeutische zusammensetzungen. ATE21248T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR8300453A FR2541280B1 (fr)	1983-01-13	1983-01-13	Nouveaux derives du 1h, 3h-pyrrolo (1,2c) thiazolecarboxamide-7, leur preparation et les medicaments qui les contiennent
EP84400057A EP0115979B1 (de)	1983-01-13	1984-01-12	Derivate von 1H,3H-Pyrrolo(1,2-c)thiazol, ihre Herstellung und sie enthaltende pharmazeutische Zusammensetzungen

Publications (1)

Publication Number	Publication Date
ATE21248T1 true ATE21248T1 (de)	1986-08-15

Family

ID=9284898

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT84400057T ATE21248T1 (de)	1983-01-13	1984-01-12	Derivate von 1h,3h-pyrrolo(1,2-c)thiazol, ihre herstellung und sie enthaltende pharmazeutische zusammensetzungen.

Country Status (28)

Country	Link
US (1)	US4529728A (de)
EP (1)	EP0115979B1 (de)
JP (2)	JPS59137490A (de)
KR (1)	KR910001482B1 (de)
AR (1)	AR240828A1 (de)
AT (1)	ATE21248T1 (de)
AU (1)	AU562795B2 (de)
BG (2)	BG40144A3 (de)
CA (1)	CA1229603A (de)
CS (1)	CS262417B2 (de)
DD (1)	DD218362A5 (de)
DE (1)	DE3460401D1 (de)
DK (1)	DK13984A (de)
ES (2)	ES8407058A1 (de)
FI (1)	FI76577C (de)
FR (1)	FR2541280B1 (de)
GR (1)	GR81679B (de)
HU (1)	HU193277B (de)
IE (1)	IE56839B1 (de)
IL (1)	IL70664A (de)
MA (1)	MA20001A1 (de)
MX (5)	MX160610A (de)
NO (1)	NO167031C (de)
NZ (1)	NZ206807A (de)
PL (2)	PL140595B1 (de)
PT (1)	PT77952B (de)
SU (3)	SU1245263A3 (de)
ZA (2)	ZA84233B (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2557111B1 (fr) *	1983-12-21	1986-04-11	Rhone Poulenc Sante	Nouveaux derives ortho-condenses du pyrrole, leur preparation et les medicaments qui les contiennent
FR2601016B1 (fr) *	1986-07-04	1988-10-07	Rhone Poulenc Sante	Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2601015B1 (fr) *	1986-07-04	1988-08-05	Rhone Poulenc Sante	Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent
CN1030415A (zh) *	1987-02-20	1989-01-18	山之内制药株式会社	饱和的杂环碳酰胺衍生物和它的制备方法
FR2617484B1 (fr) *	1987-07-02	1989-10-20	Rhone Poulenc Sante	Procede de preparation de l'acide (pyridyl-3)-3 1h-3h-pyrrolo (1,2-c) thiazolecarboxylique-7 dextrogyre
FR2626004B1 (fr) *	1988-01-20	1991-08-02	Rhone Poulenc Sante	Procede de preparation du (pyridyl-3)-3 1h, 3h-pyrrolo (1,2-c) thiazolecarbonitrile-7
FR2644456B1 (fr) *	1989-03-17	1991-07-05	Rhone Poulenc Sante	Nouveaux derives du 1h, 3h-pyrrolo(1,2-c)thiazolecarboxamide-7, leur preparation et les compositions pharmaceutiques qui les contiennent
WO1991000093A1 (en) *	1989-06-26	1991-01-10	The Research Foundation Of State University Of New York	Bis-acyloxymethyl derivatives
FR2678834A1 (fr) *	1991-07-09	1993-01-15	Rhone Poulenc Rorer Sa	Nouvelle application therapeutique du pyridylpyrrolothiazole carboxamide.
US5459152A (en) *	1991-07-17	1995-10-17	Abbott Laboratories	Platelet activating factor antagonists
HU230518B1 (hu) *	2005-12-20	2016-10-28	Richter Gedeon Nyrt.	Bradykinin B1 receptor szelektív antagonista hatással rendelkező új fenatridin származékok, eljárás előállításukra, és az ezeket tartalmazó gyógyszerkészítmények

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3544590A (en) *	1967-04-28	1970-12-01	Exxon Research Engineering Co	Cyclic amines and the process for their formation
US3865839A (en) *	1973-03-01	1975-02-11	Hoechst Co American	Thiopyranopyrrolylsalicyclic acids and derivatives thereof

1983
- 1983-01-13 FR FR8300453A patent/FR2541280B1/fr not_active Expired
1984
- 1984-01-10 CS CS84197A patent/CS262417B2/cs unknown
- 1984-01-10 BG BG8465203A patent/BG40144A3/xx unknown
- 1984-01-10 BG BG8465204A patent/BG40145A3/xx unknown
- 1984-01-11 IL IL70664A patent/IL70664A/xx unknown
- 1984-01-11 GR GR73491A patent/GR81679B/el unknown
- 1984-01-11 MA MA20222A patent/MA20001A1/fr unknown
- 1984-01-11 ZA ZA84233A patent/ZA84233B/xx unknown
- 1984-01-11 DD DD84259351A patent/DD218362A5/de not_active IP Right Cessation
- 1984-01-11 NZ NZ206807A patent/NZ206807A/en unknown
- 1984-01-11 AU AU23202/84A patent/AU562795B2/en not_active Ceased
- 1984-01-11 US US06/569,908 patent/US4529728A/en not_active Expired - Fee Related
- 1984-01-11 ZA ZA84235A patent/ZA84235B/xx unknown
- 1984-01-12 PT PT77952A patent/PT77952B/pt not_active IP Right Cessation
- 1984-01-12 EP EP84400057A patent/EP0115979B1/de not_active Expired
- 1984-01-12 DE DE8484400057T patent/DE3460401D1/de not_active Expired
- 1984-01-12 AT AT84400057T patent/ATE21248T1/de not_active IP Right Cessation
- 1984-01-12 IE IE64/84A patent/IE56839B1/en not_active IP Right Cessation
- 1984-01-12 DK DK13984A patent/DK13984A/da not_active Application Discontinuation
- 1984-01-12 NO NO840106A patent/NO167031C/no unknown
- 1984-01-12 HU HU8480A patent/HU193277B/hu unknown
- 1984-01-12 KR KR8400095A patent/KR910001482B1/ko not_active IP Right Cessation
- 1984-01-12 MX MX6146A patent/MX160610A/es unknown
- 1984-01-12 SU SU843692013A patent/SU1245263A3/ru active
- 1984-01-12 CA CA000445146A patent/CA1229603A/fr not_active Expired
- 1984-01-12 FI FI840106A patent/FI76577C/fi not_active IP Right Cessation
- 1984-01-13 JP JP59003687A patent/JPS59137490A/ja active Granted
- 1984-01-13 JP JP59003686A patent/JPH0653748B2/ja not_active Expired - Lifetime
- 1984-01-13 ES ES528873A patent/ES8407058A1/es not_active Expired
- 1984-01-13 PL PL1984251304A patent/PL140595B1/pl unknown
- 1984-01-13 PL PL1984245701A patent/PL141846B1/pl unknown
- 1984-01-13 AR AR295414A patent/AR240828A1/es active
- 1984-04-11 ES ES531518A patent/ES531518A0/es active Granted
- 1984-10-17 SU SU843801005A patent/SU1266472A3/ru active
- 1984-10-17 SU SU843799806A patent/SU1284459A3/ru active
1988
- 1988-10-05 MX MX1329288A patent/MX13292A/es unknown
- 1988-10-05 MX MX1329188A patent/MX13291A/es unknown
- 1988-10-18 MX MX1346388A patent/MX13463A/es unknown
- 1988-10-18 MX MX1346288A patent/MX13462A/es unknown

Also Published As

Publication number	Publication date
PL140595B1 (en)	1987-05-30
FI840106A (fi)	1984-07-14
FI840106A0 (fi)	1984-01-12
AR240828A2 (es)	1991-02-28
EP0115979A1 (de)	1984-08-15
JPS59137490A (ja)	1984-08-07
SU1245263A3 (ru)	1986-07-15
MX160610A (es)	1990-03-28
AR240828A1 (es)	1991-02-28
NZ206807A (en)	1985-12-13
SU1284459A3 (ru)	1987-01-15
PL141846B1 (en)	1987-08-31
GR81679B (de)	1984-12-12
PT77952A (fr)	1984-02-01
KR910001482B1 (ko)	1991-03-09
DK13984D0 (da)	1984-01-12
EP0115979B1 (de)	1986-08-06
KR840007419A (ko)	1984-12-07
IL70664A0 (en)	1984-04-30
ZA84235B (en)	1984-09-26
JPH0547548B2 (de)	1993-07-19
IL70664A (en)	1986-10-31
DE3460401D1 (en)	1986-09-11
IE56839B1 (en)	1992-01-01
MX13292A (es)	1993-11-01
AU2320284A (en)	1984-07-19
FI76577B (fi)	1988-07-29
HUT34986A (en)	1985-05-28
IE840064L (en)	1984-07-13
FR2541280A1 (fr)	1984-08-24
PL245701A1 (en)	1985-05-07
US4529728A (en)	1985-07-16
ZA84233B (en)	1984-09-26
BG40144A3 (en)	1986-10-15
SU1266472A3 (ru)	1986-10-23
FI76577C (fi)	1988-11-10
PT77952B (fr)	1986-07-14
ES8502123A1 (es)	1984-12-16
MA20001A1 (fr)	1984-10-01
JPS59134798A (ja)	1984-08-02
MX13462A (es)	1993-08-01
ES528873A0 (es)	1984-08-16
ES531518A0 (es)	1984-12-16
AU562795B2 (en)	1987-06-18
ES8407058A1 (es)	1984-08-16
DK13984A (da)	1984-07-14
DD218362A5 (de)	1985-02-06
MX13291A (es)	1993-11-01
MX13463A (es)	1993-10-01
CS19784A2 (en)	1988-08-16
CA1229603A (fr)	1987-11-24
NO167031B (no)	1991-06-17
BG40145A3 (en)	1986-10-15
NO167031C (no)	1991-09-25
HU193277B (en)	1987-09-28
PL251304A1 (en)	1985-09-24
NO840106L (no)	1984-07-16
CS262417B2 (en)	1989-03-14
JPH0653748B2 (ja)	1994-07-20
FR2541280B1 (fr)	1985-06-21

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Legal Events

Date	Code	Title	Description
1986-11-15	UEP	Publication of translation of european patent specification
1997-10-15	REN	Ceased due to non-payment of the annual fee