CR11860A - Derivados de dibenzotiazepina y sus usos - 424 - Google Patents

Derivados de dibenzotiazepina y sus usos - 424

Info

Publication number
CR11860A
CR11860A CR11860A CR11860A CR11860A CR 11860 A CR11860 A CR 11860A CR 11860 A CR11860 A CR 11860A CR 11860 A CR11860 A CR 11860A CR 11860 A CR11860 A CR 11860A
Authority
CR
Costa Rica
Prior art keywords
dibenzotiazepina
derivatives
compositions
compounds
formula
Prior art date
Application number
CR11860A
Other languages
English (en)
Inventor
Brown Dean
R Damewood James
Edwards Phil
Hulsizer James
Campbell Muir James
Edward Pierson M Jr
Bhikkappa Shenvi Askokkumar
Wesolowski Steven
Widzowski Dan
Wood Michael
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41431860&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR11860(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of CR11860A publication Critical patent/CR11860A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • C07D281/16—[b, f]-condensed

Abstract

Los compuestos de la fórmula I, donde Z se describe en la descripción, sales farmacéuticamente aceptables de estos, composiciones que los comprenden y métodos para tratar el transtorno bipolar.
CR11860A 2008-06-20 2010-12-20 Derivados de dibenzotiazepina y sus usos - 424 CR11860A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US7441708P 2008-06-20 2008-06-20

Publications (1)

Publication Number Publication Date
CR11860A true CR11860A (es) 2011-02-25

Family

ID=41431860

Family Applications (1)

Application Number Title Priority Date Filing Date
CR11860A CR11860A (es) 2008-06-20 2010-12-20 Derivados de dibenzotiazepina y sus usos - 424

Country Status (38)

Country Link
US (3) US20110160184A1 (es)
EP (1) EP2307389B1 (es)
JP (2) JP5468068B2 (es)
KR (1) KR20110019781A (es)
CN (1) CN102131791B (es)
AR (1) AR072200A1 (es)
AU (1) AU2009260905B2 (es)
BR (1) BRPI0914231A2 (es)
CA (1) CA2728675A1 (es)
CL (1) CL2010001471A1 (es)
CR (1) CR11860A (es)
CU (1) CU23884B1 (es)
CY (1) CY1113845T1 (es)
DK (1) DK2307389T3 (es)
DO (1) DOP2010000393A (es)
EA (1) EA201001889A1 (es)
EC (1) ECSP10010698A (es)
ES (1) ES2402084T3 (es)
HK (1) HK1156308A1 (es)
HN (1) HN2010002683A (es)
HR (1) HRP20130234T1 (es)
IL (2) IL210081A (es)
ME (1) ME01516B (es)
MX (1) MX2010014203A (es)
MY (1) MY157518A (es)
NI (1) NI201000224A (es)
NZ (1) NZ590616A (es)
PE (1) PE20110029A1 (es)
PL (1) PL2307389T3 (es)
PT (1) PT2307389E (es)
RS (1) RS52703B (es)
SI (1) SI2307389T1 (es)
SV (1) SV2010003769A (es)
TW (1) TWI488854B (es)
UA (1) UA105903C2 (es)
UY (1) UY31919A (es)
WO (1) WO2009154563A1 (es)
ZA (1) ZA201100488B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA201001889A1 (ru) * 2008-06-20 2011-08-30 Астразенека Аб Производные дибензотиазепина и их применение
CN105981027A (zh) * 2013-08-12 2016-09-28 哥莱菲特软件公司 安全认证并切换至加密域
CN103524455A (zh) * 2013-10-30 2014-01-22 苏州敬业医药化工有限公司 一种制备2-氯-二苯并[b,f][1,4]硫氮杂卓-11-[10H]酮的方法
CN106134230A (zh) 2013-11-21 2016-11-16 哥莱菲特软件公司 用于移动信息设备上的远程内容和配置控制的管理域
CN104447615A (zh) * 2014-02-28 2015-03-25 广东东阳光药业有限公司 喹硫平中间体的制备方法

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Also Published As

Publication number Publication date
ES2402084T3 (es) 2013-04-26
US8158618B2 (en) 2012-04-17
IL210081A0 (en) 2011-02-28
AU2009260905B2 (en) 2012-08-23
US20090318415A1 (en) 2009-12-24
SV2010003769A (es) 2011-05-20
JP2011524898A (ja) 2011-09-08
CN102131791A (zh) 2011-07-20
US8653257B2 (en) 2014-02-18
SI2307389T1 (sl) 2013-04-30
HK1156308A1 (en) 2012-06-08
CU23884B1 (es) 2013-04-19
DK2307389T3 (da) 2013-04-02
CN102131791B (zh) 2014-12-24
NZ590616A (en) 2012-09-28
EP2307389A4 (en) 2012-04-11
KR20110019781A (ko) 2011-02-28
PT2307389E (pt) 2013-03-28
IL229560A0 (en) 2014-01-30
TW201002702A (en) 2010-01-16
EP2307389A1 (en) 2011-04-13
DOP2010000393A (es) 2011-01-31
IL229560A (en) 2015-07-30
WO2009154563A1 (en) 2009-12-23
IL210081A (en) 2013-12-31
TWI488854B (zh) 2015-06-21
JP5468068B2 (ja) 2014-04-09
PE20110029A1 (es) 2011-02-11
CL2010001471A1 (es) 2011-05-06
US20110160184A1 (en) 2011-06-30
ME01516B (me) 2014-04-20
ECSP10010698A (es) 2011-01-31
AR072200A1 (es) 2010-08-11
UA105903C2 (uk) 2014-07-10
US20120202991A1 (en) 2012-08-09
HN2010002683A (es) 2013-01-15
EA201001889A1 (ru) 2011-08-30
CU20100252A7 (es) 2011-11-15
BRPI0914231A2 (pt) 2015-11-03
MY157518A (en) 2016-06-15
CY1113845T1 (el) 2016-07-27
NI201000224A (es) 2012-03-19
CA2728675A1 (en) 2009-12-23
UY31919A (es) 2010-01-29
HRP20130234T1 (hr) 2013-04-30
ZA201100488B (en) 2011-10-26
EP2307389B1 (en) 2013-01-23
JP2014098006A (ja) 2014-05-29
PL2307389T3 (pl) 2013-05-31
RS52703B (en) 2013-08-30
MX2010014203A (es) 2011-02-22
AU2009260905A1 (en) 2009-12-23

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