AR072200A1 - Derivados dibenzotiazepina y usos de los mismos - Google Patents

Derivados dibenzotiazepina y usos de los mismos

Info

Publication number
AR072200A1
AR072200A1 ARP090102240A ARP090102240A AR072200A1 AR 072200 A1 AR072200 A1 AR 072200A1 AR P090102240 A ARP090102240 A AR P090102240A AR P090102240 A ARP090102240 A AR P090102240A AR 072200 A1 AR072200 A1 AR 072200A1
Authority
AR
Argentina
Prior art keywords
disorder
dibenzotiazepine
derivatives
same
schizophrenia
Prior art date
Application number
ARP090102240A
Other languages
English (en)
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41431860&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR072200(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of AR072200A1 publication Critical patent/AR072200A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • C07D281/16—[b, f]-condensed

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Steroid Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Composiciones que los comprenden, y metodos para el tratamiento de un trastorno bipolar, un trastorno de ansiedad, un trastorno del talante o esquizofrenia u otro trastorno psicotico, con dichos compuestos. Reivindicacion 1: Un compuesto de formula 1o una sal farmaceuticamente aceptable del mismo, donde Z es H, C(=O)-R1, C(=O)OR1 o C(R1)-NHC(=O)R2, donde R1 y R2 son cada uno independientemente cada vez que aparecen alquilo, cicloalquilo, arilo, heteroarilo o heterocicloalquilo.
ARP090102240A 2008-06-20 2009-06-19 Derivados dibenzotiazepina y usos de los mismos AR072200A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US7441708P 2008-06-20 2008-06-20

Publications (1)

Publication Number Publication Date
AR072200A1 true AR072200A1 (es) 2010-08-11

Family

ID=41431860

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP090102240A AR072200A1 (es) 2008-06-20 2009-06-19 Derivados dibenzotiazepina y usos de los mismos

Country Status (38)

Country Link
US (3) US20110160184A1 (es)
EP (1) EP2307389B1 (es)
JP (2) JP5468068B2 (es)
KR (1) KR20110019781A (es)
CN (1) CN102131791B (es)
AR (1) AR072200A1 (es)
AU (1) AU2009260905B2 (es)
BR (1) BRPI0914231A2 (es)
CA (1) CA2728675A1 (es)
CL (1) CL2010001471A1 (es)
CR (1) CR11860A (es)
CU (1) CU23884B1 (es)
CY (1) CY1113845T1 (es)
DK (1) DK2307389T3 (es)
DO (1) DOP2010000393A (es)
EA (1) EA201001889A1 (es)
EC (1) ECSP10010698A (es)
ES (1) ES2402084T3 (es)
HK (1) HK1156308A1 (es)
HN (1) HN2010002683A (es)
HR (1) HRP20130234T1 (es)
IL (2) IL210081A (es)
ME (1) ME01516B (es)
MX (1) MX2010014203A (es)
MY (1) MY157518A (es)
NI (1) NI201000224A (es)
NZ (1) NZ590616A (es)
PE (1) PE20110029A1 (es)
PL (1) PL2307389T3 (es)
PT (1) PT2307389E (es)
RS (1) RS52703B (es)
SI (1) SI2307389T1 (es)
SV (1) SV2010003769A (es)
TW (1) TWI488854B (es)
UA (1) UA105903C2 (es)
UY (1) UY31919A (es)
WO (1) WO2009154563A1 (es)
ZA (1) ZA201100488B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ590616A (en) * 2008-06-20 2012-09-28 Astrazeneca Ab Dibenzothiazepine derivatives and use thereof
KR102096550B1 (ko) * 2013-08-12 2020-04-02 씨아이에스 맥스웰, 엘엘씨 운영 시스템 통합 도메인 관리
CN103524455A (zh) * 2013-10-30 2014-01-22 苏州敬业医药化工有限公司 一种制备2-氯-二苯并[b,f][1,4]硫氮杂卓-11-[10H]酮的方法
EP3072320A4 (en) 2013-11-21 2017-05-24 Graphite Software Corporation Managed domains for remote content and configuration control on mobile information devices
CN104447615A (zh) * 2014-02-28 2015-03-25 广东东阳光药业有限公司 喹硫平中间体的制备方法

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Also Published As

Publication number Publication date
BRPI0914231A2 (pt) 2015-11-03
CU23884B1 (es) 2013-04-19
JP2011524898A (ja) 2011-09-08
PT2307389E (pt) 2013-03-28
MX2010014203A (es) 2011-02-22
MY157518A (en) 2016-06-15
EA201001889A1 (ru) 2011-08-30
NI201000224A (es) 2012-03-19
HN2010002683A (es) 2013-01-15
ZA201100488B (en) 2011-10-26
JP2014098006A (ja) 2014-05-29
IL229560A0 (en) 2014-01-30
EP2307389B1 (en) 2013-01-23
SV2010003769A (es) 2011-05-20
DOP2010000393A (es) 2011-01-31
AU2009260905A1 (en) 2009-12-23
WO2009154563A1 (en) 2009-12-23
KR20110019781A (ko) 2011-02-28
HK1156308A1 (en) 2012-06-08
ES2402084T3 (es) 2013-04-26
TWI488854B (zh) 2015-06-21
HRP20130234T1 (hr) 2013-04-30
CL2010001471A1 (es) 2011-05-06
CN102131791A (zh) 2011-07-20
JP5468068B2 (ja) 2014-04-09
CR11860A (es) 2011-02-25
PL2307389T3 (pl) 2013-05-31
US8653257B2 (en) 2014-02-18
IL210081A0 (en) 2011-02-28
US20090318415A1 (en) 2009-12-24
SI2307389T1 (sl) 2013-04-30
US8158618B2 (en) 2012-04-17
EP2307389A4 (en) 2012-04-11
CA2728675A1 (en) 2009-12-23
ECSP10010698A (es) 2011-01-31
PE20110029A1 (es) 2011-02-11
AU2009260905B2 (en) 2012-08-23
DK2307389T3 (da) 2013-04-02
NZ590616A (en) 2012-09-28
IL210081A (en) 2013-12-31
CY1113845T1 (el) 2016-07-27
ME01516B (me) 2014-04-20
CU20100252A7 (es) 2011-11-15
RS52703B (en) 2013-08-30
UA105903C2 (uk) 2014-07-10
US20120202991A1 (en) 2012-08-09
EP2307389A1 (en) 2011-04-13
CN102131791B (zh) 2014-12-24
US20110160184A1 (en) 2011-06-30
UY31919A (es) 2010-01-29
TW201002702A (en) 2010-01-16
IL229560A (en) 2015-07-30

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