CO6821937A2 - Nuevos inhibidores de cinasa de proteína de indolinona - Google Patents

Nuevos inhibidores de cinasa de proteína de indolinona

Info

Publication number
CO6821937A2
CO6821937A2 CO13236301A CO13236301A CO6821937A2 CO 6821937 A2 CO6821937 A2 CO 6821937A2 CO 13236301 A CO13236301 A CO 13236301A CO 13236301 A CO13236301 A CO 13236301A CO 6821937 A2 CO6821937 A2 CO 6821937A2
Authority
CO
Colombia
Prior art keywords
protein kinase
kinase inhibitors
new
indolinone protein
new indolinone
Prior art date
Application number
CO13236301A
Other languages
English (en)
Inventor
Do Zhang
Guojian Xie
Original Assignee
Beta Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beta Pharma Inc filed Critical Beta Pharma Inc
Publication of CO6821937A2 publication Critical patent/CO6821937A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
CO13236301A 2011-04-08 2013-10-04 Nuevos inhibidores de cinasa de proteína de indolinona CO6821937A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201161473724P 2011-04-08 2011-04-08

Publications (1)

Publication Number Publication Date
CO6821937A2 true CO6821937A2 (es) 2013-12-31

Family

ID=46966568

Family Applications (1)

Application Number Title Priority Date Filing Date
CO13236301A CO6821937A2 (es) 2011-04-08 2013-10-04 Nuevos inhibidores de cinasa de proteína de indolinona

Country Status (13)

Country Link
US (1) US9163010B2 (es)
EP (1) EP2694058B1 (es)
JP (1) JP5797324B2 (es)
KR (1) KR20140027972A (es)
CN (1) CN103945696B (es)
AU (1) AU2012240018A1 (es)
BR (1) BR112013025679A2 (es)
CA (1) CA2831474A1 (es)
CO (1) CO6821937A2 (es)
IL (1) IL228726A0 (es)
MX (1) MX2013011481A (es)
SG (1) SG193527A1 (es)
WO (1) WO2012139019A2 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102499917B (zh) 2011-10-25 2014-12-17 澳门大学 吲哚酮类化合物在制备神经保护药物中的应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ520640A (en) * 2000-02-15 2005-04-29 Upjohn Co Pyrrole substituted 2-indolinone protein kinase inhibitors
AR042586A1 (es) * 2001-02-15 2005-06-29 Sugen Inc 3-(4-amidopirrol-2-ilmetiliden)-2-indolinona como inhibidores de la protein quinasa; sus composiciones farmaceuticas; un metodo para la modulacion de la actividad catalitica de la proteinquinasa; un metodo para tratar o prevenir una afeccion relacionada con la proteinquinasa
WO2003031438A1 (en) * 2001-10-10 2003-04-17 Sugen, Inc. 3-[4-(substituted heterocyclyl)-pyrrol-2-ylmethylidene]-2-indolinone derivatives as kinase inhibitors
US7119209B2 (en) 2002-02-15 2006-10-10 Pharmacia & Upjohn Company Process for preparing indolinone derivatives
WO2009030270A1 (en) * 2007-09-03 2009-03-12 Novartis Ag Dihydroindole derivatives useful in parkinson's disease

Also Published As

Publication number Publication date
WO2012139019A2 (en) 2012-10-11
BR112013025679A2 (pt) 2016-07-19
CA2831474A1 (en) 2012-10-11
CN103945696B (zh) 2016-06-29
KR20140027972A (ko) 2014-03-07
JP5797324B2 (ja) 2015-10-21
SG193527A1 (en) 2013-10-30
US9163010B2 (en) 2015-10-20
MX2013011481A (es) 2014-02-17
EP2694058A2 (en) 2014-02-12
EP2694058B1 (en) 2015-11-04
AU2012240018A1 (en) 2013-10-10
CN103945696A (zh) 2014-07-23
US20120258995A1 (en) 2012-10-11
EP2694058A4 (en) 2014-08-20
JP2014515745A (ja) 2014-07-03
IL228726A0 (en) 2013-12-31
WO2012139019A3 (en) 2014-05-01

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