CN105801559A - 4-甲基-3-[[4-(3-吡啶基)-2-嘧啶基]氨基]苯甲酸乙酯的制备方法 - Google Patents
4-甲基-3-[[4-(3-吡啶基)-2-嘧啶基]氨基]苯甲酸乙酯的制备方法 Download PDFInfo
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- CN105801559A CN105801559A CN201610279915.XA CN201610279915A CN105801559A CN 105801559 A CN105801559 A CN 105801559A CN 201610279915 A CN201610279915 A CN 201610279915A CN 105801559 A CN105801559 A CN 105801559A
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- methyl
- pyridine radicals
- amino
- radicals
- pyrimidine
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyridine Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Description
Claims (10)
Priority Applications (1)
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CN201610279915.XA CN105801559B (zh) | 2016-04-28 | 2016-04-28 | 4-甲基-3-[[4-(3-吡啶基)-2-嘧啶基]氨基]苯甲酸乙酯的制备方法 |
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CN201610279915.XA CN105801559B (zh) | 2016-04-28 | 2016-04-28 | 4-甲基-3-[[4-(3-吡啶基)-2-嘧啶基]氨基]苯甲酸乙酯的制备方法 |
Publications (2)
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CN105801559A true CN105801559A (zh) | 2016-07-27 |
CN105801559B CN105801559B (zh) | 2019-03-01 |
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CN201610279915.XA Active CN105801559B (zh) | 2016-04-28 | 2016-04-28 | 4-甲基-3-[[4-(3-吡啶基)-2-嘧啶基]氨基]苯甲酸乙酯的制备方法 |
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Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2021074138A1 (en) * | 2019-10-14 | 2021-04-22 | Esco Aster Pte. Ltd. | Synthesis of 6-methyl-n1-(4-(pyridin-3-yl)pyrimidin-2-yl)benzene-1,3-diamine |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1675195A (zh) * | 2002-07-05 | 2005-09-28 | 诺瓦提斯公司 | 酪氨酸激酶抑制剂 |
US20060149061A1 (en) * | 2004-12-30 | 2006-07-06 | Huang Anli | Novel process for preparing Imatinib |
WO2008103068A2 (ru) * | 2007-02-20 | 2008-08-28 | Yury Iosifovich Kopyrin | Способ получения 2-aнилинoпиpимидинoв или их солей |
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2016
- 2016-04-28 CN CN201610279915.XA patent/CN105801559B/zh active Active
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1675195A (zh) * | 2002-07-05 | 2005-09-28 | 诺瓦提斯公司 | 酪氨酸激酶抑制剂 |
US20060149061A1 (en) * | 2004-12-30 | 2006-07-06 | Huang Anli | Novel process for preparing Imatinib |
WO2008103068A2 (ru) * | 2007-02-20 | 2008-08-28 | Yury Iosifovich Kopyrin | Способ получения 2-aнилинoпиpимидинoв или их солей |
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2021074138A1 (en) * | 2019-10-14 | 2021-04-22 | Esco Aster Pte. Ltd. | Synthesis of 6-methyl-n1-(4-(pyridin-3-yl)pyrimidin-2-yl)benzene-1,3-diamine |
CN114585615A (zh) * | 2019-10-14 | 2022-06-03 | 新加坡艺思高艾斯特生物科技有限公司 | 6-甲基-n1-(4-(吡啶-3-基)嘧啶-2-基)苯-1,3-二胺的合成 |
TWI832015B (zh) * | 2019-10-14 | 2024-02-11 | 新加坡商藝思高艾斯特私人有限公司 | 酪胺酸激酶抑制物之合成 |
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CB03 | Change of inventor or designer information | ||
CB03 | Change of inventor or designer information |
Inventor after: Qiao Renzhong Inventor after: Zhang Huizheng Inventor after: Li Huina Inventor after: Zhang Jin Inventor after: Li Chao Inventor before: Qiao Renzhong Inventor before: Li Huina Inventor before: Zhang Jin Inventor before: Li Chao |
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Effective date of registration: 20230615 Address after: No. 17, Linghe Road, Lingshan Town, Jimo District, Qingdao, Shandong 266219 Patentee after: Shandong Dayi Jingcheng Pharmaceutical Co.,Ltd. Address before: 100029, No. 15 East Third Ring Road, Chaoyang District, Beijing Patentee before: BEIJING University OF CHEMICAL TECHNOLOGY |