CL2008000690A1 - Compuestos derivados del acido indol-3-propionico; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como hiperlipidemia, hipertension; entre otras. - Google Patents
Compuestos derivados del acido indol-3-propionico; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como hiperlipidemia, hipertension; entre otras.Info
- Publication number
- CL2008000690A1 CL2008000690A1 CL200800690A CL2008000690A CL2008000690A1 CL 2008000690 A1 CL2008000690 A1 CL 2008000690A1 CL 200800690 A CL200800690 A CL 200800690A CL 2008000690 A CL2008000690 A CL 2008000690A CL 2008000690 A1 CL2008000690 A1 CL 2008000690A1
- Authority
- CL
- Chile
- Prior art keywords
- hyperlipidemia
- indol
- hypertension
- diseases
- treatment
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/405—Indole-alkanecarboxylic acids; Derivatives thereof, e.g. tryptophan, indomethacin
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- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
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- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/32—Oxygen atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Neurology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Neurosurgery (AREA)
- Hematology (AREA)
- Biomedical Technology (AREA)
- Obesity (AREA)
- Urology & Nephrology (AREA)
- Dermatology (AREA)
- Virology (AREA)
- Immunology (AREA)
- Endocrinology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Ophthalmology & Optometry (AREA)
- Emergency Medicine (AREA)
- Molecular Biology (AREA)
- Reproductive Health (AREA)
- Hospice & Palliative Care (AREA)
- Rheumatology (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US89387107P | 2007-03-08 | 2007-03-08 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2008000690A1 true CL2008000690A1 (es) | 2008-09-12 |
Family
ID=39590187
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL200800690A CL2008000690A1 (es) | 2007-03-08 | 2008-03-07 | Compuestos derivados del acido indol-3-propionico; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como hiperlipidemia, hipertension; entre otras. |
Country Status (16)
Country | Link |
---|---|
US (2) | US8053463B2 (es) |
EP (1) | EP2114879A1 (es) |
JP (1) | JP2010520877A (es) |
KR (1) | KR20090118055A (es) |
CN (1) | CN101679250A (es) |
AR (1) | AR065633A1 (es) |
AU (1) | AU2008222810A1 (es) |
BR (1) | BRPI0808440A2 (es) |
CA (1) | CA2679411A1 (es) |
CL (1) | CL2008000690A1 (es) |
IL (1) | IL200548A0 (es) |
MX (1) | MX2009009292A (es) |
PE (1) | PE20090159A1 (es) |
RU (1) | RU2009137124A (es) |
TW (1) | TW200845980A (es) |
WO (1) | WO2008109700A1 (es) |
Families Citing this family (42)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2008063888A2 (en) | 2006-11-22 | 2008-05-29 | Plexxikon, Inc. | Compounds modulating c-fms and/or c-kit activity and uses therefor |
US20100190777A1 (en) | 2007-07-17 | 2010-07-29 | Plexxikon Inc. | Compounds and methods for kinase modulation, and indications therefor |
WO2009143018A2 (en) | 2008-05-19 | 2009-11-26 | Plexxikon, Inc. | Compounds and methods for kinase modulation, and indications therefor |
WO2011063159A1 (en) | 2009-11-18 | 2011-05-26 | Plexxikon, Inc. | Compounds and methods for kinase modulation, and indications therefor |
JP5815558B2 (ja) | 2009-12-23 | 2015-11-17 | プレキシコン インコーポレーテッドPlexxikon Inc. | キナーゼ調節のための化合物及び方法ならびにそれらの適応症 |
WO2011107494A1 (de) | 2010-03-03 | 2011-09-09 | Sanofi | Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
TWI619713B (zh) | 2010-04-21 | 2018-04-01 | 普雷辛肯公司 | 用於激酶調節的化合物和方法及其適應症 |
US8933024B2 (en) | 2010-06-18 | 2015-01-13 | Sanofi | Azolopyridin-3-one derivatives as inhibitors of lipases and phospholipases |
US8530413B2 (en) | 2010-06-21 | 2013-09-10 | Sanofi | Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments |
TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
AU2012214762B2 (en) | 2011-02-07 | 2015-08-13 | Plexxikon Inc. | Compounds and methods for kinase modulation, and indications therefor |
JP6113151B2 (ja) | 2011-05-17 | 2017-04-12 | プレキシコン インコーポレーテッドPlexxikon Inc. | キナーゼ調節およびその適応症 |
WO2013037390A1 (en) | 2011-09-12 | 2013-03-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
WO2013045413A1 (en) | 2011-09-27 | 2013-04-04 | Sanofi | 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
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- 2008-03-05 KR KR1020097018693A patent/KR20090118055A/ko not_active Application Discontinuation
- 2008-03-05 MX MX2009009292A patent/MX2009009292A/es not_active Application Discontinuation
- 2008-03-05 EP EP08731467A patent/EP2114879A1/en not_active Withdrawn
- 2008-03-05 US US12/043,069 patent/US8053463B2/en active Active
- 2008-03-05 CN CN200880013794A patent/CN101679250A/zh active Pending
- 2008-03-05 RU RU2009137124/04A patent/RU2009137124A/ru not_active Application Discontinuation
- 2008-03-05 BR BRPI0808440-8A patent/BRPI0808440A2/pt not_active IP Right Cessation
- 2008-03-05 AU AU2008222810A patent/AU2008222810A1/en not_active Abandoned
- 2008-03-05 JP JP2009552869A patent/JP2010520877A/ja active Pending
- 2008-03-05 WO PCT/US2008/055955 patent/WO2008109700A1/en active Application Filing
- 2008-03-05 CA CA002679411A patent/CA2679411A1/en not_active Abandoned
- 2008-03-07 TW TW097108189A patent/TW200845980A/zh unknown
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2009
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2011
- 2011-09-23 US US13/243,703 patent/US20120015966A1/en not_active Abandoned
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AU2008222810A1 (en) | 2008-09-12 |
CN101679250A (zh) | 2010-03-24 |
EP2114879A1 (en) | 2009-11-11 |
RU2009137124A (ru) | 2011-04-20 |
IL200548A0 (en) | 2010-05-17 |
PE20090159A1 (es) | 2009-02-21 |
BRPI0808440A2 (pt) | 2014-07-29 |
AR065633A1 (es) | 2009-06-17 |
TW200845980A (en) | 2008-12-01 |
JP2010520877A (ja) | 2010-06-17 |
US20080255201A1 (en) | 2008-10-16 |
CA2679411A1 (en) | 2008-09-12 |
WO2008109700A1 (en) | 2008-09-12 |
US20120015966A1 (en) | 2012-01-19 |
KR20090118055A (ko) | 2009-11-17 |
US8053463B2 (en) | 2011-11-08 |
MX2009009292A (es) | 2009-09-10 |
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