BRPI0906937A2 - composto, composição farmacêutica, e, uso de um composto - Google Patents
composto, composição farmacêutica, e, uso de um compostoInfo
- Publication number
- BRPI0906937A2 BRPI0906937A2 BRPI0906937A BRPI0906937A BRPI0906937A2 BR PI0906937 A2 BRPI0906937 A2 BR PI0906937A2 BR PI0906937 A BRPI0906937 A BR PI0906937A BR PI0906937 A BRPI0906937 A BR PI0906937A BR PI0906937 A2 BRPI0906937 A2 BR PI0906937A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- pharmaceutical composition
- pharmaceutical
- composition
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/18—Bridged systems
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP08151199 | 2008-02-08 | ||
PCT/EP2009/051366 WO2009098283A1 (en) | 2008-02-08 | 2009-02-06 | (dihydro)pyrrolo[2,1-a]isoquinolines |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0906937A2 true BRPI0906937A2 (pt) | 2016-04-19 |
Family
ID=39516937
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0906937A BRPI0906937A2 (pt) | 2008-02-08 | 2009-02-06 | composto, composição farmacêutica, e, uso de um composto |
Country Status (27)
Country | Link |
---|---|
US (1) | US8394789B2 (pt) |
EP (1) | EP2252611B1 (pt) |
JP (1) | JP5620823B2 (pt) |
KR (1) | KR101586870B1 (pt) |
CN (1) | CN102216297B (pt) |
AR (1) | AR070345A1 (pt) |
AT (1) | ATE527260T1 (pt) |
AU (1) | AU2009211296B2 (pt) |
BR (1) | BRPI0906937A2 (pt) |
CA (1) | CA2713173C (pt) |
CL (1) | CL2009000281A1 (pt) |
CO (1) | CO6241120A2 (pt) |
DK (1) | DK2252611T3 (pt) |
EC (1) | ECSP10010303A (pt) |
ES (1) | ES2373022T3 (pt) |
HK (1) | HK1150597A1 (pt) |
HR (1) | HRP20110942T1 (pt) |
IL (1) | IL206378A0 (pt) |
MX (1) | MX2010008717A (pt) |
NZ (1) | NZ587164A (pt) |
PE (1) | PE20091413A1 (pt) |
PL (1) | PL2252611T3 (pt) |
PT (1) | PT2252611E (pt) |
RU (1) | RU2495037C2 (pt) |
SI (1) | SI2252611T1 (pt) |
TW (1) | TW200944523A (pt) |
WO (1) | WO2009098283A1 (pt) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8071587B2 (en) | 2009-05-27 | 2011-12-06 | N. V. Organon | (Dihydro)imidazoiso[5,1-A]quinolines |
TWI461426B (zh) * | 2009-05-27 | 2014-11-21 | Merck Sharp & Dohme | (二氫)咪唑並異〔5,1-a〕喹啉類 |
EP2504316A1 (en) | 2009-11-23 | 2012-10-03 | MSD Oss B.V. | Heterocylic compounds as antagonists of the orexin receptors |
US20120174381A1 (en) | 2011-01-10 | 2012-07-12 | David Messick | Apparatus and method for frame crimping |
WO2012112956A2 (en) * | 2011-02-19 | 2012-08-23 | The Broad Institute, Inc | Compounds and methods for targeting leukemic stem cells |
CA2849111C (en) | 2011-09-22 | 2019-03-26 | Merck Sharp & Dohme B.V. | Fsh receptor antagonists |
SI2796460T1 (sl) * | 2011-12-21 | 2018-10-30 | Jiangsu Hengrui Medicine Co. Ltd | Pirolni šestčlenski derivat heteroarilnega obroča, postopek priprave zanj in medicinske uporabe le-tega |
CN102718695B (zh) * | 2012-06-25 | 2014-04-02 | 华东师范大学 | 一种氮杂双环[3.3.0]辛烷衍生物的合成方法 |
RU2649004C2 (ru) | 2012-11-29 | 2018-03-29 | Кемосентрикс, Инк. | Антагонисты cxcr7 |
RU2550366C1 (ru) * | 2014-05-22 | 2015-05-10 | Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Российский университет дружбы народов" (РУДН) | СПОСОБ ПОЛУЧЕНИЯ ПРОИЗВОДНЫХ 5,6-ДИГИДРОПИРРОЛО[2,1-a]ИЗОХИНОЛИНОВ |
KR20210102338A (ko) * | 2018-12-12 | 2021-08-19 | 케모센트릭스, 인크. | 암의 치료를 위한 cxcr7 억제제 |
CN110540519B (zh) * | 2019-09-05 | 2022-12-02 | 宁波大学 | 一种1,6-烯炔类化合物与酮类化合物的自由基环化反应方法 |
CN113999103A (zh) * | 2021-11-26 | 2022-02-01 | 八叶草健康产业研究院(厦门)有限公司 | 一种α-羟基-环丁烷甲酸的制备方法 |
Family Cites Families (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8718980D0 (en) * | 1987-08-11 | 1987-09-16 | May & Baker Ltd | Compositions of matter |
DE4343649A1 (de) * | 1993-12-21 | 1995-06-22 | Boehringer Ingelheim Kg | Neue Pyridazino[4',5':3,4]pyrrolo-[2,1-a]isochinoline und deren Verwendung für die Herstellung von pharmazeutischen Zubereitungen |
FR2761358B1 (fr) * | 1997-03-27 | 1999-05-07 | Adir | Nouveaux composes de n-aryl piperidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
ATE279407T1 (de) | 1998-08-07 | 2004-10-15 | Applied Research Systems | Fsh mimetika zur behandlung von infertilität |
WO2000048144A1 (fr) | 1999-02-15 | 2000-08-17 | Medailles Souvenirs | Dispositif de personnalisation et de distribution de medailles |
WO2002009706A1 (en) | 2000-07-27 | 2002-02-07 | Smithkline Beecham Corporation | Agonists of follicle stimulating hormone activity |
EP1347973A1 (en) * | 2000-12-13 | 2003-10-01 | Bayer Aktiengesellschaft | Pyrrolo (2.1-a) dihydroisoquinolines and their use as phosphodiesterase 10a inhibitors |
KR100908468B1 (ko) | 2001-07-02 | 2009-07-21 | 엔.브이.오가논 | 테트라히드로퀴놀린 유도체 |
WO2003014115A1 (en) | 2001-08-06 | 2003-02-20 | Bayer Aktiengesellschaft | 3-substituted pyrrolo (2.1-a) isoquinoline derivatives |
US20030236276A1 (en) | 2001-08-06 | 2003-12-25 | Ulrich Niewohner | Pyrrolo[2.1-a]isoquinoline derivatives |
WO2003051877A1 (en) * | 2001-12-18 | 2003-06-26 | Bayer Corporation | 2-substituted pyrrolo[2.1-a]isoquinolines against cancer |
CA2499732A1 (en) * | 2002-09-20 | 2004-04-15 | Applied Research Systems Ars Holding N.V. | Piperazine derivatives and methods of use |
RS20050945A (en) | 2003-06-30 | 2008-06-05 | Altana Pharma Ag., | Novel pyrrolodihydroisoquinolines useful in the treatment of cancer |
EP1641457B1 (en) | 2003-06-30 | 2009-08-05 | Nycomed GmbH | Pyrrolo-dihydroisoquinoline derivatives as pde10 inhibitors |
WO2005087765A1 (en) | 2004-03-04 | 2005-09-22 | Arena Pharmaceuticals, Inc. | Ligands of follicle stimulating hormone receptor and methods of use thereof |
WO2006075012A2 (en) | 2005-01-12 | 2006-07-20 | Nycomed Gmbh | Pyrrolodihydroisoquinolines as antiproliferative agents |
US20080161338A1 (en) | 2005-01-12 | 2008-07-03 | Altana Pharma Ag | Novel Pyrrolodihydroisoquinolines as Pde 10 Inhibitors |
UA92007C2 (ru) | 2005-05-04 | 2010-09-27 | Н.В. Органон | Производные 4-фенил-5-оксо-1,4,5,6,7,8-гексагидрохинолина для лечения бесплодности |
PL1879866T3 (pl) | 2005-05-04 | 2011-07-29 | N V Organon | Pochodne dihydropirydynowe |
UA92009C2 (ru) | 2005-05-04 | 2010-09-27 | Н.В. Органон | Производные 4-фенил-5-оксо-1,4,5,6,7,8-гексагидрохинолина для лечения бесплодия |
UA92008C2 (en) | 2005-05-04 | 2010-09-27 | Н.В. Органон | 4-PHENYL-5-OXO-l,4,5,6,7,8-HEXAHYDROQUINOLINE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF INFERTILITY |
-
2009
- 2009-01-19 TW TW098101900A patent/TW200944523A/zh unknown
- 2009-02-05 PE PE2009000177A patent/PE20091413A1/es not_active Application Discontinuation
- 2009-02-06 KR KR1020107020092A patent/KR101586870B1/ko not_active IP Right Cessation
- 2009-02-06 AT AT09708584T patent/ATE527260T1/de active
- 2009-02-06 CA CA2713173A patent/CA2713173C/en not_active Expired - Fee Related
- 2009-02-06 US US12/866,468 patent/US8394789B2/en active Active
- 2009-02-06 DK DK09708584.9T patent/DK2252611T3/da active
- 2009-02-06 RU RU2010136057/04A patent/RU2495037C2/ru not_active IP Right Cessation
- 2009-02-06 BR BRPI0906937A patent/BRPI0906937A2/pt not_active IP Right Cessation
- 2009-02-06 MX MX2010008717A patent/MX2010008717A/es active IP Right Grant
- 2009-02-06 AU AU2009211296A patent/AU2009211296B2/en not_active Ceased
- 2009-02-06 PL PL09708584T patent/PL2252611T3/pl unknown
- 2009-02-06 JP JP2010545476A patent/JP5620823B2/ja not_active Expired - Fee Related
- 2009-02-06 PT PT09708584T patent/PT2252611E/pt unknown
- 2009-02-06 SI SI200930133T patent/SI2252611T1/sl unknown
- 2009-02-06 CL CL2009000281A patent/CL2009000281A1/es unknown
- 2009-02-06 EP EP09708584A patent/EP2252611B1/en active Active
- 2009-02-06 AR ARP090100410A patent/AR070345A1/es unknown
- 2009-02-06 NZ NZ587164A patent/NZ587164A/en not_active IP Right Cessation
- 2009-02-06 ES ES09708584T patent/ES2373022T3/es active Active
- 2009-02-06 CN CN200980103881.7A patent/CN102216297B/zh not_active Expired - Fee Related
- 2009-02-06 WO PCT/EP2009/051366 patent/WO2009098283A1/en active Application Filing
-
2010
- 2010-06-15 IL IL206378A patent/IL206378A0/en unknown
- 2010-06-23 EC EC2010010303A patent/ECSP10010303A/es unknown
- 2010-08-06 CO CO10096219A patent/CO6241120A2/es not_active Application Discontinuation
-
2011
- 2011-05-09 HK HK11104579.8A patent/HK1150597A1/xx not_active IP Right Cessation
- 2011-12-16 HR HR20110942T patent/HRP20110942T1/hr unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B25A | Requested transfer of rights approved |
Owner name: MSD OSS B.V. (NL) |
|
B25A | Requested transfer of rights approved |
Owner name: ORGANON BIOSCIENCES NEDERLAND B.V. (NL) |
|
B25A | Requested transfer of rights approved |
Owner name: MERCK SHARP AND DOHME B.V. (NL) |
|
B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] | ||
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 10A ANUIDADE. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2500 DE 04-12-2018 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |