BRPI0716698A2 - Composto, composição farmacêutica e uso de um composto - Google Patents

Composto, composição farmacêutica e uso de um composto

Info

Publication number
BRPI0716698A2
BRPI0716698A2 BRPI0716698-2A2A BRPI0716698A BRPI0716698A2 BR PI0716698 A2 BRPI0716698 A2 BR PI0716698A2 BR PI0716698 A BRPI0716698 A BR PI0716698A BR PI0716698 A2 BRPI0716698 A2 BR PI0716698A2
Authority
BR
Brazil
Prior art keywords
compound
pharmaceutical composition
pharmaceutical
composition
Prior art date
Application number
BRPI0716698-2A2A
Other languages
English (en)
Inventor
Kumar Sukeerthi
Balasubramanian Gopalan
Srinivas Gullapalli
Neelima Khairatkar Joshi
Shridhar Narayanan
Pallavi V Karnik
Meyyappan Muthuppalantappan
Original Assignee
Glenmark Pharmaceuticals Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39344661&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0716698(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glenmark Pharmaceuticals Sa filed Critical Glenmark Pharmaceuticals Sa
Publication of BRPI0716698A2 publication Critical patent/BRPI0716698A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
BRPI0716698-2A2A 2006-11-03 2007-11-21 Composto, composição farmacêutica e uso de um composto BRPI0716698A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN1838MU2006 2006-11-03
PCT/IB2007/003337 WO2008053341A2 (en) 2006-11-03 2007-11-02 Bridged bicyclic indazoles as cannabinoid receptor ligands

Publications (1)

Publication Number Publication Date
BRPI0716698A2 true BRPI0716698A2 (pt) 2014-02-25

Family

ID=39344661

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0716698-2A2A BRPI0716698A2 (pt) 2006-11-03 2007-11-21 Composto, composição farmacêutica e uso de um composto

Country Status (13)

Country Link
US (1) US20080200501A1 (pt)
EP (1) EP2091921A2 (pt)
JP (1) JP2010509201A (pt)
CN (1) CN101573339A (pt)
AR (1) AR063558A1 (pt)
AU (1) AU2007315848A1 (pt)
BR (1) BRPI0716698A2 (pt)
CA (1) CA2668491A1 (pt)
CL (1) CL2007003183A1 (pt)
RU (1) RU2009117203A (pt)
TW (1) TW200826933A (pt)
WO (1) WO2008053341A2 (pt)
ZA (1) ZA200903075B (pt)

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EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
CA2770866C (en) 2009-08-28 2017-10-10 Arena Pharmaceuticals, Inc. Cannabinoid receptor modulators
EP2957560B1 (en) 2010-02-08 2017-08-02 Allergan, Inc. Pyridazine derivatives useful as cannabinoid-2 agonists
US20130178453A1 (en) * 2010-02-09 2013-07-11 Ironwood Pharmaceuticals, Inc. Cannabinoid Agonists
BR112013003481A8 (pt) * 2010-07-29 2017-12-26 Astellas Pharma Inc composto fundido a anel de piridina
US9597340B2 (en) 2011-02-25 2017-03-21 Arena Pharmaceuticals, Inc. Cannabinoid receptor modulators
RU2469027C2 (ru) * 2011-02-25 2012-12-10 Государственное образовательное учреждение высшего профессионального образования "Пермский государственный университет" 3-(2-бромфенил) и 3-бензил-4,5,6,7-тетрагидроиндазола гидрохлориды, противомикробное средство на их основе
JP6043733B2 (ja) 2011-02-25 2016-12-14 アリーナ ファーマシューティカルズ， インコーポレイテッド カンナビノイド受容体モジュレーター
EP4166552A1 (en) 2011-02-25 2023-04-19 Arena Pharmaceuticals, Inc. Crystalline forms and processes for the preparation of condensed azacycles (cannabinoid receptor modulators)
CN104447499B (zh) * 2013-09-25 2016-09-21 中国科学院大连化学物理研究所 Au催化的炔基吡咯合成吡咯并七元环衍生物的方法
CN114391011A (zh) * 2019-09-12 2022-04-22 四川海思科制药有限公司 一种六氢化苯并吡唑衍生物及其制备
TW202142538A (zh) 2020-02-07 2021-11-16 美商迦舒布魯姆生物有限公司 雜環ｇｌｐ－１促效劑

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US3501471A (en) * 1966-09-21 1970-03-17 American Cyanamid Co Novel 2,3-heterocyclic fused quinuclidines,and 3-substituted quinuclidine-2-carboxylate derivatives
US3928378A (en) * 1974-01-30 1975-12-23 Hoechst Co American Fused bicyclic aminopyrazoles
WO2003057213A2 (en) * 2001-12-28 2003-07-17 Bayer Pharmaceuticals Corporation Cyclohexano- and cycloheptapyrazole derivative compounds, for use in diseases associated with the 5-ht2c receptor
DE10219294A1 (de) * 2002-04-25 2003-11-13 Schering Ag Substituierte N-(1,4,5,6-Tetrahydro-cyclopentapyrazol-3-yl)-Derivate, deren Herstellung und Verwendung als Arzneimittel
US7452997B2 (en) * 2004-03-24 2008-11-18 Janssen Pharmaceutica, N.V. Tetrahydro-indazole cannabinoid modulators
US7923465B2 (en) * 2005-06-02 2011-04-12 Glenmark Pharmaceuticals S.A. Cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation
JP2008545739A (ja) * 2005-06-02 2008-12-18 グレンマーク・ファーマシューティカルズ・エスエー 新規なカンナビノイド受容体リガンド、それらを含む薬剤組成物、およびそれらの調製方法

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AR063558A1 (es) 2009-02-04
US20080200501A1 (en) 2008-08-21
CA2668491A1 (en) 2008-05-08
RU2009117203A (ru) 2010-12-10
CL2007003183A1 (es) 2008-06-27
CN101573339A (zh) 2009-11-04
ZA200903075B (en) 2010-03-31
TW200826933A (en) 2008-07-01
AU2007315848A1 (en) 2008-05-08
WO2008053341A3 (en) 2008-10-23
JP2010509201A (ja) 2010-03-25
WO2008053341A2 (en) 2008-05-08
EP2091921A2 (en) 2009-08-26

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