BRPI0516912A2 - formulação a base do capsaicinoide em gel e usos da mesma - Google Patents
formulação a base do capsaicinoide em gel e usos da mesmaInfo
- Publication number
- BRPI0516912A2 BRPI0516912A2 BRPI0516912-7A BRPI0516912A BRPI0516912A2 BR PI0516912 A2 BRPI0516912 A2 BR PI0516912A2 BR PI0516912 A BRPI0516912 A BR PI0516912A BR PI0516912 A2 BRPI0516912 A2 BR PI0516912A2
- Authority
- BR
- Brazil
- Prior art keywords
- capsaicinoid
- gel
- gel formulation
- âμg
- human
- Prior art date
Links
- YKPUWZUDDOIDPM-SOFGYWHQSA-N capsaicin Chemical compound COC1=CC(CNC(=O)CCCC\C=C\C(C)C)=CC=C1O YKPUWZUDDOIDPM-SOFGYWHQSA-N 0.000 title abstract 6
- 238000009472 formulation Methods 0.000 title abstract 3
- 239000000203 mixture Substances 0.000 title abstract 3
- 241001465754 Metazoa Species 0.000 abstract 2
- 208000004550 Postoperative Pain Diseases 0.000 abstract 2
- 238000011477 surgical intervention Methods 0.000 abstract 2
- 229960002504 capsaicin Drugs 0.000 abstract 1
- 235000017663 capsaicin Nutrition 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K36/00—Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
- A61K36/18—Magnoliophyta (angiosperms)
- A61K36/185—Magnoliopsida (dicotyledons)
- A61K36/81—Solanaceae (Potato family), e.g. tobacco, nightshade, tomato, belladonna, capsicum or jimsonweed
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A61K9/0024—Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/06—Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
- A61P23/02—Local anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P41/00—Drugs used in surgical methods, e.g. surgery adjuvants for preventing adhesion or for vitreum substitution
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
FORMULAçãO A BASE DO CAPSAICINOIDE EM GEL E USOS DA MESMA. A presente invençâo proporciona formulações à base de capsaicinoide em gel emétodos para aliviar a dor pré e pós-cirúrgico em um local em um ser humano ou em um animal mediante a administração no lugar da intervenção cirúrgica no ser humano ou animal que o necessita de uma dose de capsaicinoide em gel em uma quantidade efetiva para atenuar a dor pós-cirúrgica no lugar da intervenção cirúrgica, a dose de capsaicina oscila de desde 100<109>g A 10.000<109>g.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US63057704P | 2004-11-24 | 2004-11-24 | |
PCT/US2005/042578 WO2006058140A2 (en) | 2004-11-24 | 2005-11-23 | Capsaicinoid gel formulation and uses thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0516912A2 true BRPI0516912A2 (pt) | 2009-06-23 |
Family
ID=36498519
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0516912-7A BRPI0516912A2 (pt) | 2004-11-24 | 2005-11-23 | formulação a base do capsaicinoide em gel e usos da mesma |
Country Status (11)
Country | Link |
---|---|
US (1) | US20060148903A1 (pt) |
EP (1) | EP1827405A2 (pt) |
JP (1) | JP2008521815A (pt) |
CN (1) | CN101119713A (pt) |
AU (1) | AU2005309586A1 (pt) |
BR (1) | BRPI0516912A2 (pt) |
CA (1) | CA2596194A1 (pt) |
EA (1) | EA200701131A1 (pt) |
IL (1) | IL183332A0 (pt) |
MX (1) | MX2007006253A (pt) |
WO (1) | WO2006058140A2 (pt) |
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JP2006513267A (ja) | 2002-12-18 | 2006-04-20 | アルゴルクス ファーマスーティカルズ,インク | カプサイシノイドの投与 |
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-
2005
- 2005-11-23 MX MX2007006253A patent/MX2007006253A/es not_active Application Discontinuation
- 2005-11-23 CN CNA2005800471530A patent/CN101119713A/zh active Pending
- 2005-11-23 US US11/286,059 patent/US20060148903A1/en not_active Abandoned
- 2005-11-23 EP EP05852112A patent/EP1827405A2/en not_active Ceased
- 2005-11-23 JP JP2007543484A patent/JP2008521815A/ja active Pending
- 2005-11-23 CA CA002596194A patent/CA2596194A1/en not_active Abandoned
- 2005-11-23 BR BRPI0516912-7A patent/BRPI0516912A2/pt not_active Application Discontinuation
- 2005-11-23 EA EA200701131A patent/EA200701131A1/ru unknown
- 2005-11-23 WO PCT/US2005/042578 patent/WO2006058140A2/en active Application Filing
- 2005-11-23 AU AU2005309586A patent/AU2005309586A1/en not_active Abandoned
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2007
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CA2596194A1 (en) | 2006-06-01 |
WO2006058140A3 (en) | 2007-01-04 |
MX2007006253A (es) | 2007-10-18 |
US20060148903A1 (en) | 2006-07-06 |
EA200701131A1 (ru) | 2007-12-28 |
IL183332A0 (en) | 2007-10-31 |
JP2008521815A (ja) | 2008-06-26 |
AU2005309586A1 (en) | 2006-06-01 |
CN101119713A (zh) | 2008-02-06 |
EP1827405A2 (en) | 2007-09-05 |
WO2006058140A2 (en) | 2006-06-01 |
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