BRPI0409517A - processo para a preparação de derivados de 2-amino metil piridina, derivados 2-nitro metil piridina e processo para a preparação de derivados de 2-nitro metil piridina - Google Patents
processo para a preparação de derivados de 2-amino metil piridina, derivados 2-nitro metil piridina e processo para a preparação de derivados de 2-nitro metil piridinaInfo
- Publication number
- BRPI0409517A BRPI0409517A BRPI0409517-0A BRPI0409517A BRPI0409517A BR PI0409517 A BRPI0409517 A BR PI0409517A BR PI0409517 A BRPI0409517 A BR PI0409517A BR PI0409517 A BRPI0409517 A BR PI0409517A
- Authority
- BR
- Brazil
- Prior art keywords
- pyridine derivatives
- methyl pyridine
- preparing
- nitro
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/36—Radicals substituted by singly-bound nitrogen atoms
- C07D213/38—Radicals substituted by singly-bound nitrogen atoms having only hydrogen or hydrocarbon radicals attached to the substituent nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/26—Radicals substituted by halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyridine Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
"PROCESSO PARA A PREPARAçãO DE DERIVADOS DE 2-AMINO METIL PIRIDINA, DERIVADOS 2-NITRO METIL PIRIDINA E PROCESSO PARA A PREPARAçãO DE DERIVADOS DE 2-NITRO METIL PIRIDINA". A presente invenção refere-se a um novo processo para a preparação de derivados de 2-amino metil piridina da fórmula (I), o qual compreende a reação, em uma primeira etapa, de derivados de piridina substituída na posição 2 da fórmula (II), com um nitroalcano da fórmula (III), na presença de uma base, resultando em derivados de 2-nitro metil piridina da fórmula (IV), e hidrogenação desses derivados de 2-nitro metil piridina da fórmula (IV) em uma segunda etapa, na presença de um catalisador e na presença de um ácido, onde nas fórmulas n, X, Y R¬ 1¬, R¬ 2¬ e A são tal como definido na descrição.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0309631.0A GB0309631D0 (en) | 2003-04-28 | 2003-04-28 | Novel process for the preparation of 2-aminomethylpyridine derivatives |
PCT/EP2004/006075 WO2004096772A1 (en) | 2003-04-28 | 2004-04-26 | Novel process for the preparation of 2-aminomethylpyridine derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0409517A true BRPI0409517A (pt) | 2006-04-18 |
Family
ID=9957269
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0409517-0A BRPI0409517A (pt) | 2003-04-28 | 2004-04-26 | processo para a preparação de derivados de 2-amino metil piridina, derivados 2-nitro metil piridina e processo para a preparação de derivados de 2-nitro metil piridina |
Country Status (15)
Country | Link |
---|---|
US (1) | US7608720B2 (pt) |
EP (1) | EP1620404B1 (pt) |
JP (1) | JP4718446B2 (pt) |
KR (2) | KR101130601B1 (pt) |
CN (1) | CN100413847C (pt) |
AT (1) | ATE356116T1 (pt) |
BR (1) | BRPI0409517A (pt) |
DE (1) | DE602004005175T2 (pt) |
DK (1) | DK1620404T3 (pt) |
ES (1) | ES2279383T3 (pt) |
GB (1) | GB0309631D0 (pt) |
IL (1) | IL170657A (pt) |
PL (1) | PL1620404T3 (pt) |
TW (1) | TWI359139B (pt) |
WO (1) | WO2004096772A1 (pt) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US9434684B2 (en) | 2012-07-12 | 2016-09-06 | Nissan Chemical Industries, Ltd. | Oxime-substituted amide compound and pest control agent |
CN106220555B (zh) * | 2016-07-29 | 2019-06-21 | 天津市均凯化工科技有限公司 | 一种制备2-氨甲基-3-氯-5-三氟甲基吡啶的方法 |
TWI650318B (zh) * | 2017-10-30 | 2019-02-11 | 財團法人工業技術研究院 | 以結晶法純化2,5-呋喃二甲酸的粗產物之方法與聚酯之形成方法 |
US11236070B2 (en) | 2019-05-16 | 2022-02-01 | Novartis Ag | Chemical process |
CN115819330A (zh) * | 2022-12-28 | 2023-03-21 | 天津均凯农业科技有限公司 | 一种连续化制备2-氨基甲基-3-氯-5-三氟甲基吡啶的方法 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3615293A1 (de) * | 1986-05-06 | 1987-11-12 | Bayer Ag | Verwendung von heteroarylethylaminen zur leistungsfoerderung bei tieren, heteroarylethylamine und verfahren zu ihrer herstellung |
ZA885069B (en) | 1987-07-24 | 1989-03-29 | Fujisawa Pharmaceutical Co | Sustained-release percutaneous preparations |
FR2649978B1 (fr) * | 1989-07-20 | 1991-10-25 | Rhone Poulenc Chimie | Procede d'hydrogenation de derives halogeno nitroaromatiques en presence d'iodures |
CA2415842A1 (en) * | 2000-08-25 | 2002-02-28 | Michael Mellor | Process for the preparation of 2-aminoethylpyridines |
DE10101647A1 (de) | 2001-01-16 | 2002-07-18 | Degussa | Verfahren zur Herstellung von substituierten Aminen durch Hydrierung von substituierten organischen Nitroverbindungen |
-
2003
- 2003-04-28 GB GBGB0309631.0A patent/GB0309631D0/en not_active Ceased
-
2004
- 2004-04-12 TW TW093110136A patent/TWI359139B/zh not_active IP Right Cessation
- 2004-04-26 DK DK04739624T patent/DK1620404T3/da active
- 2004-04-26 ES ES04739624T patent/ES2279383T3/es not_active Expired - Lifetime
- 2004-04-26 EP EP04739624A patent/EP1620404B1/en not_active Expired - Lifetime
- 2004-04-26 AT AT04739624T patent/ATE356116T1/de not_active IP Right Cessation
- 2004-04-26 US US10/554,880 patent/US7608720B2/en not_active Expired - Fee Related
- 2004-04-26 WO PCT/EP2004/006075 patent/WO2004096772A1/en active IP Right Grant
- 2004-04-26 KR KR1020057020214A patent/KR101130601B1/ko active IP Right Grant
- 2004-04-26 PL PL04739624T patent/PL1620404T3/pl unknown
- 2004-04-26 KR KR1020117027963A patent/KR101213005B1/ko active IP Right Grant
- 2004-04-26 DE DE602004005175T patent/DE602004005175T2/de not_active Expired - Lifetime
- 2004-04-26 CN CNB2004800110082A patent/CN100413847C/zh not_active Expired - Lifetime
- 2004-04-26 BR BRPI0409517-0A patent/BRPI0409517A/pt active Search and Examination
- 2004-04-26 JP JP2006505421A patent/JP4718446B2/ja not_active Expired - Lifetime
-
2005
- 2005-09-04 IL IL170657A patent/IL170657A/en active IP Right Grant
Also Published As
Publication number | Publication date |
---|---|
CN1777588A (zh) | 2006-05-24 |
CN100413847C (zh) | 2008-08-27 |
JP4718446B2 (ja) | 2011-07-06 |
US20060235229A1 (en) | 2006-10-19 |
DE602004005175T2 (de) | 2007-12-20 |
DK1620404T3 (da) | 2007-04-02 |
EP1620404B1 (en) | 2007-03-07 |
GB0309631D0 (en) | 2003-06-04 |
KR20110133063A (ko) | 2011-12-09 |
PL1620404T3 (pl) | 2007-07-31 |
EP1620404A1 (en) | 2006-02-01 |
JP2006524665A (ja) | 2006-11-02 |
IL170657A (en) | 2011-02-28 |
DE602004005175D1 (de) | 2007-04-19 |
ATE356116T1 (de) | 2007-03-15 |
ES2279383T3 (es) | 2007-08-16 |
TW200502220A (en) | 2005-01-16 |
WO2004096772A1 (en) | 2004-11-11 |
KR101213005B1 (ko) | 2012-12-18 |
KR101130601B1 (ko) | 2012-04-02 |
TWI359139B (en) | 2012-03-01 |
KR20060005396A (ko) | 2006-01-17 |
US7608720B2 (en) | 2009-10-27 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
B25A | Requested transfer of rights approved |
Owner name: BAYER CROPSCIENCE LTD. (GB) |
|
B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
B11D | Dismissal acc. art. 38, par 2 of ipl - failure to pay fee after grant in time |