BR112015020823A8 - 1-hidróxi-benzooxaboróis como agentes antiparasíticos, seus usos, e formulação". - Google Patents

1-hidróxi-benzooxaboróis como agentes antiparasíticos, seus usos, e formulação". Download PDF

Info

Publication number
BR112015020823A8
BR112015020823A8 BR112015020823A BR112015020823A BR112015020823A8 BR 112015020823 A8 BR112015020823 A8 BR 112015020823A8 BR 112015020823 A BR112015020823 A BR 112015020823A BR 112015020823 A BR112015020823 A BR 112015020823A BR 112015020823 A8 BR112015020823 A8 BR 112015020823A8
Authority
BR
Brazil
Prior art keywords
benzooxaborols
hydroxy
control
antiparasitic agents
formulation
Prior art date
Application number
BR112015020823A
Other languages
English (en)
Other versions
BR112015020823A2 (pt
Inventor
J Plattner Jacob
Jarnagin Kurt
Roland Pulley Shon
Akama Tsutomu
Hunter White William
Zhou Yasheen
Zhang Yong-Kang
Original Assignee
Anacor Pharmaceuticals Inc
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anacor Pharmaceuticals Inc, Lilly Co Eli filed Critical Anacor Pharmaceuticals Inc
Publication of BR112015020823A2 publication Critical patent/BR112015020823A2/pt
Publication of BR112015020823A8 publication Critical patent/BR112015020823A8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
    • A01N55/08—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur containing boron
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Epidemiology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Steroid Compounds (AREA)

Abstract

resumo patente de invenção: "1-hidróxi-benzooxaboróis como agentes antiparasíticos". são fornecidos compostos úteis para o controle de endoparasitas tanto em animais quanto em agricultura. são também fornecidos métodos para o controle de infestações por endoparasita de um animal administrando uma quantidade efetiva de um composto como descrito acima, ou um sal farmaceuticamente aceitável do mesmo, a um animal, bem como formulações para o controle de infestações por endoparasita, usando os compostos descritos acima ou um sal aceitável do mesmo, e um veículo aceitável. os compostos reivindicados são descritos pela seguinte fórmula markush: um exemplo típico para um composto de acordo com a fórmula acima é:
BR112015020823A 2013-03-15 2014-03-06 1-hidróxi-benzooxaboróis como agentes antiparasíticos, seus usos, e formulação". BR112015020823A8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361786839P 2013-03-15 2013-03-15
PCT/US2014/020966 WO2014149793A1 (en) 2013-03-15 2014-03-06 1 -hydroxy-benzooxaboroles as antiparasitic agents

Publications (2)

Publication Number Publication Date
BR112015020823A2 BR112015020823A2 (pt) 2017-07-18
BR112015020823A8 true BR112015020823A8 (pt) 2019-09-17

Family

ID=50382679

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015020823A BR112015020823A8 (pt) 2013-03-15 2014-03-06 1-hidróxi-benzooxaboróis como agentes antiparasíticos, seus usos, e formulação".

Country Status (24)

Country Link
US (1) US9617285B2 (pt)
EP (1) EP2970339B1 (pt)
JP (1) JP6121043B2 (pt)
KR (1) KR101727421B1 (pt)
CN (1) CN105051048B (pt)
AR (1) AR094961A1 (pt)
AU (1) AU2014237862B2 (pt)
BR (1) BR112015020823A8 (pt)
CA (1) CA2899972A1 (pt)
CY (1) CY1119473T1 (pt)
DK (1) DK2970339T3 (pt)
EA (1) EA027430B1 (pt)
ES (1) ES2645687T3 (pt)
HR (1) HRP20171517T1 (pt)
HU (1) HUE035545T2 (pt)
LT (1) LT2970339T (pt)
MX (1) MX2015013051A (pt)
NO (1) NO2904426T3 (pt)
PL (1) PL2970339T3 (pt)
PT (1) PT2970339T (pt)
RS (1) RS56532B1 (pt)
SI (1) SI2970339T1 (pt)
TW (1) TW201506031A (pt)
WO (1) WO2014149793A1 (pt)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11039617B2 (en) 2013-01-30 2021-06-22 Agrofresh Inc. Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness
US10070649B2 (en) 2013-01-30 2018-09-11 Agrofresh Inc. Volatile applications against pathogens
JP6605513B2 (ja) 2014-07-01 2019-11-13 第一三共株式会社 抗菌剤としての三環式ベンゾオキサボロール
AU2017229098B2 (en) 2016-03-07 2021-05-27 Agrofresh Inc. Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops
CA3026316A1 (en) 2016-06-03 2017-12-07 Basf Se Benzoxaborole compounds
WO2018156554A1 (en) * 2017-02-21 2018-08-30 Dow Agrosciences Llc 1-HYDROXY-1,3-DIHYDROBENZO[c][1,2]OXABOROLES AND THEIR USE AS HERBICIDES
CN108864160A (zh) * 2017-05-16 2018-11-23 苏州旺山旺水生物医药有限公司 含硼小分子的制备方法
WO2019025250A1 (en) 2017-08-04 2019-02-07 Basf Se SUBSTITUTED TRIFLUOROMETHYLOXADIAZOLES FOR COMBATING PHYTOPATHOGENIC FUNGI
BR112020010927A2 (pt) 2017-11-30 2020-12-01 Boragen, Inc. compostos de benzoxaborol e formulações dos mesmos
JP2021534247A (ja) 2018-08-18 2021-12-09 ボラゲン，インコーポレーテッド 置換ベンゾキサボロールの固体形態およびその組成物
US20230340530A1 (en) 2020-08-31 2023-10-26 Pfizer Inc. Methods of Protecting RNA
CN112321510A (zh) * 2020-10-27 2021-02-05 无锡双启科技有限公司 一种4-溴-5-甲基-1h-吲唑的制备方法
CN112745270B (zh) * 2020-12-30 2023-02-24 河北医科大学 新化合物及其制备苯唑草酮中间体的方法
EP4137485A1 (en) * 2021-08-20 2023-02-22 Henkel AG & Co. KGaA Vinyl ethers

Family Cites Families (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6239077B1 (en) 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
DE60126838T2 (de) 2000-12-20 2007-11-08 Novartis Ag Amidoacetonitrile zur Bekämpfung von Endoparasiten
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
TWI236341B (en) 2001-06-15 2005-07-21 Novartis Ag Aminoacetonitrile compounds for use in the control of endoparasites
AR038156A1 (es) 2002-01-21 2004-12-29 Novartis Ag Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica
TW200305556A (en) 2002-03-21 2003-11-01 Novartis Ag Organic compounds
AR040229A1 (es) 2002-05-22 2005-03-23 Novartis Ag Amidoacetonitrilos
AR040082A1 (es) 2002-05-22 2005-03-16 Novartis Ag Derivados de n-acilaminoacetonitrilo y su uso para el control de parasitos
AR039961A1 (es) 2002-06-06 2005-03-09 Novartis Ag Derivados de amidoacetonitrilo y su uso como pesticida
TW200400932A (en) 2002-06-19 2004-01-16 Novartis Ag Organic compounds
GB0402677D0 (en) 2003-11-06 2004-03-10 Novartis Ag Organic compounds
AR046757A1 (es) 2003-12-10 2005-12-21 Novartis Ag Amidoacetonitrilos utiles como pesticidas
TW200613251A (en) 2004-06-10 2006-05-01 Novartis Ag Organic compounds
KR101337045B1 (ko) * 2005-02-16 2013-12-05 아나코르 파마슈티칼스 인코포레이티드 보론함유 소분자
JP2009502834A (ja) 2005-07-25 2009-01-29 ノバルティス アクチエンゲゼルシャフト アミドニトリル化合物
EP1976536A4 (en) 2005-12-30 2011-03-02 Anacor Pharmaceuticals Inc SMALL MOLECULES CONTAINING BORON
WO2008102232A1 (en) 2007-02-21 2008-08-28 Pfizer Limited Benzofuran antiparasitic agents
US20100026457A1 (en) * 2008-08-04 2010-02-04 Cooper Technologies Company Location of Tagged Boxes
EA026649B1 (ru) 2008-10-21 2017-05-31 Мериал, Инк. Тиоамидные соединения, способ их получения и способ их применения
AU2010281439A1 (en) 2009-07-28 2012-03-15 Anacor Pharmaceuticals, Inc. Trisubstituted boron-containing molecules
WO2011019612A1 (en) * 2009-08-14 2011-02-17 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
EP2314292A1 (en) 2009-10-20 2011-04-27 Novartis AG Endoparasiticidal compositions
WO2011049971A1 (en) * 2009-10-20 2011-04-28 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
UY32992A (es) 2009-11-23 2011-04-29 Novartis Ag Compuestos orgánicos
AP2016009046A0 (en) * 2013-08-09 2016-02-29 Anacor Pharmaceuticals Inc Tricyclic benzoxaborole compounds and uses thereof

Also Published As

Publication number Publication date
PL2970339T3 (pl) 2018-01-31
CN105051048A (zh) 2015-11-11
EA201591512A9 (ru) 2016-04-29
NO2904426T3 (pt) 2018-02-10
CA2899972A1 (en) 2014-09-25
JP2016516032A (ja) 2016-06-02
LT2970339T (lt) 2017-11-10
AU2014237862B2 (en) 2017-01-12
EP2970339B1 (en) 2017-08-16
BR112015020823A2 (pt) 2017-07-18
HUE035545T2 (en) 2018-05-28
RS56532B1 (sr) 2018-02-28
US9617285B2 (en) 2017-04-11
EA027430B1 (ru) 2017-07-31
ES2645687T3 (es) 2017-12-07
KR20150119154A (ko) 2015-10-23
US20150353581A1 (en) 2015-12-10
EA201591512A1 (ru) 2016-01-29
SI2970339T1 (sl) 2017-10-30
TW201506031A (zh) 2015-02-16
JP6121043B2 (ja) 2017-04-26
AU2014237862A1 (en) 2015-08-13
HRP20171517T1 (hr) 2017-11-17
PT2970339T (pt) 2017-11-14
MX2015013051A (es) 2016-05-05
KR101727421B1 (ko) 2017-04-14
CY1119473T1 (el) 2018-03-07
EP2970339A1 (en) 2016-01-20
DK2970339T3 (en) 2017-10-02
AR094961A1 (es) 2015-09-09
CN105051048B (zh) 2017-03-15
WO2014149793A1 (en) 2014-09-25

Similar Documents

Publication Publication Date Title
BR112015020823A8 (pt) 1-hidróxi-benzooxaboróis como agentes antiparasíticos, seus usos, e formulação".
BR112013028132A2 (pt) compostos de di-hidroxisoxazol parasiticida
BR112015020787A2 (pt) inibidores quinazolínicos de formas mutantes ativantes do receptor do fator de crescimento epidérmico
CY1119170T1 (el) Ενωση γουανιδινης
BR112015024078A2 (pt) derivados de benzimidazolona como inibidores de bromodomínio
CA2918938C (en) Substituted aminopyrimidine compounds and methods of use
BR112015016001A2 (pt) compostos, composições farmacêuticas e respectivos usos e método para tratar ou prevenir infecção bacteriana
BR112015018738A8 (pt) compostos de tetra-hidropirrolotiazina, seus usos, e composição farmacêutica
BR112015029512A8 (pt) derivados de pirazolopirrolidina, seus usos, e composição e combinação farmacêuticas
BR112015021983A2 (pt) compostos heterocíclicos e usos dos mesmos
BR112015023412A8 (pt) 3-pirimidin-4-il-oxazolidin-2-onas como inibidores de idh mutante, sua composição farmacêutica e seu uso.
HRP20191523T1 (hr) Paraziticidne kombinacije spirocikličkog izoksazolina
BR112016003348A2 (pt) composto ou sal farmaceuticamente aceitável do mesmo, composição farmacêutica e usos de quantidade efetiva de composto ou sal farmaceuticamente aceitável do mesmo ou composição farmacêutica
EA201590371A1 (ru) 1,4-дизамещенные аналоги пиридазина и способы лечения связанных с дефицитом smn состояний
EA201490647A1 (ru) Производные бензотиазол-6-илуксусной кислоты и их применение для лечения вич-инфекции
EA201591727A1 (ru) Соединения биариламида в качестве ингибиторов киназы
BR112015001419A8 (pt) composto, composição farmacêutica, e, uso de um composto ou de um sal farmaceuticamente aceitável do mesmo
EA201291348A1 (ru) Активаторы растворимой гуанилатциклазы
BR112015029401A8 (pt) derivados de pirazolo-pirrolidin-4-ona, seus usos, e composição e combinação farmacêuticas
DOP2013000243A (es) Inhibidores sustituidos de acetil-coa carboxilasa
MX2013011086A (es) (aralquilamino y heteroarilalquilamino alfa-sustituidos)pirimidini lo y 1,3,5-triazinilbenzimidazoles, composiciones farmacéuticas que los contienen, y estos compuestos para su uso en el tratamiento de enfermedades proliferativas.
DOP2015000169A (es) Compuestos tetracíclicos sustituidos con heterociclo y usos de los mismos para el tratamiento de enfermedades víricas
EA201491525A1 (ru) Спиро[2.4]гептаны для лечения инфекций, вызванных flaviviridae
BR112015004523A2 (pt) compostos de tetraciclina
BR112014031752A2 (pt) composição herbicida tendo atividade herbicida melhorada

Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according art. 34 industrial property law
B07D Technical examination (opinion) related to article 229 of industrial property law

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B08F Application fees: dismissal - article 86 of industrial property law

Free format text: REFERENTE A 6A ANUIDADE.

B08K Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87)

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2556 DE 31/12/2019.

B07E Notice of approval relating to section 229 industrial property law