MX2015013051A - 1-hidroxi-benzooxaboroles como agentes antiparasitarios. - Google Patents
1-hidroxi-benzooxaboroles como agentes antiparasitarios.Info
- Publication number
- MX2015013051A MX2015013051A MX2015013051A MX2015013051A MX2015013051A MX 2015013051 A MX2015013051 A MX 2015013051A MX 2015013051 A MX2015013051 A MX 2015013051A MX 2015013051 A MX2015013051 A MX 2015013051A MX 2015013051 A MX2015013051 A MX 2015013051A
- Authority
- MX
- Mexico
- Prior art keywords
- benzooxaboroles
- hydroxy
- compounds
- controlling
- antiparasitic agents
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
- A01N55/08—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur containing boron
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Abstract
Se proporcionan compuestos útiles para controlar endoparásitos tanto en animales como en agricultura. Además se proporcionan métodos para controlar infestaciones de endoparásitos de un animal al administrar una cantidad efectiva de un compuesto como se describe antes, o una sal farmacéuticamente aceptable del mismo, a un animal, así como formulaciones para controlar infestaciones de endoparásitos que usa los compuestos descritos antes o una sal aceptable de los mismos, y un portador aceptable. Los compuestos reclamados son descritos mediante la siguiente fórmula de Markush: Un ejemplo típico de un compuesto de acuerdo con la fórmula anterior es: Un ejemplo típico para un compuesto de acuerdo con la fórmula anterior es: (véase formula).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201361786839P | 2013-03-15 | 2013-03-15 | |
PCT/US2014/020966 WO2014149793A1 (en) | 2013-03-15 | 2014-03-06 | 1 -hydroxy-benzooxaboroles as antiparasitic agents |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2015013051A true MX2015013051A (es) | 2016-05-05 |
Family
ID=50382679
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2015013051A MX2015013051A (es) | 2013-03-15 | 2014-03-06 | 1-hidroxi-benzooxaboroles como agentes antiparasitarios. |
Country Status (24)
Country | Link |
---|---|
US (1) | US9617285B2 (es) |
EP (1) | EP2970339B1 (es) |
JP (1) | JP6121043B2 (es) |
KR (1) | KR101727421B1 (es) |
CN (1) | CN105051048B (es) |
AR (1) | AR094961A1 (es) |
AU (1) | AU2014237862B2 (es) |
BR (1) | BR112015020823A8 (es) |
CA (1) | CA2899972A1 (es) |
CY (1) | CY1119473T1 (es) |
DK (1) | DK2970339T3 (es) |
EA (1) | EA027430B1 (es) |
ES (1) | ES2645687T3 (es) |
HR (1) | HRP20171517T1 (es) |
HU (1) | HUE035545T2 (es) |
LT (1) | LT2970339T (es) |
MX (1) | MX2015013051A (es) |
NO (1) | NO2904426T3 (es) |
PL (1) | PL2970339T3 (es) |
PT (1) | PT2970339T (es) |
RS (1) | RS56532B1 (es) |
SI (1) | SI2970339T1 (es) |
TW (1) | TW201506031A (es) |
WO (1) | WO2014149793A1 (es) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US10070649B2 (en) | 2013-01-30 | 2018-09-11 | Agrofresh Inc. | Volatile applications against pathogens |
US11039617B2 (en) | 2013-01-30 | 2021-06-22 | Agrofresh Inc. | Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness |
JP6605513B2 (ja) | 2014-07-01 | 2019-11-13 | 第一三共株式会社 | 抗菌剤としての三環式ベンゾオキサボロール |
CA3015662A1 (en) | 2016-03-07 | 2017-09-14 | Agrofresh Inc. | Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops |
EA201892639A1 (ru) | 2016-06-03 | 2019-06-28 | Басф Се | Соединения бензоксаборола |
WO2018156554A1 (en) * | 2017-02-21 | 2018-08-30 | Dow Agrosciences Llc | 1-HYDROXY-1,3-DIHYDROBENZO[c][1,2]OXABOROLES AND THEIR USE AS HERBICIDES |
CN108864160A (zh) * | 2017-05-16 | 2018-11-23 | 苏州旺山旺水生物医药有限公司 | 含硼小分子的制备方法 |
WO2019025250A1 (en) | 2017-08-04 | 2019-02-07 | Basf Se | SUBSTITUTED TRIFLUOROMETHYLOXADIAZOLES FOR COMBATING PHYTOPATHOGENIC FUNGI |
WO2019108982A1 (en) | 2017-11-30 | 2019-06-06 | Boragen, Inc. | Benzoxaborole compounds and formulations thereof |
EP3836938A4 (en) | 2018-08-18 | 2022-05-11 | Boragen, Inc. | SOLID FORMS OF SUBSTITUTED BENZOXAZOLE AND COMPOSITIONS THEREOF |
US20230340530A1 (en) | 2020-08-31 | 2023-10-26 | Pfizer Inc. | Methods of Protecting RNA |
CN112321510A (zh) * | 2020-10-27 | 2021-02-05 | 无锡双启科技有限公司 | 一种4-溴-5-甲基-1h-吲唑的制备方法 |
CN112745270B (zh) * | 2020-12-30 | 2023-02-24 | 河北医科大学 | 新化合物及其制备苯唑草酮中间体的方法 |
EP4137485A1 (en) * | 2021-08-20 | 2023-02-22 | Henkel AG & Co. KGaA | Vinyl ethers |
Family Cites Families (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6239077B1 (en) | 1998-05-01 | 2001-05-29 | Nihon Nohyaku Co., Ltd. | Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof |
EP1392281B1 (en) | 2000-12-20 | 2007-02-21 | Novartis AG | Anti-endoparasitic amidoacetonitrils |
AR035531A1 (es) | 2001-01-22 | 2004-06-02 | Novartis Ag | Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos |
TWI236341B (en) | 2001-06-15 | 2005-07-21 | Novartis Ag | Aminoacetonitrile compounds for use in the control of endoparasites |
AR038156A1 (es) | 2002-01-21 | 2004-12-29 | Novartis Ag | Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica |
TW200305556A (en) | 2002-03-21 | 2003-11-01 | Novartis Ag | Organic compounds |
TW200400004A (en) | 2002-05-22 | 2004-01-01 | Novartis Ag | Organic compounds |
TW200400931A (en) | 2002-05-22 | 2004-01-16 | Novartis Ag | Organic compounds |
AR039961A1 (es) | 2002-06-06 | 2005-03-09 | Novartis Ag | Derivados de amidoacetonitrilo y su uso como pesticida |
TW200400932A (en) | 2002-06-19 | 2004-01-16 | Novartis Ag | Organic compounds |
GB0402677D0 (en) | 2003-11-06 | 2004-03-10 | Novartis Ag | Organic compounds |
AR046757A1 (es) | 2003-12-10 | 2005-12-21 | Novartis Ag | Amidoacetonitrilos utiles como pesticidas |
AR049391A1 (es) | 2004-06-10 | 2006-07-26 | Novartis Ag | Derivados de aminoacetonitrilo y su uso para controlar parasitos en animales de sangre caliente |
JP5038912B2 (ja) * | 2005-02-16 | 2012-10-03 | アナコール ファーマシューティカルズ,インコーポレイテッド | ホウ素含有小分子 |
AU2006278867A1 (en) | 2005-07-25 | 2007-02-15 | Novartis Ag | Amidonitrile compounds |
CN106008583A (zh) | 2005-12-30 | 2016-10-12 | 安纳考尔医药公司 | 含硼的小分子 |
BRPI0807354A2 (pt) | 2007-02-21 | 2014-05-06 | Pfizer Ltd | Agentes antiparasíticos |
US20100026457A1 (en) * | 2008-08-04 | 2010-02-04 | Cooper Technologies Company | Location of Tagged Boxes |
US7964621B2 (en) | 2008-10-21 | 2011-06-21 | Merial Limited | Thioamide compounds, method of making and method of using thereof |
BR112012001987A2 (pt) * | 2009-07-28 | 2015-09-01 | Anacor Pharmaceuticals Inc | Composto, combinação, formulação farmacêutica, uso de um composto, uma combinação ou um sal farmaceuticamente aceitável dos mesmos, e, métodos para tratar uma infecção bacteriana, para matar ou inibir o crescimento de uma bactéria, e para inibir uma beta-lactamase. |
WO2011019612A1 (en) | 2009-08-14 | 2011-02-17 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
WO2011049971A1 (en) * | 2009-10-20 | 2011-04-28 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
EP2314292A1 (en) | 2009-10-20 | 2011-04-27 | Novartis AG | Endoparasiticidal compositions |
UY32992A (es) | 2009-11-23 | 2011-04-29 | Novartis Ag | Compuestos orgánicos |
KR102093783B1 (ko) * | 2013-08-09 | 2020-03-26 | 글락소스미스클라인 인털렉츄얼 프로퍼티 (넘버 2) 리미티드 | 트리시클릭 벤족사보롤 화합물 및 이의 용도 |
-
2014
- 2014-02-28 AR ARP140100676A patent/AR094961A1/es unknown
- 2014-03-06 TW TW103107747A patent/TW201506031A/zh unknown
- 2014-03-06 AU AU2014237862A patent/AU2014237862B2/en not_active Ceased
- 2014-03-06 WO PCT/US2014/020966 patent/WO2014149793A1/en active Application Filing
- 2014-03-06 CN CN201480014758.9A patent/CN105051048B/zh not_active Expired - Fee Related
- 2014-03-06 PL PL14712939T patent/PL2970339T3/pl unknown
- 2014-03-06 CA CA2899972A patent/CA2899972A1/en not_active Abandoned
- 2014-03-06 RS RS20171064A patent/RS56532B1/sr unknown
- 2014-03-06 PT PT147129399T patent/PT2970339T/pt unknown
- 2014-03-06 EP EP14712939.9A patent/EP2970339B1/en active Active
- 2014-03-06 SI SI201430345T patent/SI2970339T1/sl unknown
- 2014-03-06 US US14/760,208 patent/US9617285B2/en not_active Expired - Fee Related
- 2014-03-06 BR BR112015020823A patent/BR112015020823A8/pt active Search and Examination
- 2014-03-06 JP JP2016500695A patent/JP6121043B2/ja active Active
- 2014-03-06 HU HUE14712939A patent/HUE035545T2/en unknown
- 2014-03-06 MX MX2015013051A patent/MX2015013051A/es unknown
- 2014-03-06 LT LTEP14712939.9T patent/LT2970339T/lt unknown
- 2014-03-06 DK DK14712939.9T patent/DK2970339T3/en active
- 2014-03-06 KR KR1020157024782A patent/KR101727421B1/ko active IP Right Grant
- 2014-03-06 ES ES14712939.9T patent/ES2645687T3/es active Active
- 2014-03-06 EA EA201591512A patent/EA027430B1/ru not_active IP Right Cessation
- 2014-11-18 NO NO14799476A patent/NO2904426T3/no unknown
-
2017
- 2017-10-09 HR HRP20171517TT patent/HRP20171517T1/hr unknown
- 2017-10-20 CY CY20171101096T patent/CY1119473T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
ES2645687T3 (es) | 2017-12-07 |
KR20150119154A (ko) | 2015-10-23 |
US20150353581A1 (en) | 2015-12-10 |
JP2016516032A (ja) | 2016-06-02 |
EP2970339A1 (en) | 2016-01-20 |
HUE035545T2 (en) | 2018-05-28 |
SI2970339T1 (sl) | 2017-10-30 |
EA027430B1 (ru) | 2017-07-31 |
DK2970339T3 (en) | 2017-10-02 |
AU2014237862A1 (en) | 2015-08-13 |
PL2970339T3 (pl) | 2018-01-31 |
CA2899972A1 (en) | 2014-09-25 |
NO2904426T3 (es) | 2018-02-10 |
TW201506031A (zh) | 2015-02-16 |
WO2014149793A1 (en) | 2014-09-25 |
AU2014237862B2 (en) | 2017-01-12 |
JP6121043B2 (ja) | 2017-04-26 |
CN105051048A (zh) | 2015-11-11 |
US9617285B2 (en) | 2017-04-11 |
BR112015020823A8 (pt) | 2019-09-17 |
EP2970339B1 (en) | 2017-08-16 |
CY1119473T1 (el) | 2018-03-07 |
EA201591512A1 (ru) | 2016-01-29 |
LT2970339T (lt) | 2017-11-10 |
HRP20171517T1 (hr) | 2017-11-17 |
KR101727421B1 (ko) | 2017-04-14 |
RS56532B1 (sr) | 2018-02-28 |
AR094961A1 (es) | 2015-09-09 |
CN105051048B (zh) | 2017-03-15 |
EA201591512A9 (ru) | 2016-04-29 |
BR112015020823A2 (pt) | 2017-07-18 |
PT2970339T (pt) | 2017-11-14 |
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