MX2015013051A - 1-hidroxi-benzooxaboroles como agentes antiparasitarios. - Google Patents

1-hidroxi-benzooxaboroles como agentes antiparasitarios.

Info

Publication number
MX2015013051A
MX2015013051A MX2015013051A MX2015013051A MX2015013051A MX 2015013051 A MX2015013051 A MX 2015013051A MX 2015013051 A MX2015013051 A MX 2015013051A MX 2015013051 A MX2015013051 A MX 2015013051A MX 2015013051 A MX2015013051 A MX 2015013051A
Authority
MX
Mexico
Prior art keywords
benzooxaboroles
hydroxy
compounds
controlling
antiparasitic agents
Prior art date
Application number
MX2015013051A
Other languages
English (en)
Inventor
Jacob J Plattner
William Hunter White
Yong-Kang Zhang
Tsutomu Akama
Kurt Jarnagin
Shon Roland Pulley
Yasheen Zhou
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of MX2015013051A publication Critical patent/MX2015013051A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N55/00Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
    • A01N55/08Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur containing boron
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics

Abstract

Se proporcionan compuestos útiles para controlar endoparásitos tanto en animales como en agricultura. Además se proporcionan métodos para controlar infestaciones de endoparásitos de un animal al administrar una cantidad efectiva de un compuesto como se describe antes, o una sal farmacéuticamente aceptable del mismo, a un animal, así como formulaciones para controlar infestaciones de endoparásitos que usa los compuestos descritos antes o una sal aceptable de los mismos, y un portador aceptable. Los compuestos reclamados son descritos mediante la siguiente fórmula de Markush: Un ejemplo típico de un compuesto de acuerdo con la fórmula anterior es: Un ejemplo típico para un compuesto de acuerdo con la fórmula anterior es: (véase formula).
MX2015013051A 2013-03-15 2014-03-06 1-hidroxi-benzooxaboroles como agentes antiparasitarios. MX2015013051A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361786839P 2013-03-15 2013-03-15
PCT/US2014/020966 WO2014149793A1 (en) 2013-03-15 2014-03-06 1 -hydroxy-benzooxaboroles as antiparasitic agents

Publications (1)

Publication Number Publication Date
MX2015013051A true MX2015013051A (es) 2016-05-05

Family

ID=50382679

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2015013051A MX2015013051A (es) 2013-03-15 2014-03-06 1-hidroxi-benzooxaboroles como agentes antiparasitarios.

Country Status (24)

Country Link
US (1) US9617285B2 (es)
EP (1) EP2970339B1 (es)
JP (1) JP6121043B2 (es)
KR (1) KR101727421B1 (es)
CN (1) CN105051048B (es)
AR (1) AR094961A1 (es)
AU (1) AU2014237862B2 (es)
BR (1) BR112015020823A8 (es)
CA (1) CA2899972A1 (es)
CY (1) CY1119473T1 (es)
DK (1) DK2970339T3 (es)
EA (1) EA027430B1 (es)
ES (1) ES2645687T3 (es)
HR (1) HRP20171517T1 (es)
HU (1) HUE035545T2 (es)
LT (1) LT2970339T (es)
MX (1) MX2015013051A (es)
NO (1) NO2904426T3 (es)
PL (1) PL2970339T3 (es)
PT (1) PT2970339T (es)
RS (1) RS56532B1 (es)
SI (1) SI2970339T1 (es)
TW (1) TW201506031A (es)
WO (1) WO2014149793A1 (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10070649B2 (en) 2013-01-30 2018-09-11 Agrofresh Inc. Volatile applications against pathogens
US11039617B2 (en) 2013-01-30 2021-06-22 Agrofresh Inc. Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness
JP6605513B2 (ja) 2014-07-01 2019-11-13 第一三共株式会社 抗菌剤としての三環式ベンゾオキサボロール
CA3015662A1 (en) 2016-03-07 2017-09-14 Agrofresh Inc. Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops
EA201892639A1 (ru) 2016-06-03 2019-06-28 Басф Се Соединения бензоксаборола
WO2018156554A1 (en) * 2017-02-21 2018-08-30 Dow Agrosciences Llc 1-HYDROXY-1,3-DIHYDROBENZO[c][1,2]OXABOROLES AND THEIR USE AS HERBICIDES
CN108864160A (zh) * 2017-05-16 2018-11-23 苏州旺山旺水生物医药有限公司 含硼小分子的制备方法
WO2019025250A1 (en) 2017-08-04 2019-02-07 Basf Se SUBSTITUTED TRIFLUOROMETHYLOXADIAZOLES FOR COMBATING PHYTOPATHOGENIC FUNGI
WO2019108982A1 (en) 2017-11-30 2019-06-06 Boragen, Inc. Benzoxaborole compounds and formulations thereof
EP3836938A4 (en) 2018-08-18 2022-05-11 Boragen, Inc. SOLID FORMS OF SUBSTITUTED BENZOXAZOLE AND COMPOSITIONS THEREOF
US20230340530A1 (en) 2020-08-31 2023-10-26 Pfizer Inc. Methods of Protecting RNA
CN112321510A (zh) * 2020-10-27 2021-02-05 无锡双启科技有限公司 一种4-溴-5-甲基-1h-吲唑的制备方法
CN112745270B (zh) * 2020-12-30 2023-02-24 河北医科大学 新化合物及其制备苯唑草酮中间体的方法
EP4137485A1 (en) * 2021-08-20 2023-02-22 Henkel AG & Co. KGaA Vinyl ethers

Family Cites Families (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6239077B1 (en) 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
EP1392281B1 (en) 2000-12-20 2007-02-21 Novartis AG Anti-endoparasitic amidoacetonitrils
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
TWI236341B (en) 2001-06-15 2005-07-21 Novartis Ag Aminoacetonitrile compounds for use in the control of endoparasites
AR038156A1 (es) 2002-01-21 2004-12-29 Novartis Ag Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica
TW200305556A (en) 2002-03-21 2003-11-01 Novartis Ag Organic compounds
TW200400004A (en) 2002-05-22 2004-01-01 Novartis Ag Organic compounds
TW200400931A (en) 2002-05-22 2004-01-16 Novartis Ag Organic compounds
AR039961A1 (es) 2002-06-06 2005-03-09 Novartis Ag Derivados de amidoacetonitrilo y su uso como pesticida
TW200400932A (en) 2002-06-19 2004-01-16 Novartis Ag Organic compounds
GB0402677D0 (en) 2003-11-06 2004-03-10 Novartis Ag Organic compounds
AR046757A1 (es) 2003-12-10 2005-12-21 Novartis Ag Amidoacetonitrilos utiles como pesticidas
AR049391A1 (es) 2004-06-10 2006-07-26 Novartis Ag Derivados de aminoacetonitrilo y su uso para controlar parasitos en animales de sangre caliente
JP5038912B2 (ja) * 2005-02-16 2012-10-03 アナコール ファーマシューティカルズ,インコーポレイテッド ホウ素含有小分子
AU2006278867A1 (en) 2005-07-25 2007-02-15 Novartis Ag Amidonitrile compounds
CN106008583A (zh) 2005-12-30 2016-10-12 安纳考尔医药公司 含硼的小分子
BRPI0807354A2 (pt) 2007-02-21 2014-05-06 Pfizer Ltd Agentes antiparasíticos
US20100026457A1 (en) * 2008-08-04 2010-02-04 Cooper Technologies Company Location of Tagged Boxes
US7964621B2 (en) 2008-10-21 2011-06-21 Merial Limited Thioamide compounds, method of making and method of using thereof
BR112012001987A2 (pt) * 2009-07-28 2015-09-01 Anacor Pharmaceuticals Inc Composto, combinação, formulação farmacêutica, uso de um composto, uma combinação ou um sal farmaceuticamente aceitável dos mesmos, e, métodos para tratar uma infecção bacteriana, para matar ou inibir o crescimento de uma bactéria, e para inibir uma beta-lactamase.
WO2011019612A1 (en) 2009-08-14 2011-02-17 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
WO2011049971A1 (en) * 2009-10-20 2011-04-28 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
EP2314292A1 (en) 2009-10-20 2011-04-27 Novartis AG Endoparasiticidal compositions
UY32992A (es) 2009-11-23 2011-04-29 Novartis Ag Compuestos orgánicos
KR102093783B1 (ko) * 2013-08-09 2020-03-26 글락소스미스클라인 인털렉츄얼 프로퍼티 (넘버 2) 리미티드 트리시클릭 벤족사보롤 화합물 및 이의 용도

Also Published As

Publication number Publication date
ES2645687T3 (es) 2017-12-07
KR20150119154A (ko) 2015-10-23
US20150353581A1 (en) 2015-12-10
JP2016516032A (ja) 2016-06-02
EP2970339A1 (en) 2016-01-20
HUE035545T2 (en) 2018-05-28
SI2970339T1 (sl) 2017-10-30
EA027430B1 (ru) 2017-07-31
DK2970339T3 (en) 2017-10-02
AU2014237862A1 (en) 2015-08-13
PL2970339T3 (pl) 2018-01-31
CA2899972A1 (en) 2014-09-25
NO2904426T3 (es) 2018-02-10
TW201506031A (zh) 2015-02-16
WO2014149793A1 (en) 2014-09-25
AU2014237862B2 (en) 2017-01-12
JP6121043B2 (ja) 2017-04-26
CN105051048A (zh) 2015-11-11
US9617285B2 (en) 2017-04-11
BR112015020823A8 (pt) 2019-09-17
EP2970339B1 (en) 2017-08-16
CY1119473T1 (el) 2018-03-07
EA201591512A1 (ru) 2016-01-29
LT2970339T (lt) 2017-11-10
HRP20171517T1 (hr) 2017-11-17
KR101727421B1 (ko) 2017-04-14
RS56532B1 (sr) 2018-02-28
AR094961A1 (es) 2015-09-09
CN105051048B (zh) 2017-03-15
EA201591512A9 (ru) 2016-04-29
BR112015020823A2 (pt) 2017-07-18
PT2970339T (pt) 2017-11-14

Similar Documents

Publication Publication Date Title
MX2015013051A (es) 1-hidroxi-benzooxaboroles como agentes antiparasitarios.
MX341739B (es) Compuestos de dihidroisoxazol parasiticidas.
MX363127B (es) Derivados de benzotiofeno como inhibidores del receptor de estrogeno.
GEP20207105B (en) 1,1,1-trifluoro-3-hydroxypropan-2-yl carbamate derivatives and 1,1,1-trifluoro-4-hydroxybutan-2yl carbamate derivatives as magl inhibitors
TN2017000204A1 (en) Triazolopyrimidine compounds and uses thereof
NZ736709A (en) Benzimidazole and imidazopyridine carboximidamide compounds having activity as inhibitors of indoleamine 2,3-dioxygenase
EA201690752A1 (ru) Ингибиторы g12c kras
MX2016006336A (es) Compuestos pirazolopirimidina.
MX2013011551A (es) Compuestos y derivados hetero - biciclicos n - sustituidos para combatir las pestes en animales.
EA033168B1 (ru) СТИМУЛЯТОРЫ sGC
NZ716840A (en) Combination formulation of two antiviral compounds
MX2014011829A (es) Compuestos de piridinilideno n-sustituidos y derivados para combatir plagas de animales.
EA201491362A1 (ru) Анестезирующие соединения и способы их применения
EA201390884A1 (ru) Азабензимидазолы в качестве противовирусных средств в отношении респираторного синцитиального вируса
MX2020007023A (es) Analogos detiadiazol y metodos para el tratamiento de afecciones relacionadas con la deficiencia del gen de supervivencia de las neuronas motoras (smn).
MX345238B (es) (aralquilamino y heteroarilalquilamino alfa-substituidos)pirimidin ilo y 1,3,5-triazinilbenzimidazoles, composiciones farmacéuticas que los contienen, y estos compuestos para su uso en el tratamiento de enfermedades proliferativas.
MY162167A (en) Substituted acetyl-coa carboxylase inhibitors
PH12015502802A1 (en) Formulation comprising a hypolipidemic agent
MX2015003594A (es) Agente terapeutico o profilactico para sindrome de lisis tumoral.
MX2014011752A (es) Compuestos heterobiciclicos n-sustituidos y derivados para combatir plagas de animales ii.
EA201491525A1 (ru) Спиро[2.4]гептаны для лечения инфекций, вызванных flaviviridae
MX364400B (es) Compuestos de tetraciclina.
MX348979B (es) Agente de control de enfermedades de las plantas.
EP2585446A4 (en) COMPOUNDS WITH ANTAGONISTIC EFFECT AGAINST TRPV1 AND THEIR USE
MX2015007116A (es) Nuevos derivados de 1,4-ditiina sustituida y su uso como fungicidas.